BRPI0907578A2 - derivados de 3-aminoalquil-1,3-di-hidro-2h-indol-2-ona, o respectivo preparo e a respectiva aplicação em terapêutica - Google Patents

derivados de 3-aminoalquil-1,3-di-hidro-2h-indol-2-ona, o respectivo preparo e a respectiva aplicação em terapêutica

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Publication number
BRPI0907578A2
BRPI0907578A2 BRPI0907578A BRPI0907578A BRPI0907578A2 BR PI0907578 A2 BRPI0907578 A2 BR PI0907578A2 BR PI0907578 A BRPI0907578 A BR PI0907578A BR PI0907578 A BRPI0907578 A BR PI0907578A BR PI0907578 A2 BRPI0907578 A2 BR PI0907578A2
Authority
BR
Brazil
Prior art keywords
indol
aminoalkyl
dihydro
derivatives
preparation
Prior art date
Application number
BRPI0907578A
Other languages
English (en)
Inventor
Pouzet Brigitte
Serradeil-Le Gal Claudine
Valette Gérard
Goullieux Laurent
Foulon Loïc
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of BRPI0907578A2 publication Critical patent/BRPI0907578A2/pt

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/32—Oxygen atoms
    • C07D209/34—Oxygen atoms in position 2
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BRPI0907578A 2008-02-19 2009-02-18 derivados de 3-aminoalquil-1,3-di-hidro-2h-indol-2-ona, o respectivo preparo e a respectiva aplicação em terapêutica BRPI0907578A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0800866A FR2927625B1 (fr) 2008-02-19 2008-02-19 Nouveaux derives de 3-aminoalkyl-1,3-dihydro-2h-indol-2-one, leur preparation et leur application en therapeutique
PCT/FR2009/000179 WO2009115685A1 (fr) 2008-02-19 2009-02-18 Nouveaux derives de 3-aminoalkyl-1,3-dihydro-2h-indol-2-one, leur preparation et leur application en therapeutique.

Publications (1)

Publication Number Publication Date
BRPI0907578A2 true BRPI0907578A2 (pt) 2019-09-24

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BRPI0907578A BRPI0907578A2 (pt) 2008-02-19 2009-02-18 derivados de 3-aminoalquil-1,3-di-hidro-2h-indol-2-ona, o respectivo preparo e a respectiva aplicação em terapêutica

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Country Link
US (1) US8362067B2 (pt)
EP (1) EP2265582B1 (pt)
JP (1) JP5602639B2 (pt)
KR (1) KR20100126401A (pt)
CN (1) CN102015642A (pt)
AR (1) AR070438A1 (pt)
AT (1) ATE540023T1 (pt)
AU (1) AU2009227111A1 (pt)
BR (1) BRPI0907578A2 (pt)
CA (1) CA2716035A1 (pt)
FR (1) FR2927625B1 (pt)
IL (1) IL207629A0 (pt)
MX (1) MX2010009092A (pt)
RU (1) RU2010138575A (pt)
WO (1) WO2009115685A1 (pt)

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Publication number Priority date Publication date Assignee Title
FR2927625B1 (fr) 2008-02-19 2010-03-12 Sanofi Aventis Nouveaux derives de 3-aminoalkyl-1,3-dihydro-2h-indol-2-one, leur preparation et leur application en therapeutique
AU2011272738B2 (en) 2010-07-01 2015-08-20 Azevan Pharmaceuticals, Inc. Methods for treating post traumatic stress disorder
BR112016022575A2 (pt) * 2014-03-28 2017-08-15 Azevan Pharmaceuticals Inc Composições e métodos para o tratamento de doenças neurodegenerativas
CN104592088B (zh) * 2015-01-05 2019-01-01 内蒙古工业大学 月桂酸催化制备3-胺烷基吲哚的方法
CN105061290B (zh) * 2015-08-28 2017-11-10 福建品派包装有限公司 一种吲哚酮类化合物的合成方法
CN105061291B (zh) * 2015-09-08 2017-08-04 江俞 一种杂稠环取代的吲哚酮类化合物的合成方法
CA3075759A1 (en) 2017-09-15 2019-03-21 Azevan Pharmaceuticals, Inc. Compositions and methods for treating brain injury
CN108675945B (zh) * 2018-06-22 2020-09-22 湖南科技大学 ((2-羟基苄基)胺基)苯基脲类化合物及其制备方法和用途

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Publication number Priority date Publication date Assignee Title
AU550845B2 (en) 1981-03-30 1986-04-10 Sumitomo Chemical Company, Limited Tetrahydrophthalimides and their starting compounds
FR2665441B1 (fr) 1990-07-31 1992-12-04 Sanofi Sa Derives de la n-sulfonyl indoline, leur preparation, les compositions pharmaceutiques en contenant.
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JP5125501B2 (ja) 2005-01-28 2013-01-23 大正製薬株式会社 １，３−ジヒドロ−２ｈ−インドール−２−オン化合物、及び芳香族複素環が縮合したピロリジン−２−オン化合物
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IL207629A0 (en) 2010-12-30
CN102015642A (zh) 2011-04-13
US8362067B2 (en) 2013-01-29
FR2927625B1 (fr) 2010-03-12
EP2265582B1 (fr) 2012-01-04
AU2009227111A1 (en) 2009-09-24
JP5602639B2 (ja) 2014-10-08
KR20100126401A (ko) 2010-12-01
FR2927625A1 (fr) 2009-08-21
CA2716035A1 (fr) 2009-09-24
MX2010009092A (es) 2011-09-21
RU2010138575A (ru) 2012-03-27
US20110059955A1 (en) 2011-03-10
EP2265582A1 (fr) 2010-12-29
WO2009115685A1 (fr) 2009-09-24
ATE540023T1 (de) 2012-01-15
AR070438A1 (es) 2010-04-07
JP2011512389A (ja) 2011-04-21

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Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2543 DE 01-10-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.