CN106170486B - 新吲唑甲酰胺、其制备方法、包含其的药物制剂及其用于制备药物的用途 - Google Patents

新吲唑甲酰胺、其制备方法、包含其的药物制剂及其用于制备药物的用途 Download PDF

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CN106170486B
CN106170486B CN201480075834.7A CN201480075834A CN106170486B CN 106170486 B CN106170486 B CN 106170486B CN 201480075834 A CN201480075834 A CN 201480075834A CN 106170486 B CN106170486 B CN 106170486B
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carboxamide
oxoethyl
pyridine
indazol
trifluoromethyl
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CN106170486A (zh
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U·博特
H·斯贝内切
N·施密特
A·罗特盖里
U·鲍默
S·灵
H·伊尔巴切
J·冈瑟
H·施托伊贝尔
M·兰格
M·沙弗尔
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Bayer Pharma AG
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CN201480075834.7A 2013-12-19 2014-12-16 新吲唑甲酰胺、其制备方法、包含其的药物制剂及其用于制备药物的用途 Active CN106170486B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP13198463.5 2013-12-19
EP13198463 2013-12-19
EP14189216.6 2014-10-16
EP14189216 2014-10-16
PCT/EP2014/077877 WO2015091426A1 (de) 2013-12-19 2014-12-16 Neue indazolcarboxamide, verfahren zu ihrer herstellung, pharmazeutische präparate die diese enthalten, sowie deren verwendung zur herstellung von arzneimitteln

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CN106170486A CN106170486A (zh) 2016-11-30
CN106170486B true CN106170486B (zh) 2019-01-15

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US (1) US9951086B2 (enrdf_load_stackoverflow)
EP (1) EP3083586B1 (enrdf_load_stackoverflow)
JP (1) JP6530406B2 (enrdf_load_stackoverflow)
KR (1) KR20160094381A (enrdf_load_stackoverflow)
CN (1) CN106170486B (enrdf_load_stackoverflow)
AP (1) AP2016009273A0 (enrdf_load_stackoverflow)
AU (1) AU2014364744B2 (enrdf_load_stackoverflow)
BR (1) BR112016013632B1 (enrdf_load_stackoverflow)
CA (1) CA2934137C (enrdf_load_stackoverflow)
CL (1) CL2016001579A1 (enrdf_load_stackoverflow)
CR (1) CR20160278A (enrdf_load_stackoverflow)
CU (1) CU20160087A7 (enrdf_load_stackoverflow)
CY (1) CY1120437T1 (enrdf_load_stackoverflow)
DK (1) DK3083586T3 (enrdf_load_stackoverflow)
DO (1) DOP2016000150A (enrdf_load_stackoverflow)
EA (1) EA032621B1 (enrdf_load_stackoverflow)
ES (1) ES2677996T3 (enrdf_load_stackoverflow)
HR (1) HRP20181107T1 (enrdf_load_stackoverflow)
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IL (1) IL246032B (enrdf_load_stackoverflow)
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SG (1) SG11201604685RA (enrdf_load_stackoverflow)
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UY (1) UY35907A (enrdf_load_stackoverflow)
WO (1) WO2015091426A1 (enrdf_load_stackoverflow)
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JP6479850B2 (ja) 2014-01-13 2019-03-06 アウリジーン ディスカバリー テクノロジーズ リミテッド Ｉｒａｋ４阻害剤としての二環式ヘテロシクリル誘導体
JO3705B1 (ar) 2014-11-26 2021-01-31 Bayer Pharma AG إندازولات مستبدلة جديدة، عمليات لتحضيرها، مستحضرات دوائية تحتوي عليها واستخدامها في إنتاج أدوية
UY36660A (es) 2015-04-30 2016-11-30 Bayer Pharma AG Combinaciones de inhibidores de irak4
EP3195865A1 (de) 2016-01-25 2017-07-26 Bayer Pharma Aktiengesellschaft Kombinationen von irak4 inhibitoren und btk inhibitoren
HK1256242A1 (zh) 2015-08-04 2019-09-20 Rigel Pharmaceuticals, Inc. 吲哚化合物以及製備和使用該化合物的方法
WO2017108744A1 (de) * 2015-12-22 2017-06-29 Bayer Pharma Aktiengesellschaft Neue substituierte indazole, verfahren zu ihrer herstellung, pharmazeutische präparate die diese enthalten, sowie deren verwendung zur herstellung von arzneimitteln
CA3016364A1 (en) * 2016-03-03 2017-09-08 Bayer Pharma Aktiengesellschaft New 2-substituted indazoles, methods for producing same, pharmaceutical preparations that contain same, and use of same to produce drugs
EP3219329A1 (en) * 2016-03-17 2017-09-20 Bayer Pharma Aktiengesellschaft Combinations of copanlisib
PE20190172A1 (es) 2016-04-29 2019-02-01 Bayer Pharma AG Sintesis de indazoles
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