CN102686571B - 三环杂环化合物 - Google Patents

三环杂环化合物 Download PDF

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Publication number
CN102686571B
CN102686571B CN201080059932.3A CN201080059932A CN102686571B CN 102686571 B CN102686571 B CN 102686571B CN 201080059932 A CN201080059932 A CN 201080059932A CN 102686571 B CN102686571 B CN 102686571B
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isoxazole
base
phenyl
trifluoromethyl
methyl
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Expired - Fee Related
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Chinese (zh)
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CN102686571A (zh
Inventor
T.G.M.达尔
肖海云
S.H.沃特森
S.S.科
A.J.迪克曼
C.M.朗格维尼
J.达斯
R.J.彻尼
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Bristol Myers Squibb Co
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Bristol Myers Squibb Co
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CN201080059932.3A 2009-10-29 2010-10-29 三环杂环化合物 Expired - Fee Related CN102686571B (zh)

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US25599909P 2009-10-29 2009-10-29
US61/255,999 2009-10-29
PCT/US2010/054594 WO2011059784A1 (en) 2009-10-29 2010-10-29 Tricyclic heterocyclic compounds

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CN102686571B true CN102686571B (zh) 2015-11-25

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US (1) US9216972B2 (https=)
EP (3) EP2592071B1 (https=)
JP (1) JP5728487B2 (https=)
KR (1) KR20130036171A (https=)
CN (1) CN102686571B (https=)
AU (1) AU2010319879A1 (https=)
ES (1) ES2759949T3 (https=)
MX (1) MX336881B (https=)
WO (1) WO2011059784A1 (https=)

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US8580841B2 (en) 2008-07-23 2013-11-12 Arena Pharmaceuticals, Inc. Substituted 1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid derivatives useful in the treatment of autoimmune and inflammatory disorders
HRP20160890T1 (hr) 2008-08-27 2016-09-23 Arena Pharmaceuticals, Inc. Derivati supstituirane tricikličke kiseline kao agonisti s1p1-receptora korisni u liječenju autoimunih i upalnih poremećaja
JP5856980B2 (ja) 2010-01-27 2016-02-10 アリーナ ファーマシューティカルズ, インコーポレイテッド (R)−2−(7−(4−シクロペンチル−3−(トリフルオロメチル)ベンジルオキシ)−1,2,3,4−テトラヒドロシクロペンタ[b]インドール−3−イル)酢酸およびその塩の調製のためのプロセス
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