UY31864A - Derivados de urea hetericíclica y métodos de uso de los mismos-332 - Google Patents
Derivados de urea hetericíclica y métodos de uso de los mismos-332Info
- Publication number
- UY31864A UY31864A UY0001031864A UY31864A UY31864A UY 31864 A UY31864 A UY 31864A UY 0001031864 A UY0001031864 A UY 0001031864A UY 31864 A UY31864 A UY 31864A UY 31864 A UY31864 A UY 31864A
- Authority
- UY
- Uruguay
- Prior art keywords
- hetericíclica
- urea
- derivatives
- methods
- same
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/06—Peri-condensed systems
Abstract
Se describen compuestos de fórmula (I) y sus sales farmacéuticamente aceptables. También se describen procesos para su preparación, composiciones farmacéuticas que los contienen, su uso como medicamentos y su uso en el tratamiento de infecciones bacterianas.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US5873608P | 2008-06-04 | 2008-06-04 |
Publications (1)
Publication Number | Publication Date |
---|---|
UY31864A true UY31864A (es) | 2010-01-29 |
Family
ID=40823415
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY0001031864A UY31864A (es) | 2008-06-04 | 2009-06-03 | Derivados de urea hetericíclica y métodos de uso de los mismos-332 |
Country Status (23)
Country | Link |
---|---|
US (1) | US8283361B2 (es) |
EP (1) | EP2300463A1 (es) |
JP (1) | JP2011522026A (es) |
KR (1) | KR20110014710A (es) |
CN (1) | CN102105469A (es) |
AR (1) | AR072045A1 (es) |
AU (1) | AU2009254930A1 (es) |
BR (1) | BRPI0915471A2 (es) |
CA (1) | CA2725568A1 (es) |
CL (1) | CL2009001349A1 (es) |
CO (1) | CO6382176A2 (es) |
CR (1) | CR11825A (es) |
DO (1) | DOP2010000373A (es) |
EA (1) | EA201001858A1 (es) |
EC (1) | ECSP10010664A (es) |
IL (1) | IL209503A0 (es) |
MX (1) | MX2010013310A (es) |
PE (1) | PE20100155A1 (es) |
SV (1) | SV2010003752A (es) |
TW (1) | TW201000475A (es) |
UY (1) | UY31864A (es) |
WO (1) | WO2009147433A1 (es) |
ZA (1) | ZA201008610B (es) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20100130737A1 (en) * | 2005-02-18 | 2010-05-27 | Takeda Pharmaceutical Company Limited | Regulating Agent of GPR34 Receptor Function |
TW201102065A (en) * | 2009-05-29 | 2011-01-16 | Astrazeneca Ab | Heterocyclic urea derivatives and methods of use thereof |
WO2010142978A1 (en) * | 2009-06-08 | 2010-12-16 | Astrazeneca Ab | Heterocyclic urea derivatives and methods of use thereof |
MX2012010666A (es) | 2010-03-31 | 2012-10-05 | Actelion Pharmaceuticals Ltd | Derivados de isoquinolin-3-ilurea antibacterianos. |
AR088729A1 (es) | 2011-03-29 | 2014-07-02 | Actelion Pharmaceuticals Ltd | Derivados de 3-ureidoisoquinolin-8-ilo y una composicion farmaceutica |
CN105067814A (zh) * | 2015-07-24 | 2015-11-18 | 中国科学院成都生物研究所 | 解旋酶水解atp活性测定方法 |
WO2018048882A1 (en) | 2016-09-06 | 2018-03-15 | The Research Foundation For The State University Of New York | Positron imaging tomography imaging agent composition and method for bacterial infection |
WO2018074880A2 (ko) * | 2016-10-20 | 2018-04-26 | 한국화학연구원 | 퀴놀린 4-온 유도체 또는 이의 약학적으로 허용 가능한 염을 유효성분으로 포함하는 폐렴의 예방 또는 치료용 약학적 조성물 |
WO2018174288A1 (ja) | 2017-03-24 | 2018-09-27 | 大正製薬株式会社 | 2(1h)-キノリノン誘導体 |
CN111808089B (zh) * | 2019-04-10 | 2023-04-11 | 四川大学华西医院 | 一种治疗糖尿病的药物依格列净或其衍生物的制备方法 |
Family Cites Families (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1993000342A1 (en) | 1991-06-21 | 1993-01-07 | Boehringer Mannheim Italia S.P.A. | 2-amino-4-aryl-thiazoles with antiasthmatic and anti-inflammatory activities on the respiratory tract |
MXPA03005298A (es) | 2000-12-15 | 2003-10-06 | Vertex Pharma | Inhibidores de girasa y usos de los mismos. |
AR042956A1 (es) | 2003-01-31 | 2005-07-13 | Vertex Pharma | Inhibidores de girasa y usos de los mismos |
WO2006092599A2 (en) * | 2005-03-04 | 2006-09-08 | Astrazeneca Ab | Pyrrole derivatives as dna gyrase and topoisomerase inhibitors |
US8022816B2 (en) | 2005-03-21 | 2011-09-20 | Vela Systems, Inc. | System and method for field management using radio frequency tags |
US7569907B2 (en) | 2005-03-28 | 2009-08-04 | Cooper Technologies Company | Hybrid chip fuse assembly having wire leads and fabrication method therefor |
ATE435489T1 (de) | 2005-04-13 | 2009-07-15 | Koninkl Philips Electronics Nv | Modifizierte dct transformation zur basisband- phasenmodulation von einem mp3 bitstream, und einfügung von wasserzeichen. |
WO2007071965A2 (en) * | 2005-12-23 | 2007-06-28 | Astrazeneca Ab | Antibacterial pyrrolopyridines, pyrrolopyrimidines, and pyrroloazepines |
DE102006012337B3 (de) | 2006-03-17 | 2007-11-29 | Amphenol-Tuchel Electronics Gmbh | Elektrischer Steckverbinder |
CN101627038A (zh) * | 2006-12-04 | 2010-01-13 | 阿斯利康(瑞典)有限公司 | 抗菌多环脲化合物 |
CN201038186Y (zh) | 2007-03-08 | 2008-03-19 | 鹤山丽得电子实业有限公司 | 一种大功率led |
TW200940537A (en) * | 2008-02-26 | 2009-10-01 | Astrazeneca Ab | Heterocyclic urea derivatives and methods of use thereof |
WO2009110688A2 (ko) | 2008-03-06 | 2009-09-11 | Jang Gum Sik | 태양광 발전 장치 |
WO2010142978A1 (en) * | 2009-06-08 | 2010-12-16 | Astrazeneca Ab | Heterocyclic urea derivatives and methods of use thereof |
-
2009
- 2009-06-03 TW TW098118462A patent/TW201000475A/zh unknown
- 2009-06-03 CL CL2009001349A patent/CL2009001349A1/es unknown
- 2009-06-03 WO PCT/GB2009/050611 patent/WO2009147433A1/en active Application Filing
- 2009-06-03 BR BRPI0915471A patent/BRPI0915471A2/pt not_active IP Right Cessation
- 2009-06-03 JP JP2011512216A patent/JP2011522026A/ja active Pending
- 2009-06-03 EP EP09757805A patent/EP2300463A1/en not_active Withdrawn
- 2009-06-03 CN CN2009801294194A patent/CN102105469A/zh active Pending
- 2009-06-03 MX MX2010013310A patent/MX2010013310A/es not_active Application Discontinuation
- 2009-06-03 KR KR1020117000030A patent/KR20110014710A/ko not_active Application Discontinuation
- 2009-06-03 CA CA2725568A patent/CA2725568A1/en not_active Abandoned
- 2009-06-03 EA EA201001858A patent/EA201001858A1/ru unknown
- 2009-06-03 AU AU2009254930A patent/AU2009254930A1/en not_active Abandoned
- 2009-06-03 UY UY0001031864A patent/UY31864A/es not_active Application Discontinuation
- 2009-06-03 US US12/477,781 patent/US8283361B2/en not_active Expired - Fee Related
- 2009-06-04 PE PE2009000774A patent/PE20100155A1/es not_active Application Discontinuation
- 2009-06-04 AR ARP090102012A patent/AR072045A1/es unknown
-
2010
- 2010-11-22 IL IL209503A patent/IL209503A0/en unknown
- 2010-11-30 ZA ZA2010/08610A patent/ZA201008610B/en unknown
- 2010-12-03 DO DO2010000373A patent/DOP2010000373A/es unknown
- 2010-12-06 SV SV2010003752A patent/SV2010003752A/es not_active Application Discontinuation
- 2010-12-06 CR CR11825A patent/CR11825A/es not_active Application Discontinuation
- 2010-12-07 EC EC2010010664A patent/ECSP10010664A/es unknown
- 2010-12-22 CO CO10160874A patent/CO6382176A2/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
AU2009254930A1 (en) | 2009-12-10 |
CA2725568A1 (en) | 2009-12-10 |
CN102105469A (zh) | 2011-06-22 |
DOP2010000373A (es) | 2011-01-15 |
CR11825A (es) | 2011-02-04 |
ZA201008610B (en) | 2012-08-29 |
IL209503A0 (en) | 2011-01-31 |
SV2010003752A (es) | 2011-04-14 |
AR072045A1 (es) | 2010-08-04 |
CO6382176A2 (es) | 2012-02-15 |
MX2010013310A (es) | 2011-03-01 |
KR20110014710A (ko) | 2011-02-11 |
JP2011522026A (ja) | 2011-07-28 |
EP2300463A1 (en) | 2011-03-30 |
US8283361B2 (en) | 2012-10-09 |
TW201000475A (en) | 2010-01-01 |
PE20100155A1 (es) | 2010-03-25 |
WO2009147433A1 (en) | 2009-12-10 |
ECSP10010664A (es) | 2011-01-31 |
US20100190745A1 (en) | 2010-07-29 |
BRPI0915471A2 (pt) | 2017-06-27 |
CL2009001349A1 (es) | 2010-12-31 |
EA201001858A1 (ru) | 2011-08-30 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
109 | Application deemed to be withdrawn |
Effective date: 20181029 |