CN1914180A - 作为激素敏感性脂肪酶抑制剂的吲唑衍生物 - Google Patents

作为激素敏感性脂肪酶抑制剂的吲唑衍生物 Download PDF

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Publication number
CN1914180A
CN1914180A CNA2005800037984A CN200580003798A CN1914180A CN 1914180 A CN1914180 A CN 1914180A CN A2005800037984 A CNA2005800037984 A CN A2005800037984A CN 200580003798 A CN200580003798 A CN 200580003798A CN 1914180 A CN1914180 A CN 1914180A
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China
Prior art keywords
alkyl
indazole
indazole derivatives
ring system
desired formula
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CNA2005800037984A
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English (en)
Chinese (zh)
Inventor
G·策勒
S·佩特里
G·米勒
H·霍耶尔
K-H·巴林豪斯
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Sanofi Aventis Deutschland GmbH
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Sanofi Aventis Deutschland GmbH
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Publication of CN1914180A publication Critical patent/CN1914180A/zh
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    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
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  • Obesity (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Dermatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Cardiology (AREA)
  • Psychology (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Endocrinology (AREA)
  • Hospice & Palliative Care (AREA)
  • Emergency Medicine (AREA)
  • Psychiatry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CNA2005800037984A 2004-02-02 2005-01-15 作为激素敏感性脂肪酶抑制剂的吲唑衍生物 Pending CN1914180A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102004005172A DE102004005172A1 (de) 2004-02-02 2004-02-02 Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
DE102004005172.0 2004-02-02

Publications (1)

Publication Number Publication Date
CN1914180A true CN1914180A (zh) 2007-02-14

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CNA2005800037984A Pending CN1914180A (zh) 2004-02-02 2005-01-15 作为激素敏感性脂肪酶抑制剂的吲唑衍生物

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US (2) US7528155B2 (US20070167479A1-20070719-C00034.png)
EP (1) EP1713779B1 (US20070167479A1-20070719-C00034.png)
JP (1) JP4714158B2 (US20070167479A1-20070719-C00034.png)
KR (1) KR20060128958A (US20070167479A1-20070719-C00034.png)
CN (1) CN1914180A (US20070167479A1-20070719-C00034.png)
AR (1) AR047520A1 (US20070167479A1-20070719-C00034.png)
AT (1) ATE505460T1 (US20070167479A1-20070719-C00034.png)
AU (1) AU2005209366A1 (US20070167479A1-20070719-C00034.png)
BR (1) BRPI0507370A (US20070167479A1-20070719-C00034.png)
CA (1) CA2554524A1 (US20070167479A1-20070719-C00034.png)
CR (1) CR8487A (US20070167479A1-20070719-C00034.png)
DE (2) DE102004005172A1 (US20070167479A1-20070719-C00034.png)
DO (1) DOP2005000011A (US20070167479A1-20070719-C00034.png)
EC (1) ECSP066750A (US20070167479A1-20070719-C00034.png)
HN (1) HN2005000039A (US20070167479A1-20070719-C00034.png)
IL (1) IL176912A (US20070167479A1-20070719-C00034.png)
MA (1) MA28338A1 (US20070167479A1-20070719-C00034.png)
MY (1) MY143407A (US20070167479A1-20070719-C00034.png)
NO (1) NO20063925L (US20070167479A1-20070719-C00034.png)
NZ (1) NZ548872A (US20070167479A1-20070719-C00034.png)
PE (1) PE20050690A1 (US20070167479A1-20070719-C00034.png)
RU (1) RU2370491C2 (US20070167479A1-20070719-C00034.png)
SG (1) SG149891A1 (US20070167479A1-20070719-C00034.png)
TW (1) TW200536535A (US20070167479A1-20070719-C00034.png)
UY (1) UY28735A1 (US20070167479A1-20070719-C00034.png)
WO (1) WO2005073199A1 (US20070167479A1-20070719-C00034.png)
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Cited By (1)

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CN104662002A (zh) * 2012-07-27 2015-05-27 比亚尔-珀特拉和Ca股份公司 取代脲类化合物的合成方法

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JP4734119B2 (ja) * 2004-02-12 2011-07-27 田辺三菱製薬株式会社 インダゾール化合物及びその医薬用途
EP1586573B1 (en) 2004-04-01 2007-02-07 Sanofi-Aventis Deutschland GmbH Oxadiazolones, processes for their preparation and their use as pharmaceuticals
DE102005026762A1 (de) 2005-06-09 2006-12-21 Sanofi-Aventis Deutschland Gmbh Azolopyridin-2-on-derivate als Inhibitoren von Lipasen und Phospholipasen
DE102005026808A1 (de) 2005-06-09 2006-12-14 Sanofi-Aventis Deutschland Gmbh Benzooxazol-2-on-derivate als Inhibitoren von Lipasen und Phospholipasen
DE102005048897A1 (de) 2005-10-12 2007-04-19 Sanofi-Aventis Deutschland Gmbh Diacylindazol-derivate als Inhibitoren von Lipasen und Phospholipasen
DE102005049954A1 (de) * 2005-10-19 2007-05-31 Sanofi-Aventis Deutschland Gmbh Triazolopyridin-derivate als Inhibitoren von Lipasen und Phospholipasen
DE102006014688A1 (de) 2006-03-28 2007-10-04 Sanofi-Aventis Azolopyridin-3-on-derivate als Inhibitoren von Lipasen und Phospholipasen
DE102006014685A1 (de) * 2006-03-28 2007-10-04 Sanofi-Aventis Imidazo-pyridin-2-on-derivate als Inhibitoren von Lipasen und Phospholiphasen
RU2009108280A (ru) 2006-08-08 2010-09-20 Санофи-Авентис (Fr) Ариламиноарилалкилзамещенные имидазолидин-2,4-дионы, способы их получения, содержащие эти соединения лекарственные средства и их применение
BRPI0810044A2 (pt) * 2007-04-05 2014-10-14 Sanofi Aventis 5-oxoisoxazóis como inibidores de lipases e fosfolipases
FR2915197B1 (fr) 2007-04-18 2009-06-12 Sanofi Aventis Sa Derives de triazolopyridine-carboxamides, leur preparation et leur application therapeutique.
FR2915198B1 (fr) * 2007-04-18 2009-12-18 Sanofi Aventis Derives de triazolopyridine-carboxamides et triazolopyridine -carboxamides, leur preparation et leur application en therapeutique.
FR2915199B1 (fr) 2007-04-18 2010-01-22 Sanofi Aventis Derives de triazolopyridine-carboxamides et triazolopyrimidine-carboxamides, leur preparation et leur application en therapeutique.
WO2008156757A1 (en) * 2007-06-19 2008-12-24 Takeda Pharmaceutical Company Limited Indazole compounds for activating glucokinase
EP2025674A1 (de) 2007-08-15 2009-02-18 sanofi-aventis Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
DE102007043281A1 (de) 2007-09-11 2009-05-28 Sebastian Dr. med. Chakrit Bhakdi Vorrichtung, Materialien und Verfahren zur Hochgradientenmagnetseparation biologischen Materials
UY31968A (es) 2008-07-09 2010-01-29 Sanofi Aventis Nuevos derivados heterocíclicos, sus procesos para su preparación, y sus usos terapéuticos
WO2010068601A1 (en) 2008-12-08 2010-06-17 Sanofi-Aventis A crystalline heteroaromatic fluoroglycoside hydrate, processes for making, methods of use and pharmaceutical compositions thereof
SG178880A1 (en) 2009-08-26 2012-04-27 Sanofi Sa Novel crystalline heteroaromatic fluoroglycoside hydrates, pharmaceuticals comprising these compounds and their use
WO2011107494A1 (de) 2010-03-03 2011-09-09 Sanofi Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung
WO2011157827A1 (de) 2010-06-18 2011-12-22 Sanofi Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen
US8530413B2 (en) 2010-06-21 2013-09-10 Sanofi Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
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