BRPI0810440A2 - Derivados de triazolopiridina-carboxamidas e triazolopirimidina-carboxamidas, o respectivo preparo e a respectiva aplicação em terapêutica - Google Patents

Derivados de triazolopiridina-carboxamidas e triazolopirimidina-carboxamidas, o respectivo preparo e a respectiva aplicação em terapêutica

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Publication number
BRPI0810440A2
BRPI0810440A2 BRPI0810440-9A2A BRPI0810440A BRPI0810440A2 BR PI0810440 A2 BRPI0810440 A2 BR PI0810440A2 BR PI0810440 A BRPI0810440 A BR PI0810440A BR PI0810440 A2 BRPI0810440 A2 BR PI0810440A2
Authority
BR
Brazil
Prior art keywords
carboxamides
triazolopyridine
triazolopyrimidine
therapeutic
preparation
Prior art date
Application number
BRPI0810440-9A2A
Other languages
English (en)
Inventor
Luc Even
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of BRPI0810440A2 publication Critical patent/BRPI0810440A2/pt

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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BRPI0810440-9A2A 2007-04-18 2008-04-16 Derivados de triazolopiridina-carboxamidas e triazolopirimidina-carboxamidas, o respectivo preparo e a respectiva aplicação em terapêutica BRPI0810440A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0702809A FR2915199B1 (fr) 2007-04-18 2007-04-18 Derives de triazolopyridine-carboxamides et triazolopyrimidine-carboxamides, leur preparation et leur application en therapeutique.
PCT/FR2008/000532 WO2008145839A1 (fr) 2007-04-18 2008-04-16 Dérivés de triazolopyridine-carboxamides et triazolopyrimidine-carboxamides, leur préparation et leur application en thérapeutique

Publications (1)

Publication Number Publication Date
BRPI0810440A2 true BRPI0810440A2 (pt) 2014-10-14

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BRPI0810440-9A2A BRPI0810440A2 (pt) 2007-04-18 2008-04-16 Derivados de triazolopiridina-carboxamidas e triazolopirimidina-carboxamidas, o respectivo preparo e a respectiva aplicação em terapêutica

Country Status (17)

Country Link
US (1) US8080547B2 (pt)
EP (1) EP2146990A1 (pt)
JP (1) JP2010524904A (pt)
KR (1) KR20090130057A (pt)
CN (1) CN101668758A (pt)
AR (1) AR066107A1 (pt)
AU (1) AU2008257320A1 (pt)
BR (1) BRPI0810440A2 (pt)
CA (1) CA2683929A1 (pt)
CL (1) CL2008001104A1 (pt)
FR (1) FR2915199B1 (pt)
IL (1) IL201450A0 (pt)
MX (1) MX2009011212A (pt)
RU (1) RU2009142431A (pt)
TW (1) TW200901993A (pt)
UY (1) UY31032A1 (pt)
WO (1) WO2008145839A1 (pt)

Families Citing this family (17)

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FR2915198B1 (fr) * 2007-04-18 2009-12-18 Sanofi Aventis Derives de triazolopyridine-carboxamides et triazolopyridine -carboxamides, leur preparation et leur application en therapeutique.
WO2010074588A2 (en) * 2008-12-24 2010-07-01 BIAL - PORTELA & Cª, S.A. Pharmaceutical compounds
AU2010238732B2 (en) * 2009-04-22 2015-06-11 Janssen Pharmaceutica Nv Azetidinyl diamides as monoacylglycerol lipase inhibitors
TW201103914A (en) * 2009-04-22 2011-02-01 Janssen Pharmaceutica Nv Heteroaromatic and aromatic piperazinyl azetidinyl amides as monoacylglycerol lipase inhibitors
US8415341B2 (en) 2009-04-22 2013-04-09 Janssen Pharmaceutica, Nv Heteroaromatic and aromatic piperazinyl azetidinyl amides as monoacylglycerol lipase inhibitors
CA2759714A1 (en) * 2009-04-22 2010-10-28 Janssen Pharmaceutica Nv Heteroaromatic and aromatic piperazinyl azetidinyl amides as monoacylglycerol lipase inhibitors
EP2476682B1 (en) * 2009-09-09 2017-04-26 Sumitomo Dainippon Pharma Co., Ltd. 8-oxodihydropurine derivative
WO2011085216A2 (en) 2010-01-08 2011-07-14 Ironwood Pharmaceuticals, Inc. Use of faah inhibitors for treating parkinson's disease and restless legs syndrome
WO2011101644A1 (en) 2010-02-18 2011-08-25 Centro Nacional De Investigaciones Oncologicas (Cnio) Triazolo [4, 5 - b] pyridin derivatives
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DK2571878T3 (en) * 2010-05-17 2019-02-11 Indian Incozen Therapeutics Pvt Ltd Hitherto unknown 3,5-DISUBSTITUTED-3H-IMIDAZO [4,5-B] PYRIDINE AND 3,5- DISUBSTITUTED -3H- [1,2,3] TRIAZOL [4,5-B] PYRIDINE COMPOUNDS AS MODULATORS OF PROTEIN CHINES
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FR2915199A1 (fr) 2008-10-24
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