HK1120803A1 - Pyrazolo - Google Patents

Pyrazolo

Info

Publication number
HK1120803A1
HK1120803A1 HK09100008.1A HK09100008A HK1120803A1 HK 1120803 A1 HK1120803 A1 HK 1120803A1 HK 09100008 A HK09100008 A HK 09100008A HK 1120803 A1 HK1120803 A1 HK 1120803A1
Authority
HK
Hong Kong
Prior art keywords
pyrazolo
Prior art date
Application number
HK09100008.1A
Other languages
English (en)
Inventor
Michael Brent Tollefson
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of HK1120803A1 publication Critical patent/HK1120803A1/xx

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
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  • Cardiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Urology & Nephrology (AREA)
  • Reproductive Health (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Gynecology & Obstetrics (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Psychology (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Pregnancy & Childbirth (AREA)
  • Child & Adolescent Psychology (AREA)
HK09100008.1A 2005-11-10 2009-01-02 Pyrazolo HK1120803A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US73532005P 2005-11-10 2005-11-10
PCT/IB2006/003132 WO2007054778A1 (en) 2005-11-10 2006-10-31 Pyrazolo[4,3-d]pyrimidin-5-yl)derivative used as pde5 inhibitors

Publications (1)

Publication Number Publication Date
HK1120803A1 true HK1120803A1 (en) 2009-04-09

Family

ID=37685872

Family Applications (1)

Application Number Title Priority Date Filing Date
HK09100008.1A HK1120803A1 (en) 2005-11-10 2009-01-02 Pyrazolo

Country Status (30)

Country Link
US (2) US20090156618A1 (es)
EP (1) EP1948661B1 (es)
JP (1) JP4208959B1 (es)
KR (1) KR101012592B1 (es)
CN (1) CN101305007B (es)
AP (1) AP2008004437A0 (es)
AR (1) AR057885A1 (es)
AT (1) ATE435865T1 (es)
AU (1) AU2006313486B2 (es)
BR (1) BRPI0618284A2 (es)
CA (1) CA2629339C (es)
CR (1) CR9966A (es)
DE (1) DE602006007728D1 (es)
DK (1) DK1948661T3 (es)
DO (1) DOP2006000248A (es)
EA (1) EA200800920A1 (es)
EC (1) ECSP088441A (es)
ES (1) ES2326919T3 (es)
HK (1) HK1120803A1 (es)
IL (1) IL190456A (es)
MA (1) MA29943B1 (es)
NL (1) NL2000291C2 (es)
NO (1) NO20082593L (es)
PE (1) PE20070764A1 (es)
RS (1) RS20080197A (es)
TN (1) TNSN08209A1 (es)
TW (1) TW200738723A (es)
UY (1) UY29909A1 (es)
WO (1) WO2007054778A1 (es)
ZA (1) ZA200803173B (es)

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Publication number Priority date Publication date Assignee Title
AU2009276420A1 (en) * 2008-08-01 2010-02-04 Biocryst Pharmaceuticals, Inc. Piperidine derivatives as JAK3 inhibitors
WO2010043633A1 (en) * 2008-10-15 2010-04-22 Palau Pharma, S. A. 2h-pyrazolo [4,3-d]pyrimidin-5-amine derivatives as h4 histamine receptor antagonists for the treatment of allergic, immunological and inflammatory diseases
JP2013523809A (ja) * 2010-04-05 2013-06-17 エスケー ケミカルズ カンパニー リミテッド Pde5抑制剤を含む皮膚しわ改善用組成物
JP5948683B2 (ja) * 2011-02-28 2016-07-06 国立研究開発法人国立循環器病研究センター 悪性腫瘍転移抑制用医薬
BR112013026521A2 (pt) 2011-04-21 2016-12-27 Origenis Gmbh pirazolo[4,3-d]pirimidinas úteis como inibidores de cinase
US9637491B2 (en) 2012-10-19 2017-05-02 Origenis Gmbh Pyrazolo[4,3-D]pyrimidines as kinase inhibitors
CN104755086A (zh) * 2012-10-23 2015-07-01 辉瑞公司 四取代的吡唑并[4,3-d]嘧啶化合物用于治疗糖尿病肾病的用途
EP3180008B1 (en) 2014-08-12 2023-11-29 Mezzion Pharma Co., Ltd. Methods of improving myocardial performance in fontan patients using udenafil compositions

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NZ333696A (en) 1996-07-08 2000-06-23 Du Pont Pharm Co Amidinoindoles, amidinoazoles, and analogs thereof as inhibitors of trypsin like protease enzymes like thrombin and Xa factor
CA2329077C (en) 1998-04-20 2007-09-18 Pfizer Inc. Pyrazolopyrimidinone cgmp pde5 inhibitors for the treatment of sexual dysfunction
GB9822238D0 (en) * 1998-10-12 1998-12-09 Pfizer Ltd Process for preparation of pyrazolo[4,3-D]pyrimidin-7-ones and intermediates thereof
CA2347950C (en) 1998-10-23 2005-05-03 Pfizer Inc. Pyrazolopyrimidinone cgmp pde5 inhibitors for the treatment of sexual dysfunction
DE19942474A1 (de) 1999-09-06 2001-03-15 Merck Patent Gmbh Pyrazolo[4,3-d]pyrimidine
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IL190456A0 (en) 2008-11-03
AP2008004437A0 (en) 2008-04-30
CA2629339C (en) 2010-07-27
DE602006007728D1 (de) 2009-08-20
EP1948661A1 (en) 2008-07-30
CA2629339A1 (en) 2007-05-18
KR101012592B1 (ko) 2011-02-07
RS20080197A (en) 2009-05-06
PE20070764A1 (es) 2007-08-13
NL2000291C2 (nl) 2009-02-17
JP4208959B1 (ja) 2009-01-14
DOP2006000248A (es) 2007-10-15
DK1948661T3 (da) 2009-09-07
EP1948661B1 (en) 2009-07-08
TW200738723A (en) 2007-10-16
NL2000291A1 (nl) 2007-05-11
US20110059993A1 (en) 2011-03-10
WO2007054778A1 (en) 2007-05-18
US20090156618A1 (en) 2009-06-18
ATE435865T1 (de) 2009-07-15
JP2009519215A (ja) 2009-05-14
IL190456A (en) 2012-10-31
TNSN08209A1 (fr) 2009-10-30
ES2326919T3 (es) 2009-10-21
EA200800920A1 (ru) 2008-10-30
US8518956B2 (en) 2013-08-27
AU2006313486A1 (en) 2007-05-18
ECSP088441A (es) 2008-06-30
ZA200803173B (en) 2009-01-28
MA29943B1 (fr) 2008-11-03
CN101305007A (zh) 2008-11-12
AR057885A1 (es) 2007-12-26
AU2006313486B2 (en) 2011-10-27
BRPI0618284A2 (pt) 2011-08-23
UY29909A1 (es) 2007-06-29
NO20082593L (no) 2008-07-22
KR20080063830A (ko) 2008-07-07
CN101305007B (zh) 2011-07-20
CR9966A (es) 2008-06-16

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