CL2013001340A1 - Compuestos derivados de isoindol-amida, pirrolo-piridin-amida y pirrolo-pirimimidin-amida, inhibidores de nampt y rock; composicion farmaceutica; y metodo para tratar hiperetension, insuficiencia cardiaca cronica, aterosclerosis, asma, enfermedad de alzheimer, enfermedad de parkinson y glaucoma, entre otras enfermedades. - Google Patents
Compuestos derivados de isoindol-amida, pirrolo-piridin-amida y pirrolo-pirimimidin-amida, inhibidores de nampt y rock; composicion farmaceutica; y metodo para tratar hiperetension, insuficiencia cardiaca cronica, aterosclerosis, asma, enfermedad de alzheimer, enfermedad de parkinson y glaucoma, entre otras enfermedades.Info
- Publication number
- CL2013001340A1 CL2013001340A1 CL2013001340A CL2013001340A CL2013001340A1 CL 2013001340 A1 CL2013001340 A1 CL 2013001340A1 CL 2013001340 A CL2013001340 A CL 2013001340A CL 2013001340 A CL2013001340 A CL 2013001340A CL 2013001340 A1 CL2013001340 A1 CL 2013001340A1
- Authority
- CL
- Chile
- Prior art keywords
- amide
- pyrrolo
- disease
- pyrimimidin
- hyperetension
- Prior art date
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- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D407/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing three or more hetero rings
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- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
- C07D491/044—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
- C07D491/048—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being five-membered
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- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
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TW (1) | TW201238950A (es) |
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-
2011
- 2011-11-11 SG SG10202010119TA patent/SG10202010119TA/en unknown
- 2011-11-11 SG SG2013037643A patent/SG190819A1/en unknown
- 2011-11-11 RU RU2013126657/04A patent/RU2013126657A/ru not_active Application Discontinuation
- 2011-11-11 AU AU2011329233A patent/AU2011329233A1/en not_active Abandoned
- 2011-11-11 KR KR1020137015348A patent/KR20140009251A/ko not_active Application Discontinuation
- 2011-11-11 WO PCT/US2011/060425 patent/WO2012067965A1/en active Application Filing
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- 2011-11-11 EP EP11787996.5A patent/EP2640698A1/en not_active Withdrawn
- 2011-11-11 MX MX2013005454A patent/MX2013005454A/es unknown
- 2011-11-11 US US13/294,303 patent/US9302989B2/en active Active
- 2011-11-11 CN CN2011800647158A patent/CN103313968A/zh active Pending
- 2011-11-11 BR BR112013012078A patent/BR112013012078A2/pt not_active IP Right Cessation
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- 2011-11-11 UY UY0001033726A patent/UY33726A/es not_active Application Discontinuation
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Also Published As
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US20120122842A1 (en) | 2012-05-17 |
KR20140009251A (ko) | 2014-01-22 |
EP2640698A1 (en) | 2013-09-25 |
AR083855A1 (es) | 2013-03-27 |
US20160031880A1 (en) | 2016-02-04 |
WO2012067965A1 (en) | 2012-05-24 |
UY33726A (es) | 2012-06-29 |
CR20130267A (es) | 2013-10-04 |
ECSP13012993A (es) | 2014-01-31 |
BR112013012078A2 (pt) | 2019-09-24 |
SG190819A1 (en) | 2013-07-31 |
CO6761389A2 (es) | 2013-09-30 |
CA2816594A1 (en) | 2012-05-24 |
CN103313968A (zh) | 2013-09-18 |
RU2013126657A (ru) | 2014-12-27 |
AU2017200079A1 (en) | 2017-02-02 |
US10093624B2 (en) | 2018-10-09 |
DOP2013000106A (es) | 2013-10-15 |
US9302989B2 (en) | 2016-04-05 |
TW201238950A (en) | 2012-10-01 |
SG10201602857UA (en) | 2016-05-30 |
MX2013005454A (es) | 2013-06-24 |
IL225862A0 (en) | 2013-06-27 |
AU2011329233A1 (en) | 2013-05-23 |
SG10202010119TA (en) | 2020-11-27 |
PE20140913A1 (es) | 2014-08-22 |
JP6117104B2 (ja) | 2017-04-19 |
JP2017132792A (ja) | 2017-08-03 |
JP2013542265A (ja) | 2013-11-21 |
GT201300124A (es) | 2014-12-12 |
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