CH694241A5 - Kristalle aus einem pharmazeutisch akzeptablen Salz von Citalopram. - Google Patents

Kristalle aus einem pharmazeutisch akzeptablen Salz von Citalopram. Download PDF

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Publication number
CH694241A5
CH694241A5 CH01422/03A CH14222003A CH694241A5 CH 694241 A5 CH694241 A5 CH 694241A5 CH 01422/03 A CH01422/03 A CH 01422/03A CH 14222003 A CH14222003 A CH 14222003A CH 694241 A5 CH694241 A5 CH 694241A5
Authority
CH
Switzerland
Prior art keywords
citalopram
crystals
temperature
range
pharmaceutically acceptable
Prior art date
Application number
CH01422/03A
Other languages
German (de)
English (en)
Inventor
Ken Liljegren
Sven Wagner
Per Holm
Ole Nielsen
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26068858&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CH694241(A5) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of CH694241A5 publication Critical patent/CH694241A5/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4866—Organic macromolecular compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CH01422/03A 2000-08-10 2001-08-08 Kristalle aus einem pharmazeutisch akzeptablen Salz von Citalopram. CH694241A5 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA200001202 2000-08-10
DKPA200001614 2000-10-27

Publications (1)

Publication Number Publication Date
CH694241A5 true CH694241A5 (de) 2004-10-15

Family

ID=26068858

Family Applications (2)

Application Number Title Priority Date Filing Date
CH01469/01A CH694242A5 (de) 2000-08-10 2001-08-08 Citalopram enthaltende pharmazeutische Zusammensetzung.
CH01422/03A CH694241A5 (de) 2000-08-10 2001-08-08 Kristalle aus einem pharmazeutisch akzeptablen Salz von Citalopram.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CH01469/01A CH694242A5 (de) 2000-08-10 2001-08-08 Citalopram enthaltende pharmazeutische Zusammensetzung.

Country Status (34)

Country Link
EP (1) EP1318805A2 (xx)
JP (1) JP2003531153A (xx)
KR (1) KR20030024833A (xx)
CN (1) CN1446089A (xx)
AR (1) AR030095A1 (xx)
AT (1) AT5744U1 (xx)
AU (2) AU2001100198B4 (xx)
BE (1) BE1013559A6 (xx)
BG (1) BG107578A (xx)
BR (1) BR0113250A (xx)
CA (1) CA2353693C (xx)
CH (2) CH694242A5 (xx)
CZ (1) CZ2003397A3 (xx)
DE (2) DE10139115A1 (xx)
EA (1) EA200300247A1 (xx)
ES (1) ES2172481B2 (xx)
FI (1) FI5176U1 (xx)
FR (1) FR2812811B1 (xx)
GB (1) GB2368014B (xx)
GR (1) GR1004193B (xx)
HR (1) HRP20030054A2 (xx)
HU (1) HUP0103071A3 (xx)
IE (1) IES20010693A2 (xx)
IL (1) IL154050A0 (xx)
IS (1) IS6021A (xx)
IT (1) ITMI20011637A1 (xx)
MX (1) MXPA03000837A (xx)
NL (1) NL1018741C1 (xx)
NO (1) NO20013891L (xx)
NZ (1) NZ523785A (xx)
PL (1) PL359824A1 (xx)
SK (1) SK2842003A3 (xx)
WO (1) WO2001080619A2 (xx)
YU (1) YU9003A (xx)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IS6021A (is) * 2000-08-10 2001-10-20 H. Lundbeck A/S Lyfjasamsetningar sem innihalda sítalópram
AU2001100195B4 (en) * 2001-01-05 2001-12-20 H Lundbeck As Pharmaceutical composition containing citalopram.
GB0206708D0 (en) * 2002-03-21 2002-05-01 Cipla Ltd Pharmaceutical salts
US6812355B2 (en) 2002-10-22 2004-11-02 Sekhsaria Chemicals Limited Process for the manufacture of citalopram hydrobromide from 5-bromophthalide
PT1578738E (pt) * 2002-12-23 2008-04-11 Lundbeck & Co As H Bromidrato de escitalopram e um método para a sua preparação
WO2004103361A2 (en) * 2003-05-20 2004-12-02 Ranbaxy Laboratories Limited A pharmaceutical dosage form of citalopram
HU227491B1 (en) * 2003-11-25 2011-07-28 Egis Gyogyszergyar Nyilvanosan Muekoedoe Reszvenytarsasag Tablet containing citalopram hydrogen bromide
WO2006038217A1 (en) * 2004-10-05 2006-04-13 Strides Acrolab Limited An improved drug delivery system of citalopram hydrobromide and process for producing the same
US7834201B2 (en) 2005-06-22 2010-11-16 H. Lundbeck A/S Crystalline base of escitalopram and orodispersible tablets comprising escitalopram base
CN100353939C (zh) * 2006-01-05 2007-12-12 昆明积大制药有限公司 含西酞普兰和环糊精的抗抑郁口服药用组合物
GB2446847B (en) * 2007-02-02 2012-02-22 Ubiquisys Ltd Location of Basestation
CN106389374A (zh) * 2015-08-03 2017-02-15 深圳信立泰药业股份有限公司 一种含有lcz696的药物组合物及其制备方法
WO2022153262A1 (en) * 2021-01-18 2022-07-21 Anton Frenkel Pharmaceutical dosage form
WO2024165628A1 (en) 2023-02-07 2024-08-15 Kinast Lasse An immediate-release oral pharmaceutical form of escitalopram or racemate thereof with increased api content

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US1358915A (en) * 1919-04-14 1920-11-16 Amici Domenico Aeroplane
GB1358915A (en) * 1971-09-13 1974-07-03 Merck & Co Inc Directly compressed tablet and composition therefor
GB1526331A (en) 1976-01-14 1978-09-27 Kefalas As Phthalanes
GB8419963D0 (en) 1984-08-06 1984-09-12 Lundbeck & Co As H Intermediate compound and method
GB8814057D0 (en) * 1988-06-14 1988-07-20 Lundbeck & Co As H New enantiomers & their isolation
US5296507A (en) * 1990-09-06 1994-03-22 H.Lundbeck A/S Treatment of cerbrovascular disorders
EP0714663A3 (en) * 1994-11-28 1997-01-15 Lilly Co Eli Potentiation of drug responses by serotonin 1A receptor antagonists
GB9714841D0 (en) * 1997-07-14 1997-09-17 Smithkline Beecham Plc Treatment method
GB2357762B (en) * 2000-03-13 2002-01-30 Lundbeck & Co As H Crystalline base of citalopram
US6977306B2 (en) 2000-05-02 2005-12-20 Sumitomo Chemical Company, Limited Citalopram hydrobromide crystal and method for crystallization thereof
IS6021A (is) * 2000-08-10 2001-10-20 H. Lundbeck A/S Lyfjasamsetningar sem innihalda sítalópram

Also Published As

Publication number Publication date
NO20013891L (no) 2002-02-11
ITMI20011637A1 (it) 2003-01-27
FI5176U1 (fi) 2001-12-27
GR20010100377A (el) 2002-09-06
AU2001100198A4 (en) 2001-08-16
HUP0103071A3 (en) 2002-12-28
AT5744U1 (de) 2002-11-25
CA2353693C (en) 2003-07-22
IES20010693A2 (en) 2002-07-10
WO2001080619A2 (en) 2001-11-01
GB2368014A (en) 2002-04-24
WO2001080619A3 (en) 2002-02-21
YU9003A (sh) 2006-05-25
NO20013891D0 (no) 2001-08-09
IL154050A0 (en) 2003-07-31
ES2172481B2 (es) 2004-08-01
ES2172481A1 (es) 2002-09-16
IS6021A (is) 2001-10-20
KR20030024833A (ko) 2003-03-26
AR030095A1 (es) 2003-08-13
NZ523785A (en) 2004-09-24
NL1018741C1 (nl) 2002-02-12
JP2003531153A (ja) 2003-10-21
DE20113195U1 (de) 2001-11-15
CH694242A5 (de) 2004-10-15
FR2812811B1 (fr) 2006-08-18
AU2001279591A1 (en) 2001-11-07
BR0113250A (pt) 2003-06-24
SK2842003A3 (en) 2003-09-11
HRP20030054A2 (en) 2005-02-28
CN1446089A (zh) 2003-10-01
GR1004193B (el) 2003-03-24
AU2001100198B4 (en) 2002-06-13
FR2812811A1 (fr) 2002-02-15
HU0103071D0 (en) 2001-10-28
EP1318805A2 (en) 2003-06-18
DE10139115A1 (de) 2002-03-28
BG107578A (bg) 2003-09-30
HUP0103071A2 (hu) 2002-05-29
GB2368014B (en) 2004-06-23
MXPA03000837A (es) 2003-06-06
BE1013559A6 (fr) 2002-03-05
PL359824A1 (en) 2004-09-06
ITMI20011637A0 (it) 2001-07-27
EA200300247A1 (ru) 2003-06-26
GB0118579D0 (en) 2001-09-19
CZ2003397A3 (cs) 2003-06-18
CA2353693A1 (en) 2002-01-22

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Legal Events

Date Code Title Description
PK Correction

Free format text: NAME DES VERTRETERS KORRIGIERT.

PFA Name/firm changed

Owner name: H. LUNDBECK A/S

Free format text: H. LUNDBECK A/S#9, OTTILIAVEJ#2500 VALBY-COPENHAGEN (DK) -TRANSFER TO- H. LUNDBECK A/S#9, OTTILIAVEJ#2500 VALBY-COPENHAGEN (DK)

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