DOP2009000195A - Preparacion solida que comprende alogliptina y pioglitazona cinasas - Google Patents

Preparacion solida que comprende alogliptina y pioglitazona cinasas

Info

Publication number
DOP2009000195A
DOP2009000195A DO2009000195A DO2009000195A DOP2009000195A DO P2009000195 A DOP2009000195 A DO P2009000195A DO 2009000195 A DO2009000195 A DO 2009000195A DO 2009000195 A DO2009000195 A DO 2009000195A DO P2009000195 A DOP2009000195 A DO P2009000195A
Authority
DO
Dominican Republic
Prior art keywords
solid preparation
pioglitazona
cinasas
alogliptina
compound
Prior art date
Application number
DO2009000195A
Other languages
English (en)
Inventor
Kenji Nakamura
Kenichiro Kiyoshima
Junya Nomura
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39240362&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DOP2009000195(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of DOP2009000195A publication Critical patent/DOP2009000195A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4436—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Se proporciona una preparación sólida que contiene el compuesto (I), en donde la definición del compuesto (I) es como se define en la descripción, y pioglitazona, que es útil como un fármaco terapéutico para diabetes o similar y superior en la propiedad de disolución, estabilidad química y estabilidad en la disolución. Una preparación sólida que contiene las siguientes primera y segunda partes: (1) la primera parte contiene el compuesto (I) o una de sus sales, como el primer excipiente, azúcar o alcohol de azúcar, y (2) la segunda parte contiene pioglitazona o una de sus sales y, como el segundo excipiente, azúcar o alcohol de azúcar.
DO2009000195A 2007-02-01 2009-07-31 Preparacion solida que comprende alogliptina y pioglitazona cinasas DOP2009000195A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2007023594 2007-02-01

Publications (1)

Publication Number Publication Date
DOP2009000195A true DOP2009000195A (es) 2009-08-31

Family

ID=39240362

Family Applications (1)

Application Number Title Priority Date Filing Date
DO2009000195A DOP2009000195A (es) 2007-02-01 2009-07-31 Preparacion solida que comprende alogliptina y pioglitazona cinasas

Country Status (39)

Country Link
US (1) US8637079B2 (es)
EP (1) EP2107905B1 (es)
JP (1) JP5284968B2 (es)
KR (1) KR101486091B1 (es)
CN (1) CN101646420B (es)
AR (1) AR065097A1 (es)
AT (1) ATE488227T1 (es)
AU (1) AU2008211981B2 (es)
BR (1) BRPI0807453B8 (es)
CA (1) CA2677201C (es)
CL (1) CL2008000279A1 (es)
CR (1) CR10992A (es)
CY (1) CY1111264T1 (es)
DE (1) DE602008003522D1 (es)
DK (1) DK2107905T3 (es)
DO (1) DOP2009000195A (es)
EA (1) EA015180B1 (es)
EC (1) ECSP099608A (es)
ES (1) ES2354397T3 (es)
GE (1) GEP20125410B (es)
HK (1) HK1138188A1 (es)
HR (1) HRP20110094T8 (es)
IL (1) IL200108A (es)
JO (1) JO2650B1 (es)
MA (1) MA31169B1 (es)
ME (1) ME01239B (es)
MX (1) MX2009008100A (es)
MY (1) MY147596A (es)
NZ (1) NZ579008A (es)
PE (1) PE20081663A1 (es)
PL (1) PL2107905T3 (es)
PT (1) PT2107905E (es)
RS (1) RS51592B (es)
SI (1) SI2107905T1 (es)
TN (1) TN2009000317A1 (es)
TW (2) TWI453041B (es)
UA (1) UA95828C2 (es)
WO (1) WO2008093882A1 (es)
ZA (1) ZA200905621B (es)

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Also Published As

Publication number Publication date
IL200108A0 (en) 2010-04-15
RS51592B (en) 2011-08-31
ME01239B (me) 2013-06-20
DK2107905T3 (da) 2011-01-31
CY1111264T1 (el) 2015-08-05
CR10992A (es) 2009-09-16
BRPI0807453A2 (pt) 2014-05-20
PT2107905E (pt) 2010-12-17
IL200108A (en) 2012-02-29
EP2107905A1 (en) 2009-10-14
ATE488227T1 (de) 2010-12-15
JP5284968B2 (ja) 2013-09-11
UA95828C2 (ru) 2011-09-12
PL2107905T3 (pl) 2011-04-29
JP2010517937A (ja) 2010-05-27
KR101486091B1 (ko) 2015-01-23
NZ579008A (en) 2012-02-24
HRP20110094T1 (hr) 2011-03-31
CL2008000279A1 (es) 2008-08-18
GEP20125410B (en) 2012-02-27
MX2009008100A (es) 2009-08-07
CA2677201A1 (en) 2008-08-07
BRPI0807453B1 (pt) 2021-01-05
AU2008211981A1 (en) 2008-08-07
CN101646420A (zh) 2010-02-10
EA015180B1 (ru) 2011-06-30
TW200836775A (en) 2008-09-16
US8637079B2 (en) 2014-01-28
ES2354397T3 (es) 2011-03-14
SI2107905T1 (sl) 2011-03-31
HRP20110094T8 (en) 2011-07-31
MY147596A (en) 2012-12-31
JO2650B1 (en) 2012-06-17
EA200970726A1 (ru) 2010-02-26
CA2677201C (en) 2015-11-17
ECSP099608A (es) 2009-09-29
KR20090109115A (ko) 2009-10-19
AU2008211981B2 (en) 2012-09-20
HK1138188A1 (en) 2010-08-20
WO2008093882A1 (en) 2008-08-07
DE602008003522D1 (de) 2010-12-30
MA31169B1 (fr) 2010-02-01
TW201350143A (zh) 2013-12-16
EP2107905B1 (en) 2010-11-17
TWI453041B (zh) 2014-09-21
US20100092551A1 (en) 2010-04-15
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TN2009000317A1 (en) 2010-12-31
PE20081663A1 (es) 2008-12-25
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AR065097A1 (es) 2009-05-13
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