CH623812A5 - Process for the preparation of 6,7-benzomorphane derivatives - Google Patents

Process for the preparation of 6,7-benzomorphane derivatives Download PDF

Info

Publication number
CH623812A5
CH623812A5 CH502175A CH502175A CH623812A5 CH 623812 A5 CH623812 A5 CH 623812A5 CH 502175 A CH502175 A CH 502175A CH 502175 A CH502175 A CH 502175A CH 623812 A5 CH623812 A5 CH 623812A5
Authority
CH
Switzerland
Prior art keywords
compound
formula
methyl
lower alkyl
hydrogen
Prior art date
Application number
CH502175A
Other languages
German (de)
English (en)
Inventor
Thomas Alfred Montzka
John Daniel Matiskella
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of CH623812A5 publication Critical patent/CH623812A5/de

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22Bridged ring systems
    • C07D221/26Benzomorphans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/56Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds
    • C07C45/562Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds with nitrogen as the only hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/587Unsaturated compounds containing a keto groups being part of a ring
    • C07C49/753Unsaturated compounds containing a keto groups being part of a ring containing ether groups, groups, groups, or groups
    • C07C49/755Unsaturated compounds containing a keto groups being part of a ring containing ether groups, groups, groups, or groups a keto group being part of a condensed ring system with two or three rings, at least one ring being a six-membered aromatic ring
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
CH502175A 1974-04-18 1975-04-18 Process for the preparation of 6,7-benzomorphane derivatives CH623812A5 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US46200774A 1974-04-18 1974-04-18

Publications (1)

Publication Number Publication Date
CH623812A5 true CH623812A5 (en) 1981-06-30

Family

ID=23834846

Family Applications (1)

Application Number Title Priority Date Filing Date
CH502175A CH623812A5 (en) 1974-04-18 1975-04-18 Process for the preparation of 6,7-benzomorphane derivatives

Country Status (23)

Country Link
JP (3) JPS6218552B2 (xx)
BE (1) BE828054A (xx)
CA (1) CA1040630A (xx)
CH (1) CH623812A5 (xx)
CS (1) CS199586B2 (xx)
DD (1) DD119787A5 (xx)
DE (1) DE2517220A1 (xx)
DK (2) DK155999C (xx)
FI (1) FI60564C (xx)
FR (1) FR2267774B1 (xx)
GB (1) GB1493420A (xx)
HU (1) HU173039B (xx)
IE (1) IE41003B1 (xx)
IL (1) IL47114A (xx)
LU (1) LU72315A1 (xx)
NL (1) NL159971C (xx)
NO (1) NO143155C (xx)
OA (1) OA04983A (xx)
PH (1) PH12067A (xx)
SE (1) SE427181B (xx)
SU (1) SU721002A3 (xx)
YU (1) YU93275A (xx)
ZA (1) ZA752471B (xx)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH01179624A (ja) * 1988-01-12 1989-07-17 Matsushita Refrig Co Ltd 生鮮物貯蔵装置
GB2442535B (en) 2006-10-05 2011-07-13 Ngf Europ Ltd Method and articles

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE34235B1 (en) * 1969-06-04 1975-03-19 Acf Chemiefarma Nv 6,7-benzomorphans and their preparation

Also Published As

Publication number Publication date
JPS6127390B2 (xx) 1986-06-25
HU173039B (hu) 1979-02-28
FR2267774B1 (xx) 1978-08-04
IL47114A (en) 1979-01-31
FR2267774A1 (xx) 1975-11-14
DK155999B (da) 1989-06-12
FI60564C (fi) 1982-02-10
ZA752471B (en) 1976-03-31
JPS50142568A (xx) 1975-11-17
NO143155B (no) 1980-09-15
PH12067A (en) 1978-10-30
IE41003L (en) 1975-10-18
SE427181B (sv) 1983-03-14
OA04983A (fr) 1980-11-30
DE2517220A1 (de) 1975-11-06
CS199586B2 (en) 1980-07-31
JPS6218552B2 (xx) 1987-04-23
JPS60120868A (ja) 1985-06-28
JPH0119387B2 (xx) 1989-04-11
SE7504469L (sv) 1975-10-20
IE41003B1 (en) 1979-09-26
CA1040630A (en) 1978-10-17
NL7504648A (nl) 1975-10-21
NO143155C (no) 1980-12-29
AU8025875A (en) 1976-10-21
IL47114A0 (en) 1975-06-25
DK166375A (da) 1975-10-19
FI60564B (fi) 1981-10-30
DD119787A5 (xx) 1976-05-12
NL159971C (nl) 1979-09-17
NO751371L (xx) 1975-10-21
SU721002A3 (ru) 1980-03-05
DK155999C (da) 1989-11-06
DE2517220C2 (xx) 1990-04-19
GB1493420A (en) 1977-11-30
DK194088D0 (da) 1988-04-08
FI751106A (xx) 1975-10-19
LU72315A1 (xx) 1976-03-17
BE828054A (fr) 1975-10-17
YU93275A (en) 1982-02-28
DK194088A (da) 1988-04-08
JPS60142964A (ja) 1985-07-29

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