AU2010319879A1 - Tricyclic heterocyclic compounds - Google Patents

Tricyclic heterocyclic compounds Download PDF

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Publication number
AU2010319879A1
AU2010319879A1 AU2010319879A AU2010319879A AU2010319879A1 AU 2010319879 A1 AU2010319879 A1 AU 2010319879A1 AU 2010319879 A AU2010319879 A AU 2010319879A AU 2010319879 A AU2010319879 A AU 2010319879A AU 2010319879 A1 AU2010319879 A1 AU 2010319879A1
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Australia
Prior art keywords
isoxazol
mmol
phenyl
dihydronaphtho
trifluoromethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
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AU2010319879A
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English (en)
Inventor
Robert J. Cherney
Jagabandhu Das
T.G. Murali Dhar
Alaric J. Dyckman
Soo S. Ko
Charles M. Langevine
Scott Hunter Watterson
Hai-Yun Xiao
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Bristol Myers Squibb Co
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Bristol Myers Squibb Co
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Publication of AU2010319879A1 publication Critical patent/AU2010319879A1/en
Abandoned legal-status Critical Current

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    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
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AU2010319879A 2009-10-29 2010-10-29 Tricyclic heterocyclic compounds Abandoned AU2010319879A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US25599909P 2009-10-29 2009-10-29
US61/255,999 2009-10-29
PCT/US2010/054594 WO2011059784A1 (en) 2009-10-29 2010-10-29 Tricyclic heterocyclic compounds

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AU2010319879A1 true AU2010319879A1 (en) 2012-06-14

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US (1) US9216972B2 (https=)
EP (3) EP2592071B1 (https=)
JP (1) JP5728487B2 (https=)
KR (1) KR20130036171A (https=)
CN (1) CN102686571B (https=)
AU (1) AU2010319879A1 (https=)
ES (1) ES2759949T3 (https=)
MX (1) MX336881B (https=)
WO (1) WO2011059784A1 (https=)

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EA019252B1 (ru) 2008-07-23 2014-02-28 Арена Фармасьютикалз, Инк. ЗАМЕЩЕННЫЕ ПРОИЗВОДНЫЕ (1,2,3,4-ТЕТРАГИДРОЦИКЛОПЕНТА[b]ИНДОЛ-3-ИЛ)УКСУСНОЙ КИСЛОТЫ, ПРИМЕНИМЫЕ В ЛЕЧЕНИИ АУТОИММУННЫХ И ВОСПАЛИТЕЛЬНЫХ РАССТРОЙСТВ
SI2342205T1 (sl) 2008-08-27 2016-09-30 Arena Pharmaceuticals, Inc. Substituirani triciklični kislinski derivati kot agonisti S1P1 receptorja, uporabni v zdravljenju avtoimunskih in vnetnih obolenj
SG10201906876PA (en) 2010-01-27 2019-09-27 Arena Pharm Inc Processes for the preparation of (r)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid and salts thereof
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