CR10992A - Preparacion solida que comprende alogliptina y pioglitazona - Google Patents

Preparacion solida que comprende alogliptina y pioglitazona

Info

Publication number
CR10992A
CR10992A CR10992A CR10992A CR10992A CR 10992 A CR10992 A CR 10992A CR 10992 A CR10992 A CR 10992A CR 10992 A CR10992 A CR 10992A CR 10992 A CR10992 A CR 10992A
Authority
CR
Costa Rica
Prior art keywords
solid preparation
pioglitazona
alogliptina
compound
stability
Prior art date
Application number
CR10992A
Other languages
English (en)
Inventor
Kenji Nakamura
Kenichiro Kiyoshima
Junya Nomura
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39240362&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CR10992(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of CR10992A publication Critical patent/CR10992A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4436—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Se proporciona una preparacion solida que contiene el compuesto (I), en donde la definicion del compuesto (I) es como se define en la descripcion, y pioglitazona, que es util como un farmaco terapeutico para diabetes o similar y superior en la propiedad de disolucion, estabilidad quimica y estabilidad en la disolucion.
CR10992A 2007-02-01 2009-08-24 Preparacion solida que comprende alogliptina y pioglitazona CR10992A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2007023594 2007-02-01

Publications (1)

Publication Number Publication Date
CR10992A true CR10992A (es) 2009-09-16

Family

ID=39240362

Family Applications (1)

Application Number Title Priority Date Filing Date
CR10992A CR10992A (es) 2007-02-01 2009-08-24 Preparacion solida que comprende alogliptina y pioglitazona

Country Status (39)

Country Link
US (1) US8637079B2 (es)
EP (1) EP2107905B1 (es)
JP (1) JP5284968B2 (es)
KR (1) KR101486091B1 (es)
CN (1) CN101646420B (es)
AR (1) AR065097A1 (es)
AT (1) ATE488227T1 (es)
AU (1) AU2008211981B2 (es)
BR (1) BRPI0807453B8 (es)
CA (1) CA2677201C (es)
CL (1) CL2008000279A1 (es)
CR (1) CR10992A (es)
CY (1) CY1111264T1 (es)
DE (1) DE602008003522D1 (es)
DK (1) DK2107905T3 (es)
DO (1) DOP2009000195A (es)
EA (1) EA015180B1 (es)
EC (1) ECSP099608A (es)
ES (1) ES2354397T3 (es)
GE (1) GEP20125410B (es)
HK (1) HK1138188A1 (es)
HR (1) HRP20110094T8 (es)
IL (1) IL200108A (es)
JO (1) JO2650B1 (es)
MA (1) MA31169B1 (es)
ME (1) ME01239B (es)
MX (1) MX2009008100A (es)
MY (1) MY147596A (es)
NZ (1) NZ579008A (es)
PE (1) PE20081663A1 (es)
PL (1) PL2107905T3 (es)
PT (1) PT2107905E (es)
RS (1) RS51592B (es)
SI (1) SI2107905T1 (es)
TN (1) TN2009000317A1 (es)
TW (2) TWI453041B (es)
UA (1) UA95828C2 (es)
WO (1) WO2008093882A1 (es)
ZA (1) ZA200905621B (es)

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EP1852108A1 (en) 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG DPP IV inhibitor formulations
KR101536786B1 (ko) 2007-07-19 2015-07-14 다케다 야쿠힌 고교 가부시키가이샤 알로그립틴 및 메트포르민 히드로클로라이드를 포함하는 고체 제제
PE20090938A1 (es) 2007-08-16 2009-08-08 Boehringer Ingelheim Int Composicion farmaceutica que comprende un derivado de benceno sustituido con glucopiranosilo
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CN102946875A (zh) 2010-05-05 2013-02-27 贝林格尔.英格海姆国际有限公司 组合疗法
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Also Published As

Publication number Publication date
IL200108A0 (en) 2010-04-15
RS51592B (en) 2011-08-31
ME01239B (me) 2013-06-20
DK2107905T3 (da) 2011-01-31
CY1111264T1 (el) 2015-08-05
BRPI0807453A2 (pt) 2014-05-20
PT2107905E (pt) 2010-12-17
IL200108A (en) 2012-02-29
EP2107905A1 (en) 2009-10-14
ATE488227T1 (de) 2010-12-15
JP5284968B2 (ja) 2013-09-11
UA95828C2 (ru) 2011-09-12
PL2107905T3 (pl) 2011-04-29
JP2010517937A (ja) 2010-05-27
KR101486091B1 (ko) 2015-01-23
NZ579008A (en) 2012-02-24
HRP20110094T1 (hr) 2011-03-31
CL2008000279A1 (es) 2008-08-18
DOP2009000195A (es) 2009-08-31
GEP20125410B (en) 2012-02-27
MX2009008100A (es) 2009-08-07
CA2677201A1 (en) 2008-08-07
BRPI0807453B1 (pt) 2021-01-05
AU2008211981A1 (en) 2008-08-07
CN101646420A (zh) 2010-02-10
EA015180B1 (ru) 2011-06-30
TW200836775A (en) 2008-09-16
US8637079B2 (en) 2014-01-28
ES2354397T3 (es) 2011-03-14
SI2107905T1 (sl) 2011-03-31
HRP20110094T8 (en) 2011-07-31
MY147596A (en) 2012-12-31
JO2650B1 (en) 2012-06-17
EA200970726A1 (ru) 2010-02-26
CA2677201C (en) 2015-11-17
ECSP099608A (es) 2009-09-29
KR20090109115A (ko) 2009-10-19
AU2008211981B2 (en) 2012-09-20
HK1138188A1 (en) 2010-08-20
WO2008093882A1 (en) 2008-08-07
DE602008003522D1 (de) 2010-12-30
MA31169B1 (fr) 2010-02-01
TW201350143A (zh) 2013-12-16
EP2107905B1 (en) 2010-11-17
TWI453041B (zh) 2014-09-21
US20100092551A1 (en) 2010-04-15
CN101646420B (zh) 2012-11-07
TN2009000317A1 (en) 2010-12-31
PE20081663A1 (es) 2008-12-25
BRPI0807453B8 (pt) 2021-05-25
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