CA2722582A1 - Inhibiteurs de pde4 biaryle pour traiter une inflammation - Google Patents

Inhibiteurs de pde4 biaryle pour traiter une inflammation Download PDF

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Publication number
CA2722582A1
CA2722582A1 CA2722582A CA2722582A CA2722582A1 CA 2722582 A1 CA2722582 A1 CA 2722582A1 CA 2722582 A CA2722582 A CA 2722582A CA 2722582 A CA2722582 A CA 2722582A CA 2722582 A1 CA2722582 A1 CA 2722582A1
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nhc
alkyl
mmol
chosen
compound
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Inventor
Jasbir Singh
Mark E. Gurney
Alex Burgin
Vincent Sandanayaka
Alexander Kiselyov
Adalie Motta
Gary Schultz
Georgeta Hategan
Timothy Hagen
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Decode Genetics ehf
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Decode Genetics ehf
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Publication of CA2722582A1 publication Critical patent/CA2722582A1/fr
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    • C07C275/32—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms
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    • C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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AU2008326381B2 (en) 2014-10-23
EP2222638A2 (fr) 2010-09-01

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