UY31860A - Piridinas de tiazolo como inhibidoras de la adn girasa - Google Patents

Piridinas de tiazolo como inhibidoras de la adn girasa

Info

Publication number
UY31860A
UY31860A UY0001031860A UY31860A UY31860A UY 31860 A UY31860 A UY 31860A UY 0001031860 A UY0001031860 A UY 0001031860A UY 31860 A UY31860 A UY 31860A UY 31860 A UY31860 A UY 31860A
Authority
UY
Uruguay
Prior art keywords
girasa
piridines
tiazolo
inhibitors
dna
Prior art date
Application number
UY0001031860A
Other languages
English (en)
Inventor
Manoj Ganpat Kale
Shahul Hameed Peer Mohamed
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40872366&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY31860(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of UY31860A publication Critical patent/UY31860A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Son descritos los compuestos de la fórmula (I) y sus sales farmacéuticamente aceptables. Los procesos para su preparación, las composiciones farmacéuticas que los contienen, su uso como medicamentos y su uso en el tratamiento de infecciones bacterianas son también descritos.
UY0001031860A 2008-06-04 2009-06-03 Piridinas de tiazolo como inhibidoras de la adn girasa UY31860A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US5874808P 2008-06-04 2008-06-04

Publications (1)

Publication Number Publication Date
UY31860A true UY31860A (es) 2010-01-29

Family

ID=40872366

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001031860A UY31860A (es) 2008-06-04 2009-06-03 Piridinas de tiazolo como inhibidoras de la adn girasa

Country Status (16)

Country Link
US (1) US20100137303A1 (es)
EP (1) EP2303894A1 (es)
JP (1) JP2011522024A (es)
KR (1) KR20110031419A (es)
CN (1) CN102056932A (es)
AR (1) AR072047A1 (es)
AU (1) AU2009254928A1 (es)
BR (1) BRPI0913300A2 (es)
CA (1) CA2725689A1 (es)
CL (1) CL2009001346A1 (es)
MX (1) MX2010013249A (es)
PE (1) PE20100053A1 (es)
RU (1) RU2010154499A (es)
TW (1) TW201002723A (es)
UY (1) UY31860A (es)
WO (1) WO2009147431A1 (es)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20100017689A (ko) 2007-05-09 2010-02-16 셀 인터나쵸나아레 레사아치 마아츠샤피 비이부이 에폭시화 촉매, 이 촉매의 제조방법, 및 산화올레핀, 1,2-디올, 1,2-디올 에테르, 1,2-카보네이트 또는 알칸올아민의 생산 방법
BR112012024705A2 (pt) 2010-03-31 2016-06-07 Actelion Pharmaceuticals Ltd derivados antibacterianos de isoquinolin-3-ilureia
ME02663B (me) 2010-10-06 2017-06-20 Glaxosmithkline Llc Derivati benzimidazola kao inhibitori pi3 kinaze
AR088729A1 (es) 2011-03-29 2014-07-02 Actelion Pharmaceuticals Ltd Derivados de 3-ureidoisoquinolin-8-ilo y una composicion farmaceutica
EP2721026B1 (en) * 2011-06-20 2016-03-02 Vertex Pharmaceuticals Incorporated Phosphate esters of gyrase and topoisomerase inhibitors
JP2015514063A (ja) * 2012-03-22 2015-05-18 ビオタ ヨーロッパ リミテッドＢｉｏｔａ Ｅｕｒｏｐｅ Ｌｔｄ 抗菌化合物
CN104718213B (zh) * 2012-07-18 2018-02-27 圣母大学 5,5‑杂芳族抗感染化合物
KR101602559B1 (ko) * 2014-04-29 2016-03-10 경북대학교 산학협력단 2,5,6,7-사중치환 티아졸로[4,5-b]피리딘 유도체 및 이의 용도
CN104788473B (zh) * 2015-03-25 2017-03-15 石家庄学院 一种具有抗菌能力的化合物及其制备方法与用途
CN104744493B (zh) * 2015-04-08 2017-01-25 石家庄学院 3‑苯甲酰基‑5,7‑二苯基‑5H‑噻唑并[3,2‑a]嘧啶类衍生物及其应用
WO2018095953A1 (de) 2016-11-23 2018-05-31 Bayer Cropscience Aktiengesellschaft 2-[3-(alkylsulfonyl)-2h-indazol-2-yl]-3h-imidazo[4,5-b]pyridin-derivate und ähnliche verbindungen als schädlingsbekämpfungsmittel
CA3057431A1 (en) 2017-03-24 2018-09-27 Taisho Pharmaceutical Co., Ltd. 2(1h)-quinolinone derivative
BR112019020464A2 (pt) 2017-03-30 2020-04-28 Xw Laboratories Inc. compostos derivados de heteroarila bicíclica, composição farmacêutica compreendendo os ditos compostos, adesivo transdérmico compreendendo a dita composição e uso terapêutico dos compostos e composição
WO2020048949A1 (en) 2018-09-03 2020-03-12 Univerza V Ljubljani New class of dna gyrase and/or topoisomerase iv inhibitors with activity against gram-positive and gram-negative bacteria
WO2022129327A1 (en) 2020-12-17 2022-06-23 Univerza V Ljubljani New n-phenylpyrrolamide inhibitors of dna gyrase and topoisomerase iv with antibacterial activity
WO2022165198A1 (en) * 2021-01-29 2022-08-04 Board Of Trustees Of Michigan State University Therapeutic compounds and uses thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUP0303494A3 (en) * 2000-12-15 2009-08-28 Vertex Pharma Parmaceutical compositions containing bacterial gyrase inhibitors and uses thereof
KR20060079098A (ko) * 2004-12-31 2006-07-05 주식회사 엘지생명과학 신규한([1,3]티아졸로[5,4-ｂ]피리딘-2-일)-2-카르복사마이드유도체
GB0724342D0 (en) * 2007-12-13 2008-01-30 Prolysis Ltd Anitbacterial compositions
MX2010011370A (es) * 2008-04-16 2010-12-15 Vertex Pharma Inhibidores de fosfatidilinositol 3-cinasa.

Also Published As

Publication number Publication date
JP2011522024A (ja) 2011-07-28
RU2010154499A (ru) 2012-07-20
WO2009147431A1 (en) 2009-12-10
CA2725689A1 (en) 2009-12-10
PE20100053A1 (es) 2010-02-25
EP2303894A1 (en) 2011-04-06
BRPI0913300A2 (pt) 2018-05-22
AR072047A1 (es) 2010-08-04
MX2010013249A (es) 2010-12-21
TW201002723A (en) 2010-01-16
AU2009254928A1 (en) 2009-12-10
KR20110031419A (ko) 2011-03-28
CN102056932A (zh) 2011-05-11
CL2009001346A1 (es) 2010-07-02
US20100137303A1 (en) 2010-06-03

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Effective date: 20130122