CN1751041B - 3-取代的-2-(芳基烷基)-1-氮杂二环烷烃及其使用方法 - Google Patents

3-取代的-2-(芳基烷基)-1-氮杂二环烷烃及其使用方法 Download PDF

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Publication number
CN1751041B
CN1751041B CN2004800047360A CN200480004736A CN1751041B CN 1751041 B CN1751041 B CN 1751041B CN 2004800047360 A CN2004800047360 A CN 2004800047360A CN 200480004736 A CN200480004736 A CN 200480004736A CN 1751041 B CN1751041 B CN 1751041B
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Prior art keywords
pyridyl
methyl
oct
azabicyclo
azabicyclic
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Expired - Fee Related
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CN2004800047360A
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Chinese (zh)
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CN1751041A (zh
Inventor
A·A·马祖罗夫
J·克鲁茨克
苗蓝
A·S·西曼斯
T·Y·菲力普斯
J·D·施米特
C·H·米勒
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Gyre Therapeutics Inc
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Targacept Inc
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems
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    • A61K51/04—Organic compounds
    • A61K51/041—Heterocyclic compounds
    • A61K51/044—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K51/0455—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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CN2004800047360A 2003-02-21 2004-02-20 3-取代的-2-(芳基烷基)-1-氮杂二环烷烃及其使用方法 Expired - Fee Related CN1751041B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US10/372,642 US6953855B2 (en) 1998-12-11 2003-02-21 3-substituted-2(arylalkyl)-1-azabicycloalkanes and methods of use thereof
US10/372,642 2003-02-21
PCT/US2004/005044 WO2004076449A2 (en) 2003-02-21 2004-02-20 3-substituted-2(arylalkyl)-1-azabicycloalkanes and methods of use thereof

Related Child Applications (1)

Application Number Title Priority Date Filing Date
CNA2007101598898A Division CN101220026A (zh) 2003-02-21 2004-02-20 3-取代的-2-(芳基烷基)-1-氮杂二环烷烃及其使用方法

Publications (2)

Publication Number Publication Date
CN1751041A CN1751041A (zh) 2006-03-22
CN1751041B true CN1751041B (zh) 2010-04-28

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CN2004800047360A Expired - Fee Related CN1751041B (zh) 2003-02-21 2004-02-20 3-取代的-2-(芳基烷基)-1-氮杂二环烷烃及其使用方法
CNA2007101598898A Pending CN101220026A (zh) 2003-02-21 2004-02-20 3-取代的-2-(芳基烷基)-1-氮杂二环烷烃及其使用方法

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CNA2007101598898A Pending CN101220026A (zh) 2003-02-21 2004-02-20 3-取代的-2-(芳基烷基)-1-氮杂二环烷烃及其使用方法

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US (11) US6953855B2 (enExample)
EP (1) EP1594869B9 (enExample)
JP (3) JP4828407B2 (enExample)
KR (3) KR101098481B1 (enExample)
CN (2) CN1751041B (enExample)
AT (1) ATE381563T1 (enExample)
AU (1) AU2004215386B2 (enExample)
BR (1) BRPI0407708A (enExample)
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CY (1) CY1107175T1 (enExample)
DE (1) DE602004010787T2 (enExample)
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NZ (3) NZ541794A (enExample)
PL (3) PL395717A1 (enExample)
PT (1) PT1594869E (enExample)
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ZA (1) ZA200506515B (enExample)

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SE0400708D0 (sv) * 2004-03-22 2004-03-22 Aprea Ab New compounds and use thereof
RU2417225C2 (ru) 2004-03-25 2011-04-27 Мемори Фармасьютиклз Корпорейшн Индазолы, бензотиазолы, бензоизотиазолы, бензизоксазолы и их получение и применение
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AR049401A1 (es) 2004-06-18 2006-07-26 Novartis Ag Aza-biciclononanos
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