CN1717236A - 治疗移植排斥的方法 - Google Patents

治疗移植排斥的方法 Download PDF

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Publication number
CN1717236A
CN1717236A CNA2003801042374A CN200380104237A CN1717236A CN 1717236 A CN1717236 A CN 1717236A CN A2003801042374 A CNA2003801042374 A CN A2003801042374A CN 200380104237 A CN200380104237 A CN 200380104237A CN 1717236 A CN1717236 A CN 1717236A
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CN
China
Prior art keywords
alkyl
amino
methyl
alkoxy
alkylamino
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Pending
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CNA2003801042374A
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English (en)
Chinese (zh)
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P·S·钱格里安
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Pfizer Products Inc
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Pfizer Products Inc
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Transplantation (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CNA2003801042374A 2002-11-26 2003-11-17 治疗移植排斥的方法 Pending CN1717236A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US42978402P 2002-11-26 2002-11-26
US60/429,784 2002-11-26

Publications (1)

Publication Number Publication Date
CN1717236A true CN1717236A (zh) 2006-01-04

Family

ID=32393587

Family Applications (1)

Application Number Title Priority Date Filing Date
CNA2003801042374A Pending CN1717236A (zh) 2002-11-26 2003-11-17 治疗移植排斥的方法

Country Status (15)

Country Link
US (1) US7250420B2 (enExample)
EP (1) EP1572213A1 (enExample)
JP (1) JP2006509000A (enExample)
KR (1) KR20050086784A (enExample)
CN (1) CN1717236A (enExample)
AU (1) AU2003276591A1 (enExample)
BR (1) BR0316487A (enExample)
CA (1) CA2507392A1 (enExample)
MX (1) MXPA05005576A (enExample)
MY (1) MY137250A (enExample)
NZ (1) NZ539901A (enExample)
PL (1) PL378246A1 (enExample)
TW (1) TW200418482A (enExample)
WO (1) WO2004047843A1 (enExample)
ZA (1) ZA200503811B (enExample)

Cited By (2)

* Cited by examiner, † Cited by third party
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CN103896826A (zh) * 2012-12-26 2014-07-02 上海朴颐化学科技有限公司 氮保护的(3r,4r)-3-甲氨基-4-甲基哌啶的不对称合成方法、相关中间体及原料制备方法
CN107602569A (zh) * 2017-10-23 2018-01-19 上海博悦生物科技有限公司 一种新型吡咯并[2,3‑d]嘧啶化合物及其合成方法和用途

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Cited By (3)

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Publication number Priority date Publication date Assignee Title
CN103896826A (zh) * 2012-12-26 2014-07-02 上海朴颐化学科技有限公司 氮保护的(3r,4r)-3-甲氨基-4-甲基哌啶的不对称合成方法、相关中间体及原料制备方法
CN103896826B (zh) * 2012-12-26 2016-08-03 上海朴颐化学科技有限公司 氮保护的(3r,4r)-3-甲氨基-4-甲基哌啶的不对称合成方法、相关中间体及原料制备方法
CN107602569A (zh) * 2017-10-23 2018-01-19 上海博悦生物科技有限公司 一种新型吡咯并[2,3‑d]嘧啶化合物及其合成方法和用途

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