FR2915199B1 - Derives de triazolopyridine-carboxamides et triazolopyrimidine-carboxamides, leur preparation et leur application en therapeutique. - Google Patents
Derives de triazolopyridine-carboxamides et triazolopyrimidine-carboxamides, leur preparation et leur application en therapeutique.Info
- Publication number
- FR2915199B1 FR2915199B1 FR0702809A FR0702809A FR2915199B1 FR 2915199 B1 FR2915199 B1 FR 2915199B1 FR 0702809 A FR0702809 A FR 0702809A FR 0702809 A FR0702809 A FR 0702809A FR 2915199 B1 FR2915199 B1 FR 2915199B1
- Authority
- FR
- France
- Prior art keywords
- carboxamide
- triazolopyridine
- triazolopyrimidine
- preparation
- therapeutic use
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Hematology (AREA)
- Communicable Diseases (AREA)
- Diabetes (AREA)
- Oncology (AREA)
- Pulmonology (AREA)
- Urology & Nephrology (AREA)
- Cardiology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Ophthalmology & Optometry (AREA)
- Virology (AREA)
- Obesity (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Dermatology (AREA)
- Psychology (AREA)
- AIDS & HIV (AREA)
- Vascular Medicine (AREA)
Priority Applications (17)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0702809A FR2915199B1 (fr) | 2007-04-18 | 2007-04-18 | Derives de triazolopyridine-carboxamides et triazolopyrimidine-carboxamides, leur preparation et leur application en therapeutique. |
KR1020097021591A KR20090130057A (ko) | 2007-04-18 | 2008-04-16 | 트리아졸로피리딘 카르복스아미드 유도체 및 트리아졸로피리미딘 카르복스아미드 유도체, 그의 제조 및 그의 치료학적 용도 |
PCT/FR2008/000532 WO2008145839A1 (fr) | 2007-04-18 | 2008-04-16 | Dérivés de triazolopyridine-carboxamides et triazolopyrimidine-carboxamides, leur préparation et leur application en thérapeutique |
CA002683929A CA2683929A1 (fr) | 2007-04-18 | 2008-04-16 | Derives de triazolopyridine-carboxamides et triazolopyrimidine-carboxamides, leur preparation et leur application en therapeutique |
EP08787961A EP2146990A1 (fr) | 2007-04-18 | 2008-04-16 | Dérivés de triazolopyridine-carboxamides et triazolopyrimidine-carboxamides, leur préparation et leur application en thérapeutique |
CN200880012545A CN101668758A (zh) | 2007-04-18 | 2008-04-16 | 三唑并吡啶-甲酰胺和三唑并嘧啶-甲酰胺衍生物、它们的制备和它们的治疗应用 |
AU2008257320A AU2008257320A1 (en) | 2007-04-18 | 2008-04-16 | Triazolopyridine carboxamide derivatives and triazolopyrimidine carboxamide derivatives, preparation thereof and therapeutic use thereof |
BRPI0810440-9A2A BRPI0810440A2 (pt) | 2007-04-18 | 2008-04-16 | Derivados de triazolopiridina-carboxamidas e triazolopirimidina-carboxamidas, o respectivo preparo e a respectiva aplicação em terapêutica |
MX2009011212A MX2009011212A (es) | 2007-04-18 | 2008-04-16 | Derivados de triazolopiridina carboxamida y triazolopirimidina carboxamida, su preparacion y su aplicacion terapeutica. |
RU2009142431/04A RU2009142431A (ru) | 2007-04-18 | 2008-04-16 | Производные триазолопиридинкарбоксамидов и триазолопиримидинкарбоксамидов, их получение и их применение в терапии |
JP2010503547A JP2010524904A (ja) | 2007-04-18 | 2008-04-16 | トリアゾロピリジンカルボキサミド誘導体およびトリアゾロピリミジンカルボキサミド誘導体、これらの調製、ならびにこれらの治療的使用 |
TW097114018A TW200901993A (en) | 2007-04-18 | 2008-04-17 | Triazolopyridine carboxamide and triazolopyrimidine carboxamide derivatives, their preparation and their application in therapeutics |
CL2008001104A CL2008001104A1 (es) | 2007-04-18 | 2008-04-17 | Compuestos derivados de [1,2,3]triazolo[4,5-b]piridin-carboxamidas y [1,2,3]triazolo[4,5-d]pirimidin-carboxamidas, inhibidores de mgl y faah; procedimiento de preparacion; composicion farmaceutica; y su uso en el tratamiento de delolores agudos o cronicos, vertigos, vomitos, nauseas, sindrome metaloico, dispipidemia, entre otros. |
ARP080101601A AR066107A1 (es) | 2007-04-18 | 2008-04-18 | Derivados de triazolopiridin - carboxamidas y triazolopirimidin-carboxamidas, su preparacion y su aplicacion en terapeutica como inhibidores de la enzimamonoacil glicerol lipasa y composiciones qu los contienen. |
UY31032A UY31032A1 (es) | 2007-04-18 | 2008-04-18 | Derivados de triazolopiridin-carboxamidas y triazolopirimidin-carboxinamidas, su preparacion y su aplicacion en terapeutica |
US12/573,959 US8080547B2 (en) | 2007-04-18 | 2009-10-06 | Triazolopyridine carboxamide derivatives and triazolopyrimidine carboxamide derivatives, preparation thereof and therapeutic use thereof |
IL201450A IL201450A0 (en) | 2007-04-18 | 2009-10-11 | Triazolopyridine carboxamide derivatives and triazolopyrimidine carboxamide derivatives, preparation thereof and therapeutic use thereof |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0702809A FR2915199B1 (fr) | 2007-04-18 | 2007-04-18 | Derives de triazolopyridine-carboxamides et triazolopyrimidine-carboxamides, leur preparation et leur application en therapeutique. |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2915199A1 FR2915199A1 (fr) | 2008-10-24 |
FR2915199B1 true FR2915199B1 (fr) | 2010-01-22 |
Family
ID=38776272
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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FR0702809A Expired - Fee Related FR2915199B1 (fr) | 2007-04-18 | 2007-04-18 | Derives de triazolopyridine-carboxamides et triazolopyrimidine-carboxamides, leur preparation et leur application en therapeutique. |
Country Status (17)
Country | Link |
---|---|
US (1) | US8080547B2 (fr) |
EP (1) | EP2146990A1 (fr) |
JP (1) | JP2010524904A (fr) |
KR (1) | KR20090130057A (fr) |
CN (1) | CN101668758A (fr) |
AR (1) | AR066107A1 (fr) |
AU (1) | AU2008257320A1 (fr) |
BR (1) | BRPI0810440A2 (fr) |
CA (1) | CA2683929A1 (fr) |
CL (1) | CL2008001104A1 (fr) |
FR (1) | FR2915199B1 (fr) |
IL (1) | IL201450A0 (fr) |
MX (1) | MX2009011212A (fr) |
RU (1) | RU2009142431A (fr) |
TW (1) | TW200901993A (fr) |
UY (1) | UY31032A1 (fr) |
WO (1) | WO2008145839A1 (fr) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102459167B (zh) * | 2009-04-22 | 2015-04-01 | 詹森药业有限公司 | 作为单酰甘油脂肪酶抑制剂的氮杂环丁烷基二酰胺 |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2915198B1 (fr) * | 2007-04-18 | 2009-12-18 | Sanofi Aventis | Derives de triazolopyridine-carboxamides et triazolopyridine -carboxamides, leur preparation et leur application en therapeutique. |
RU2553451C2 (ru) * | 2008-12-24 | 2015-06-20 | Биал-Портела Энд Ка, С.А. | Фармацевтические соединения |
US8435977B2 (en) | 2009-04-22 | 2013-05-07 | Janssen Pharmaceutica, Nv | Heteroaromatic and aromatic piperazinyl azetidinyl amides as monoacylglycerol lipase inhibitors |
AU2010238746B2 (en) * | 2009-04-22 | 2015-02-19 | Janssen Pharmaceutica Nv | Heteroaromatic and aromatic piperazinyl azetidinyl amides as monoacylglycerol lipase inhibitors |
EP2421852B9 (fr) * | 2009-04-22 | 2015-07-01 | Janssen Pharmaceutica N.V. | Pipérazinyl azétidinyl amides hétéroaromatiques et aromatiques en tant qu'inhibiteur de la monoacylglycérol lipase |
AU2010293429B2 (en) * | 2009-09-09 | 2015-12-17 | Sumitomo Dainippon Pharma Co., Ltd. | 8-oxodihydropurine derivative |
US20130150346A1 (en) | 2010-01-08 | 2013-06-13 | Quest Ventures Ltd. | Use of FAAH Inhibitors for Treating Parkinson's Disease and Restless Legs Syndrome |
WO2011101644A1 (fr) | 2010-02-18 | 2011-08-25 | Centro Nacional De Investigaciones Oncologicas (Cnio) | Composés bicycliques destinés à être utilisés en tant qu'inhibiteurs de kinases |
WO2011123719A2 (fr) | 2010-03-31 | 2011-10-06 | Ironwood Pharmaceuticals, Inc. | Utilisation d'inhibiteurs de faah pour le traitement des douleurs abdominales, viscérales et pelviennes |
CA2798080C (fr) * | 2010-05-17 | 2020-08-25 | Incozen Therapeutics Pvt. Ltd. | Composes pyridiniques 3,5-disubstitues-3 h-imidazo [4,5-b] et composes pyridiniques 3,5-disubstitues [1,2,3]triazolo[4,5-b] en tant que modulateurs des proteines kinases |
JP2013536852A (ja) | 2010-09-03 | 2013-09-26 | ヤンセン ファーマシューティカ エヌ.ベー. | モノアシルグリセロールリパーゼ阻害剤としてのジ−アゼチジニルジアミド |
KR20140001206A (ko) | 2010-09-27 | 2014-01-06 | 얀센 파마슈티카 엔.브이. | 모노아실글리세롤 리파아제 억제제로서의 옥소피페라진-아제티딘 아미드 및 옥소다이아제핀-아제티딘 아미드 |
US8513423B2 (en) | 2010-10-22 | 2013-08-20 | Janssen Pharmaceutica, Nv | Piperidin-4-yl-azetidine diamides as monoacylglycerol lipase inhibitors |
BR112013009828A2 (pt) | 2010-10-22 | 2016-07-26 | Janssen Pharmaceutica Nv | diamidas de amino-pirrolidina-azetidina como inibidores de monoacilglicerol lipase |
JP2014076947A (ja) * | 2011-02-03 | 2014-05-01 | Dainippon Sumitomo Pharma Co Ltd | 2−オキシ置換8−オキソジヒドロプリン誘導体 |
MX2014003883A (es) * | 2011-09-30 | 2014-08-27 | Janssen Pharmaceutica Nv | Inhibidores de monoacilglicerol lipasa para el tratamiento de enfermedades metabolicas y transtornos relacionados. |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2816938B1 (fr) * | 2000-11-22 | 2003-01-03 | Sanofi Synthelabo | Derives de 3-aroylindole, leur procede de preparation et les compositions pharmaceutiques en contenant |
GB0100624D0 (en) * | 2001-01-10 | 2001-02-21 | Vernalis Res Ltd | Chemical compounds VII |
DE10247680B4 (de) * | 2002-10-12 | 2005-09-01 | Aventis Pharma Deutschland Gmbh | Neue bicyclische Inhibitoren der Hormon Sensitiven Lipase |
DE102004005172A1 (de) * | 2004-02-02 | 2005-08-18 | Aventis Pharma Deutschland Gmbh | Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase |
US7632837B2 (en) * | 2005-06-17 | 2009-12-15 | Bristol-Myers Squibb Company | Bicyclic heterocycles as cannabinoid-1 receptor modulators |
DE102005049954A1 (de) * | 2005-10-19 | 2007-05-31 | Sanofi-Aventis Deutschland Gmbh | Triazolopyridin-derivate als Inhibitoren von Lipasen und Phospholipasen |
-
2007
- 2007-04-18 FR FR0702809A patent/FR2915199B1/fr not_active Expired - Fee Related
-
2008
- 2008-04-16 AU AU2008257320A patent/AU2008257320A1/en not_active Abandoned
- 2008-04-16 MX MX2009011212A patent/MX2009011212A/es not_active Application Discontinuation
- 2008-04-16 RU RU2009142431/04A patent/RU2009142431A/ru not_active Application Discontinuation
- 2008-04-16 JP JP2010503547A patent/JP2010524904A/ja active Pending
- 2008-04-16 BR BRPI0810440-9A2A patent/BRPI0810440A2/pt not_active IP Right Cessation
- 2008-04-16 CA CA002683929A patent/CA2683929A1/fr not_active Abandoned
- 2008-04-16 CN CN200880012545A patent/CN101668758A/zh active Pending
- 2008-04-16 EP EP08787961A patent/EP2146990A1/fr not_active Withdrawn
- 2008-04-16 WO PCT/FR2008/000532 patent/WO2008145839A1/fr active Application Filing
- 2008-04-16 KR KR1020097021591A patent/KR20090130057A/ko not_active Application Discontinuation
- 2008-04-17 TW TW097114018A patent/TW200901993A/zh unknown
- 2008-04-17 CL CL2008001104A patent/CL2008001104A1/es unknown
- 2008-04-18 AR ARP080101601A patent/AR066107A1/es unknown
- 2008-04-18 UY UY31032A patent/UY31032A1/es not_active Application Discontinuation
-
2009
- 2009-10-06 US US12/573,959 patent/US8080547B2/en not_active Expired - Fee Related
- 2009-10-11 IL IL201450A patent/IL201450A0/en unknown
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102459167B (zh) * | 2009-04-22 | 2015-04-01 | 詹森药业有限公司 | 作为单酰甘油脂肪酶抑制剂的氮杂环丁烷基二酰胺 |
Also Published As
Publication number | Publication date |
---|---|
CN101668758A (zh) | 2010-03-10 |
UY31032A1 (es) | 2008-11-28 |
MX2009011212A (es) | 2009-11-02 |
RU2009142431A (ru) | 2011-05-27 |
WO2008145839A8 (fr) | 2009-11-19 |
EP2146990A1 (fr) | 2010-01-27 |
WO2008145839A1 (fr) | 2008-12-04 |
IL201450A0 (en) | 2010-05-31 |
US20100041651A1 (en) | 2010-02-18 |
JP2010524904A (ja) | 2010-07-22 |
CL2008001104A1 (es) | 2009-01-16 |
AU2008257320A1 (en) | 2008-12-04 |
TW200901993A (en) | 2009-01-16 |
AR066107A1 (es) | 2009-07-22 |
KR20090130057A (ko) | 2009-12-17 |
BRPI0810440A2 (pt) | 2014-10-14 |
US8080547B2 (en) | 2011-12-20 |
FR2915199A1 (fr) | 2008-10-24 |
CA2683929A1 (fr) | 2008-12-04 |
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Effective date: 20121228 |