CU20160087A7 - Indazolcarboxamidas, procedimientos para su preparación, preparaciones farmacéuticas que las contienen - Google Patents

Indazolcarboxamidas, procedimientos para su preparación, preparaciones farmacéuticas que las contienen

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Publication number
CU20160087A7
CU20160087A7 CUP2016000087A CU20160087A CU20160087A7 CU 20160087 A7 CU20160087 A7 CU 20160087A7 CU P2016000087 A CUP2016000087 A CU P2016000087A CU 20160087 A CU20160087 A CU 20160087A CU 20160087 A7 CU20160087 A7 CU 20160087A7
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CU
Cuba
Prior art keywords
preparation
procedures
indazolcarboxamids
prevention
pharmaceutical preparations
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Application number
CUP2016000087A
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English (en)
Inventor
Ulrich Bothe
Holger Siebeneicher
Nicole Schmidt
Andrea Rotgeri
Ulf Bömer
Sven Ring
Horst Irlbacher
Judith Günther
Holger Steuber
Martin Lange
Martina Schäfer
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Bayer Pharma AG
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Publication date
Application filed by Bayer Pharma AG filed Critical Bayer Pharma AG
Publication of CU20160087A7 publication Critical patent/CU20160087A7/es

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    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
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    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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  • Chemical & Material Sciences (AREA)
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  • Pharmacology & Pharmacy (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

La presente solicitud se refiere a nuevos indazoles 6—sustituidos con cadena lateral de carboxamida, de fórmula general (I), ESPACIO PARA LA FÓRMULA y a procedimientos para su preparación. Los compuestos de la fórmula (I) son útiles para el tratamiento y/o la prevención de enfermedades, así como su uso para la preparación de medicamentos para el tratamiento y/o la prevención de enfermedades, en especial para el tratamiento y/o la prevención de endometriosis, linfomas, degeneración macular, EPOC y psoriasis.
CUP2016000087A 2013-12-19 2016-06-15 Indazolcarboxamidas, procedimientos para su preparación, preparaciones farmacéuticas que las contienen CU20160087A7 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP13198463 2013-12-19
EP14189216 2014-10-16
PCT/EP2014/077877 WO2015091426A1 (de) 2013-12-19 2014-12-16 Neue indazolcarboxamide, verfahren zu ihrer herstellung, pharmazeutische präparate die diese enthalten, sowie deren verwendung zur herstellung von arzneimitteln

Publications (1)

Publication Number Publication Date
CU20160087A7 true CU20160087A7 (es) 2017-03-03

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CUP2016000087A CU20160087A7 (es) 2013-12-19 2016-06-15 Indazolcarboxamidas, procedimientos para su preparación, preparaciones farmacéuticas que las contienen

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US (1) US9951086B2 (es)
EP (1) EP3083586B1 (es)
JP (1) JP6530406B2 (es)
KR (1) KR20160094381A (es)
CN (1) CN106170486B (es)
AP (1) AP2016009273A0 (es)
AU (1) AU2014364744B2 (es)
BR (1) BR112016013632B1 (es)
CA (1) CA2934137C (es)
CL (1) CL2016001579A1 (es)
CR (1) CR20160278A (es)
CU (1) CU20160087A7 (es)
CY (1) CY1120437T1 (es)
DK (1) DK3083586T3 (es)
DO (1) DOP2016000150A (es)
EA (1) EA032621B1 (es)
ES (1) ES2677996T3 (es)
HR (1) HRP20181107T1 (es)
HU (1) HUE038367T2 (es)
IL (1) IL246032B (es)
JO (1) JO3460B1 (es)
LT (1) LT3083586T (es)
MX (1) MX368413B (es)
PE (1) PE20160900A1 (es)
PH (1) PH12016501188A1 (es)
PL (1) PL3083586T3 (es)
PT (1) PT3083586T (es)
RS (1) RS57423B1 (es)
SG (1) SG11201604685RA (es)
SI (1) SI3083586T1 (es)
TW (1) TWI667233B (es)
UA (1) UA117392C2 (es)
UY (1) UY35907A (es)
WO (1) WO2015091426A1 (es)
ZA (1) ZA201603467B (es)

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JO3705B1 (ar) * 2014-11-26 2021-01-31 Bayer Pharma AG إندازولات مستبدلة جديدة، عمليات لتحضيرها، مستحضرات دوائية تحتوي عليها واستخدامها في إنتاج أدوية
TW201701879A (zh) 2015-04-30 2017-01-16 拜耳製藥公司 Ｉｒａｋ４抑制劑組合
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