UA117392C2 - Індазолкарбоксаміди, способи їх одержання, фармацевтичні препарати, що їх містять, і їх застосування для виготовлення лікарських засобів - Google Patents

Індазолкарбоксаміди, способи їх одержання, фармацевтичні препарати, що їх містять, і їх застосування для виготовлення лікарських засобів

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Publication number
UA117392C2
UA117392C2 UAA201607792A UAA201607792A UA117392C2 UA 117392 C2 UA117392 C2 UA 117392C2 UA A201607792 A UAA201607792 A UA A201607792A UA A201607792 A UAA201607792 A UA A201607792A UA 117392 C2 UA117392 C2 UA 117392C2
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Ukraine
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production
pharmaceutical preparations
producing medicaments
prophylaxis
treating
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UAA201607792A
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Ульріх Боте
Хольгер Зібенайхер
Ніколе Шмідт
Андреа Ротгері
Ульф Бьомер
Свен Рінг
Хорст Ірльбахер
Юдіт Гюнтер
Хольгер Штойбер
Мартін Ланге
Мартіна Шефер
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Байєр Фарма Акцієнгезелльшафт
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Publication of UA117392C2 publication Critical patent/UA117392C2/uk

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Abstract

Дана заявка стосується нових 6-заміщених індазолів, що містять карбоксамідний бічний ланцюг, способів їх одержання, їх застосування окремо або в комбінації для лікування і/або профілактики захворювань і їх застосування для виготовлення лікарських засобів для лікування і/або профілактики захворювань, зокрема для лікування і/або профілактики ендометріозу, лімфом, дегенерації жовтої плями, ХОЗЛ і псоріазу.
UAA201607792A 2013-12-19 2014-12-16 Індазолкарбоксаміди, способи їх одержання, фармацевтичні препарати, що їх містять, і їх застосування для виготовлення лікарських засобів UA117392C2 (uk)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP13198463 2013-12-19
EP14189216 2014-10-16
PCT/EP2014/077877 WO2015091426A1 (de) 2013-12-19 2014-12-16 Neue indazolcarboxamide, verfahren zu ihrer herstellung, pharmazeutische präparate die diese enthalten, sowie deren verwendung zur herstellung von arzneimitteln

Publications (1)

Publication Number Publication Date
UA117392C2 true UA117392C2 (uk) 2018-07-25

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UAA201607792A UA117392C2 (uk) 2013-12-19 2014-12-16 Індазолкарбоксаміди, способи їх одержання, фармацевтичні препарати, що їх містять, і їх застосування для виготовлення лікарських засобів

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US (1) US9951086B2 (uk)
EP (1) EP3083586B1 (uk)
JP (1) JP6530406B2 (uk)
KR (1) KR20160094381A (uk)
CN (1) CN106170486B (uk)
AP (1) AP2016009273A0 (uk)
AU (1) AU2014364744B2 (uk)
BR (1) BR112016013632B1 (uk)
CA (1) CA2934137C (uk)
CL (1) CL2016001579A1 (uk)
CR (1) CR20160278A (uk)
CU (1) CU20160087A7 (uk)
CY (1) CY1120437T1 (uk)
DK (1) DK3083586T3 (uk)
DO (1) DOP2016000150A (uk)
EA (1) EA032621B1 (uk)
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HR (1) HRP20181107T1 (uk)
HU (1) HUE038367T2 (uk)
IL (1) IL246032B (uk)
JO (1) JO3460B1 (uk)
LT (1) LT3083586T (uk)
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PE (1) PE20160900A1 (uk)
PH (1) PH12016501188A1 (uk)
PL (1) PL3083586T3 (uk)
PT (1) PT3083586T (uk)
RS (1) RS57423B1 (uk)
SG (1) SG11201604685RA (uk)
SI (1) SI3083586T1 (uk)
TW (1) TWI667233B (uk)
UA (1) UA117392C2 (uk)
UY (1) UY35907A (uk)
WO (1) WO2015091426A1 (uk)

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AU2015205348A1 (en) 2014-01-10 2016-07-28 Aurigene Discovery Technologies Limited Indazole compounds as IRAK4 inhibitors
NZ722019A (en) 2014-01-13 2022-07-01 Aurigene Discovery Tech Ltd Bicyclic heterocyclyl derivatives as irak4 inhibitors
JO3705B1 (ar) 2014-11-26 2021-01-31 Bayer Pharma AG إندازولات مستبدلة جديدة، عمليات لتحضيرها، مستحضرات دوائية تحتوي عليها واستخدامها في إنتاج أدوية
EP3195865A1 (de) 2016-01-25 2017-07-26 Bayer Pharma Aktiengesellschaft Kombinationen von irak4 inhibitoren und btk inhibitoren
UY36660A (es) 2015-04-30 2016-11-30 Bayer Pharma AG Combinaciones de inhibidores de irak4
ES2811136T3 (es) * 2015-08-04 2021-03-10 Rigel Pharmaceuticals Inc Compuestos de benzazol y métodos para obtener y usar los compuestos
WO2017108744A1 (de) * 2015-12-22 2017-06-29 Bayer Pharma Aktiengesellschaft Neue substituierte indazole, verfahren zu ihrer herstellung, pharmazeutische präparate die diese enthalten, sowie deren verwendung zur herstellung von arzneimitteln
US10435396B2 (en) 2016-03-03 2019-10-08 Bayer Pharma Aktiegesellschaft 2-substituted indazoles, methods for producing same, pharmaceutical preparations that contain same, and use of same to produce drugs
EP3219329A1 (en) * 2016-03-17 2017-09-20 Bayer Pharma Aktiengesellschaft Combinations of copanlisib
EA035867B1 (ru) * 2016-04-29 2020-08-24 Байер Фарма Акциенгезельшафт Синтез индазолов
WO2017186689A1 (en) 2016-04-29 2017-11-02 Bayer Pharma Aktiengesellschaft Synthesis of indazoles
AU2017256659B2 (en) * 2016-04-29 2021-05-27 Bayer Pharma Aktiengesellschaft Synthesis of indazoles
WO2017207340A1 (de) 2016-05-31 2017-12-07 Bayer Pharma Aktiengesellschaft Neue substituierte benzimidazole, verfahren zu ihrer herstellung, pharmazeutische präparate die diese enthalten, sowie deren verwendung zur herstellung von arzneimitteln
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