FR2733750B1 - Derives de l'acide gamma-oxo-alpha-(phenylmethyl)-5,6- dihydro-4h-thieno(3,4-c)pyrrole-5-butanoique, leur preparation et leur application en therapeutique - Google Patents
Derives de l'acide gamma-oxo-alpha-(phenylmethyl)-5,6- dihydro-4h-thieno(3,4-c)pyrrole-5-butanoique, leur preparation et leur application en therapeutiqueInfo
- Publication number
- FR2733750B1 FR2733750B1 FR9505260A FR9505260A FR2733750B1 FR 2733750 B1 FR2733750 B1 FR 2733750B1 FR 9505260 A FR9505260 A FR 9505260A FR 9505260 A FR9505260 A FR 9505260A FR 2733750 B1 FR2733750 B1 FR 2733750B1
- Authority
- FR
- France
- Prior art keywords
- butanoique
- thieno
- phenylmethyl
- pyrrole
- dihydro
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/02—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines
- C07D217/06—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines with the ring nitrogen atom acylated by carboxylic or carbonic acids, or with sulfur or nitrogen analogues thereof, e.g. carbamates
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Priority Applications (23)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9505260A FR2733750B1 (fr) | 1995-05-03 | 1995-05-03 | Derives de l'acide gamma-oxo-alpha-(phenylmethyl)-5,6- dihydro-4h-thieno(3,4-c)pyrrole-5-butanoique, leur preparation et leur application en therapeutique |
NZ307230A NZ307230A (en) | 1995-05-03 | 1996-04-12 | Furo[3,4-c]pyrrole, isoindole or thieno[3,4-c]pyrrole derivatives and medicaments |
CZ973466A CZ346697A3 (cs) | 1995-05-03 | 1996-04-12 | Deriváty azacykloalkanů, způsob jejich přípravy a farmaceutické kompozice tyto deriváty obsahující |
BR9608309A BR9608309A (pt) | 1995-05-03 | 1996-04-12 | Derivados de azacicloalcanos dua preparação e suas aplicações em terapêutica |
KR1019970707802A KR19990008276A (ko) | 1995-05-03 | 1996-04-12 | 아자시클로알칸 유도체, 그것의 제법 및 그것의 치료에의 이용 |
US08/945,576 US5869518A (en) | 1995-05-03 | 1996-04-12 | Azacycloalkane derivatives, their preparation and their application in therapy |
HU9903886A HUP9903886A3 (en) | 1995-05-03 | 1996-04-12 | Azacycloalcane derivatives, preparation thereof and their applications in therapy |
EP96913576A EP0823912A1 (fr) | 1995-05-03 | 1996-04-12 | Derives d'azacycloalcanes, leur preparation et leurs applications en therapeutique |
CA002220015A CA2220015A1 (fr) | 1995-05-03 | 1996-04-12 | Derives d'azacycloalcanes, leur preparation et leurs applications en therapeutique |
SK1478-97A SK147897A3 (en) | 1995-05-03 | 1996-04-12 | Azacycloalcane derivatives, preparation thereof and their applications in therapy |
AU56520/96A AU699120B2 (en) | 1995-05-03 | 1996-04-12 | Azacycloalcane derivatives, their preparation and their applications in therapy |
JP8533065A JPH11504913A (ja) | 1995-05-03 | 1996-04-12 | アザシクロアルカン誘導体、その製造および治療への適用 |
TR97/01287T TR199701287T1 (xx) | 1995-05-03 | 1996-04-12 | Azasikloalkan t�revleri, haz�rlan��lar� ve terapideki uygulamalar�. |
PCT/FR1996/000555 WO1996034870A1 (fr) | 1995-05-03 | 1996-04-12 | Derives d'azacycloalcanes, leur preparation et leurs applications en therapeutique |
PL96323177A PL323177A1 (en) | 1995-05-03 | 1996-04-12 | Azacycloalcane derivatives, method of obtaining them and their application for therapeutic purposes |
EE9700288A EE9700288A (et) | 1995-05-03 | 1996-04-12 | Asatsükloalkaani derivaadid, nende valmistamine ja kasutamine ravis |
IL11811996A IL118119A0 (en) | 1995-05-03 | 1996-05-02 | Azacycloalkane derivatives their preparation and their application in therapy |
CO96021765A CO4750652A1 (es) | 1995-05-03 | 1996-05-02 | Derivados de azacicloalcanos, su preparacion y sus aplica- ciones en terapeutica |
AR33637996A AR001838A1 (es) | 1995-05-03 | 1996-05-02 | Derivados de azacicloal canos utiles para el tratamiento de la obesidad diabetes e hiperglucemia procedimiento para prepararlos composiciones farmacéuticas que los contienen y aplicación de dichos derivados en la preparación de dichas composiciones |
ZA963485A ZA963485B (en) | 1995-05-03 | 1996-05-02 | Azacycloalkane derivatives, their preparation and their application in therapy |
MXPA/A/1997/008322A MXPA97008322A (en) | 1995-05-03 | 1997-10-29 | Derivatives of aza cicloalcano, its preparation and its applications in tera |
NO975020A NO975020L (no) | 1995-05-03 | 1997-10-31 | Azacykloalkanderivater, fremstilling derav og deres anvendelse i terapi |
BG102015A BG102015A (en) | 1995-05-03 | 1997-11-03 | Azacycloalkane derivatives, their preparation and application in therapy |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9505260A FR2733750B1 (fr) | 1995-05-03 | 1995-05-03 | Derives de l'acide gamma-oxo-alpha-(phenylmethyl)-5,6- dihydro-4h-thieno(3,4-c)pyrrole-5-butanoique, leur preparation et leur application en therapeutique |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2733750A1 FR2733750A1 (fr) | 1996-11-08 |
FR2733750B1 true FR2733750B1 (fr) | 1997-06-13 |
Family
ID=9478644
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR9505260A Expired - Fee Related FR2733750B1 (fr) | 1995-05-03 | 1995-05-03 | Derives de l'acide gamma-oxo-alpha-(phenylmethyl)-5,6- dihydro-4h-thieno(3,4-c)pyrrole-5-butanoique, leur preparation et leur application en therapeutique |
Country Status (22)
Country | Link |
---|---|
US (1) | US5869518A (fr) |
EP (1) | EP0823912A1 (fr) |
JP (1) | JPH11504913A (fr) |
KR (1) | KR19990008276A (fr) |
AR (1) | AR001838A1 (fr) |
AU (1) | AU699120B2 (fr) |
BG (1) | BG102015A (fr) |
BR (1) | BR9608309A (fr) |
CA (1) | CA2220015A1 (fr) |
CO (1) | CO4750652A1 (fr) |
CZ (1) | CZ346697A3 (fr) |
EE (1) | EE9700288A (fr) |
FR (1) | FR2733750B1 (fr) |
HU (1) | HUP9903886A3 (fr) |
IL (1) | IL118119A0 (fr) |
NO (1) | NO975020L (fr) |
NZ (1) | NZ307230A (fr) |
PL (1) | PL323177A1 (fr) |
SK (1) | SK147897A3 (fr) |
TR (1) | TR199701287T1 (fr) |
WO (1) | WO1996034870A1 (fr) |
ZA (1) | ZA963485B (fr) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1998040385A1 (fr) * | 1997-03-07 | 1998-09-17 | Novo Nordisk A/S | DERIVES DE 4,5,6,7-TETRAHYDRO-THIENO[3,2-c]PYRIDINE, LEUR PREPARATION ET LEUR UTILISATION |
US6177443B1 (en) | 1997-03-07 | 2001-01-23 | Novo Nordisk A/S | 4,5,6,7-tetrahydro-thieno[3, 2-C]pyridine derivatives, their preparation and use |
AU2610499A (en) * | 1998-03-06 | 1999-09-20 | Novo Nordisk A/S | 4,5,6,7-tetrahydro-thieno(3,2-c)pyridine derivatives |
FR2777566B1 (fr) | 1998-04-15 | 2003-02-21 | Synthelabo | Derives d'azacycloalcanes, leur preparation et leur application en therapeutique |
FR2779428B1 (fr) * | 1998-06-03 | 2001-05-18 | Synthelabo | Derives d'oxo-azacycloalcanes, leurs preparations et leurs applications en therapeutique |
US6090797A (en) * | 1998-09-02 | 2000-07-18 | Novo Nordisk A/S | 4,5,6,7-tetrahydro-thieno(2,3-C)pyridine derivatives |
AU5154699A (en) * | 1998-09-02 | 2000-03-27 | Novo Nordisk A/S | 4,5,6,7-tetrahydro-thieno(2,3-c)pyridine derivatives |
FR2793411B1 (fr) * | 1999-05-11 | 2001-06-29 | Synthelabo | Utilisation de derives de l'acide succinique pour obtenir un medicament destine au traitement de l'inflammation |
ATE257480T1 (de) * | 1999-09-30 | 2004-01-15 | Pfizer Prod Inc | Bicyclische pyrrolylamide als glycogenphosphorylase-inhibitoren |
US6797820B2 (en) | 1999-12-17 | 2004-09-28 | Vicuron Pharmaceuticals Inc. | Succinate compounds, compositions and methods of use and preparation |
DK1406893T3 (da) * | 2001-06-15 | 2007-08-06 | Vicuron Pharm Inc | Bicykliske pyrrolidinforbindelser |
AR036053A1 (es) | 2001-06-15 | 2004-08-04 | Versicor Inc | Compuestos de n-formil-hidroxilamina, un proceso para su preparacion y composiciones farmaceuticas |
US20100113664A1 (en) * | 2008-06-11 | 2010-05-06 | Ferro Corporation | Asymmetric Cyclic Diester Compounds |
US20090312470A1 (en) * | 2008-06-11 | 2009-12-17 | Ferro Corporation | Asymmetric Cyclic Diester Compounds |
CA2739740A1 (fr) * | 2008-10-24 | 2010-04-29 | Gruenenthal Gmbh | 4,5,6,7-tetrahydrothienopyridines substituees, comme modulateurs des kcnq2/3 pour le traitement de la douleur, de l'epilepsie et de l'incontinence urinaire |
SG10201602857UA (en) | 2010-11-15 | 2016-05-30 | Abbvie Inc | NAMPT And Rock Inhibitors |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3190950A (en) * | 1961-03-13 | 1965-06-22 | Acf Ind Inc | Pictorial position display |
US3706810A (en) * | 1970-09-15 | 1972-12-19 | American Cyanamid Co | N-morpholinoalkyl-thieno(3,2-b)pyrrole-5-carboxamides |
ZA821020B (en) * | 1981-02-18 | 1983-10-26 | Thomae Gmbh Dr K | Azepine derivatives, process for their preparation and pharmaceutical compositions thereof |
FR2537974A1 (fr) * | 1982-12-16 | 1984-06-22 | Adir | Nouveaux derives de thieno (2,3-b) pyrrole, leur procede de preparation et les compositions pharmaceutiques les renfermant |
FR2571723B1 (fr) * | 1984-10-12 | 1988-08-26 | Lipha | Derives de thieno et furo-(2,3-c) pyrroles, procedes de preparation et medicaments les contenant |
FR2652579B1 (fr) * | 1989-10-02 | 1992-01-24 | Sanofi Sa | Derives d'hydroxy-2 thiophene et furanne condenses avec un cycle azote, sur procede de preparation et leur application en therapeutique. |
FR2676446B1 (fr) * | 1991-05-17 | 1993-08-06 | Rhone Poulenc Rorer Sa | Nouveaux derives du thiopyranopyrrole, leur preparation et les compositions pharmaceutiques qui les contiennent. |
EP0599697A1 (fr) * | 1992-11-24 | 1994-06-01 | Synthelabo | Dérivés de pyrrole, leur préparation et leur application en thérapeutique |
FR2719844B1 (fr) * | 1994-05-10 | 1996-06-07 | Synthelabo | Dérivés de 5,6-dihydro-4h-thiéno[3,4-c]pyrrole, leur préparation et leur application en thérapeutique. |
-
1995
- 1995-05-03 FR FR9505260A patent/FR2733750B1/fr not_active Expired - Fee Related
-
1996
- 1996-04-12 CZ CZ973466A patent/CZ346697A3/cs unknown
- 1996-04-12 SK SK1478-97A patent/SK147897A3/sk unknown
- 1996-04-12 PL PL96323177A patent/PL323177A1/xx unknown
- 1996-04-12 NZ NZ307230A patent/NZ307230A/en unknown
- 1996-04-12 KR KR1019970707802A patent/KR19990008276A/ko not_active Application Discontinuation
- 1996-04-12 AU AU56520/96A patent/AU699120B2/en not_active Ceased
- 1996-04-12 CA CA002220015A patent/CA2220015A1/fr not_active Abandoned
- 1996-04-12 JP JP8533065A patent/JPH11504913A/ja active Pending
- 1996-04-12 WO PCT/FR1996/000555 patent/WO1996034870A1/fr not_active Application Discontinuation
- 1996-04-12 HU HU9903886A patent/HUP9903886A3/hu unknown
- 1996-04-12 EP EP96913576A patent/EP0823912A1/fr not_active Withdrawn
- 1996-04-12 US US08/945,576 patent/US5869518A/en not_active Expired - Fee Related
- 1996-04-12 TR TR97/01287T patent/TR199701287T1/xx unknown
- 1996-04-12 BR BR9608309A patent/BR9608309A/pt not_active Application Discontinuation
- 1996-04-12 EE EE9700288A patent/EE9700288A/xx unknown
- 1996-05-02 ZA ZA963485A patent/ZA963485B/xx unknown
- 1996-05-02 CO CO96021765A patent/CO4750652A1/es unknown
- 1996-05-02 AR AR33637996A patent/AR001838A1/es unknown
- 1996-05-02 IL IL11811996A patent/IL118119A0/xx unknown
-
1997
- 1997-10-31 NO NO975020A patent/NO975020L/no unknown
- 1997-11-03 BG BG102015A patent/BG102015A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
ZA963485B (en) | 1996-11-25 |
NO975020L (no) | 1998-01-05 |
BR9608309A (pt) | 1999-01-26 |
EE9700288A (et) | 1998-04-15 |
PL323177A1 (en) | 1998-03-16 |
HUP9903886A2 (hu) | 2000-03-28 |
US5869518A (en) | 1999-02-09 |
SK147897A3 (en) | 1998-05-06 |
WO1996034870A1 (fr) | 1996-11-07 |
CA2220015A1 (fr) | 1996-11-07 |
AR001838A1 (es) | 1997-12-10 |
FR2733750A1 (fr) | 1996-11-08 |
TR199701287T1 (xx) | 1998-03-21 |
MX9708322A (es) | 1998-06-28 |
NO975020D0 (no) | 1997-10-31 |
AU5652096A (en) | 1996-11-21 |
IL118119A0 (en) | 1996-09-12 |
AU699120B2 (en) | 1998-11-19 |
BG102015A (en) | 1998-08-31 |
KR19990008276A (ko) | 1999-01-25 |
CZ346697A3 (cs) | 1998-02-18 |
EP0823912A1 (fr) | 1998-02-18 |
CO4750652A1 (es) | 1999-03-31 |
HUP9903886A3 (en) | 2000-04-28 |
NZ307230A (en) | 1998-11-25 |
JPH11504913A (ja) | 1999-05-11 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
TP | Transmission of property | ||
ST | Notification of lapse |
Effective date: 20060131 |