BRPI0507370A - derivados de indazol como inibidores da lipase sensìvel ao hormÈnio - Google Patents

derivados de indazol como inibidores da lipase sensìvel ao hormÈnio

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Publication number
BRPI0507370A
BRPI0507370A BRPI0507370-7A BRPI0507370A BRPI0507370A BR PI0507370 A BRPI0507370 A BR PI0507370A BR PI0507370 A BRPI0507370 A BR PI0507370A BR PI0507370 A BRPI0507370 A BR PI0507370A
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BR
Brazil
Prior art keywords
lipase inhibitors
sensitive lipase
indazole derivatives
hormone sensitive
derivatives
Prior art date
Application number
BRPI0507370-7A
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English (en)
Inventor
Gerhard Zoller
Stefan Petry
Guenter Mueller
Hubert Heuer
Karl-Heinz Baringhaus
Original Assignee
Sanofi Aventis Deutschland
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Publication date
Application filed by Sanofi Aventis Deutschland filed Critical Sanofi Aventis Deutschland
Publication of BRPI0507370A publication Critical patent/BRPI0507370A/pt

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    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61P3/06—Antihyperlipidemics
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    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
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    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

Abstract

DERIVADOS DE INDAZOL COMO INIBIDORES DA LIPASE SENSìVEL AO HORMÈNIO. A presente invenção refere-se aos derivados de indazol das fórmulas gerais (l) ou (ll) com os significados indicados na descrição, seus sais farmaceuticamente utilizáveis e seu uso como medicamentos.
BRPI0507370-7A 2004-02-02 2005-01-15 derivados de indazol como inibidores da lipase sensìvel ao hormÈnio BRPI0507370A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102004005172A DE102004005172A1 (de) 2004-02-02 2004-02-02 Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
PCT/EP2005/000365 WO2005073199A1 (de) 2004-02-02 2005-01-15 Indazolderivate als inhibitoren der hormon sensitiven lipase

Publications (1)

Publication Number Publication Date
BRPI0507370A true BRPI0507370A (pt) 2007-07-10

Family

ID=34801466

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0507370-7A BRPI0507370A (pt) 2004-02-02 2005-01-15 derivados de indazol como inibidores da lipase sensìvel ao hormÈnio

Country Status (27)

Country Link
US (2) US7528155B2 (pt)
EP (1) EP1713779B1 (pt)
JP (1) JP4714158B2 (pt)
KR (1) KR20060128958A (pt)
CN (1) CN1914180A (pt)
AR (1) AR047520A1 (pt)
AT (1) ATE505460T1 (pt)
AU (1) AU2005209366A1 (pt)
BR (1) BRPI0507370A (pt)
CA (1) CA2554524A1 (pt)
CR (1) CR8487A (pt)
DE (2) DE102004005172A1 (pt)
DO (1) DOP2005000011A (pt)
EC (1) ECSP066750A (pt)
HN (1) HN2005000039A (pt)
IL (1) IL176912A (pt)
MA (1) MA28338A1 (pt)
MY (1) MY143407A (pt)
NO (1) NO20063925L (pt)
NZ (1) NZ548872A (pt)
PE (1) PE20050690A1 (pt)
RU (1) RU2370491C2 (pt)
SG (1) SG149891A1 (pt)
TW (1) TW200536535A (pt)
UY (1) UY28735A1 (pt)
WO (1) WO2005073199A1 (pt)
ZA (1) ZA200605311B (pt)

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