UY31032A1 - Derivados de triazolopiridin-carboxamidas y triazolopirimidin-carboxinamidas, su preparacion y su aplicacion en terapeutica - Google Patents

Derivados de triazolopiridin-carboxamidas y triazolopirimidin-carboxinamidas, su preparacion y su aplicacion en terapeutica

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Publication number
UY31032A1
UY31032A1 UY31032A UY31032A UY31032A1 UY 31032 A1 UY31032 A1 UY 31032A1 UY 31032 A UY31032 A UY 31032A UY 31032 A UY31032 A UY 31032A UY 31032 A1 UY31032 A1 UY 31032A1
Authority
UY
Uruguay
Prior art keywords
preparation
derivatives
triazolopirimidin
triazolopiridin
carboxinamids
Prior art date
Application number
UY31032A
Other languages
English (en)
Inventor
Even Luc
Hoornaert Christian
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of UY31032A1 publication Critical patent/UY31032A1/es

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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Abstract

Se divulgan derivados de triazolopiridin-carboxinamidas y triazolo-pirimidin-carboximidas, de la formula general (I) en la que los sustituyentes, índices y radicales son tales como se especifican en la invencion; los procedimientos para su preparacion y sus aplicaciones terapéuticas.
UY31032A 2007-04-18 2008-04-18 Derivados de triazolopiridin-carboxamidas y triazolopirimidin-carboxinamidas, su preparacion y su aplicacion en terapeutica UY31032A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0702809A FR2915199B1 (fr) 2007-04-18 2007-04-18 Derives de triazolopyridine-carboxamides et triazolopyrimidine-carboxamides, leur preparation et leur application en therapeutique.

Publications (1)

Publication Number Publication Date
UY31032A1 true UY31032A1 (es) 2008-11-28

Family

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Application Number Title Priority Date Filing Date
UY31032A UY31032A1 (es) 2007-04-18 2008-04-18 Derivados de triazolopiridin-carboxamidas y triazolopirimidin-carboxinamidas, su preparacion y su aplicacion en terapeutica

Country Status (17)

Country Link
US (1) US8080547B2 (es)
EP (1) EP2146990A1 (es)
JP (1) JP2010524904A (es)
KR (1) KR20090130057A (es)
CN (1) CN101668758A (es)
AR (1) AR066107A1 (es)
AU (1) AU2008257320A1 (es)
BR (1) BRPI0810440A2 (es)
CA (1) CA2683929A1 (es)
CL (1) CL2008001104A1 (es)
FR (1) FR2915199B1 (es)
IL (1) IL201450A0 (es)
MX (1) MX2009011212A (es)
RU (1) RU2009142431A (es)
TW (1) TW200901993A (es)
UY (1) UY31032A1 (es)
WO (1) WO2008145839A1 (es)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2915198B1 (fr) * 2007-04-18 2009-12-18 Sanofi Aventis Derives de triazolopyridine-carboxamides et triazolopyridine -carboxamides, leur preparation et leur application en therapeutique.
BR122013027950A2 (pt) * 2008-12-24 2019-12-10 BIAL PORTELA & Cª S A compostos farmacêuticos
CN102459255A (zh) * 2009-04-22 2012-05-16 詹森药业有限公司 作为单酰甘油脂肪酶抑制剂的氮杂环丁烷基二酰胺
US8435977B2 (en) 2009-04-22 2013-05-07 Janssen Pharmaceutica, Nv Heteroaromatic and aromatic piperazinyl azetidinyl amides as monoacylglycerol lipase inhibitors
PT2421852E (pt) * 2009-04-22 2014-07-31 Janssen Pharmaceutica Nv Amidas de piperazinil azetidinil heteroaromáticas e aromáticas como inibidoras da lipase de monoacilglicerol
TW201103914A (en) * 2009-04-22 2011-02-01 Janssen Pharmaceutica Nv Heteroaromatic and aromatic piperazinyl azetidinyl amides as monoacylglycerol lipase inhibitors
WO2011030798A1 (ja) 2009-09-09 2011-03-17 大日本住友製薬株式会社 ８－オキソジヒドロプリン誘導体
WO2011085216A2 (en) 2010-01-08 2011-07-14 Ironwood Pharmaceuticals, Inc. Use of faah inhibitors for treating parkinson's disease and restless legs syndrome
SG183361A1 (en) 2010-02-18 2012-09-27 Ct Nac Investigaciones Oncologicas Cnio Triazolo [4, 5 - b] pyridin derivatives
US20130224151A1 (en) 2010-03-31 2013-08-29 United States Of America Use of FAAH Inhibitors for Treating Abdominal, Visceral and Pelvic Pain
JP5960688B2 (ja) 2010-05-17 2016-08-02 インコゼン セラピューティクス プライベート リミテッド プロテインキナーゼ調節物質としての新規３，５−二置換−３ｈ−［１，２，３］トリアゾロ［４，５−ｂ］ピリジン化合物
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AR066107A1 (es) 2009-07-22
US8080547B2 (en) 2011-12-20
BRPI0810440A2 (pt) 2014-10-14
EP2146990A1 (fr) 2010-01-27
WO2008145839A8 (fr) 2009-11-19
US20100041651A1 (en) 2010-02-18
TW200901993A (en) 2009-01-16
MX2009011212A (es) 2009-11-02
FR2915199A1 (fr) 2008-10-24
FR2915199B1 (fr) 2010-01-22
RU2009142431A (ru) 2011-05-27
KR20090130057A (ko) 2009-12-17
IL201450A0 (en) 2010-05-31
WO2008145839A1 (fr) 2008-12-04
CN101668758A (zh) 2010-03-10

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