BRPI9911326B8 - análogos macrocíclicos e métodos para seu uso e preparação - Google Patents

análogos macrocíclicos e métodos para seu uso e preparação

Info

Publication number
BRPI9911326B8
BRPI9911326B8 BRPI9911326A BR9911326A BRPI9911326B8 BR PI9911326 B8 BRPI9911326 B8 BR PI9911326B8 BR PI9911326 A BRPI9911326 A BR PI9911326A BR 9911326 A BR9911326 A BR 9911326A BR PI9911326 B8 BRPI9911326 B8 BR PI9911326B8
Authority
BR
Brazil
Prior art keywords
methods
preparation
analogues
macrocyclic
cell
Prior art date
Application number
BRPI9911326A
Other languages
English (en)
Portuguese (pt)
Other versions
BR9911326B1 (pt
BR9911326A (pt
Inventor
M Seletsky Boris
A Littlefield Bruce
j yu Melvin
Palme Monica
J Towle Murray
Zheng Wanjun
Original Assignee
Eisai Co Ltd
Eisai R&D Man Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22219026&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI9911326(B8) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Eisai Co Ltd, Eisai R&D Man Co Ltd filed Critical Eisai Co Ltd
Publication of BR9911326A publication Critical patent/BR9911326A/pt
Publication of BR9911326B1 publication Critical patent/BR9911326B1/pt
Publication of BRPI9911326B8 publication Critical patent/BRPI9911326B8/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicinal Preparation (AREA)
  • Steroid Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Peptides Or Proteins (AREA)
BRPI9911326A 1998-06-17 1999-06-16 análogos macrocíclicos e métodos para seu uso e preparação BRPI9911326B8 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US8968298P 1998-06-17 1998-06-17
US60/089,682 1998-06-17
PCT/US1999/013677 WO1999065894A1 (en) 1998-06-17 1999-06-16 Macrocyclic analogs and methods of their use and preparation

Publications (3)

Publication Number Publication Date
BR9911326A BR9911326A (pt) 2001-04-03
BR9911326B1 BR9911326B1 (pt) 2015-01-06
BRPI9911326B8 true BRPI9911326B8 (pt) 2021-05-25

Family

ID=22219026

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI9911326A BRPI9911326B8 (pt) 1998-06-17 1999-06-16 análogos macrocíclicos e métodos para seu uso e preparação

Country Status (22)

Country Link
US (4) US6214865B1 (enExample)
EP (4) EP1087960B1 (enExample)
JP (1) JP4454151B2 (enExample)
KR (1) KR100798600B1 (enExample)
CN (1) CN1216051C (enExample)
AT (1) ATE502932T1 (enExample)
AU (1) AU762998B2 (enExample)
BE (1) BE2011C028I2 (enExample)
BR (1) BRPI9911326B8 (enExample)
CA (3) CA2335300C (enExample)
CY (2) CY1111516T1 (enExample)
DE (2) DE122011100031I1 (enExample)
DK (1) DK1087960T3 (enExample)
FR (1) FR11C0038I2 (enExample)
HU (1) HU227912B1 (enExample)
IL (1) IL139960A0 (enExample)
LU (1) LU91854I2 (enExample)
NO (5) NO328280B1 (enExample)
NZ (1) NZ508597A (enExample)
PT (1) PT1087960E (enExample)
WO (1) WO1999065894A1 (enExample)
ZA (1) ZA200007159B (enExample)

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Also Published As

Publication number Publication date
HK1035534A1 (en) 2001-11-30
NO328280B1 (no) 2010-01-25
CY1111516T1 (el) 2014-04-09
AU762998B2 (en) 2003-07-10
EP2277873A1 (en) 2011-01-26
CA2632433C (en) 2012-02-07
IL139960A0 (en) 2002-02-10
NO20093217L (no) 2001-02-15
NO20006316L (no) 2001-02-15
RU2245335C2 (ru) 2005-01-27
HUP0103357A2 (hu) 2002-01-28
NO20006316D0 (no) 2000-12-12
CN1216051C (zh) 2005-08-24
CA2755266C (en) 2014-08-12
EP1087960A1 (en) 2001-04-04
NO2022019I1 (no) 2022-06-03
EP2272840B1 (en) 2012-08-22
HUP0103357A3 (en) 2002-10-28
US6469182B1 (en) 2002-10-22
FR11C0038I2 (fr) 2013-01-11
DE122011100031I1 (de) 2011-12-15
BR9911326B1 (pt) 2015-01-06
FR11C0038I1 (fr) 2011-10-14
JP4454151B2 (ja) 2010-04-21
NO2011026I1 (no) 2012-01-09
DK1087960T3 (da) 2011-06-14
CY2011010I1 (el) 2014-04-09
AU762998C (en) 2000-01-05
CA2632433A1 (en) 1999-12-23
NZ508597A (en) 2004-01-30
US8148554B2 (en) 2012-04-03
EP1087960B1 (en) 2011-03-23
WO1999065894A1 (en) 1999-12-23
CA2755266A1 (en) 1999-12-23
AU4573999A (en) 2000-01-05
ATE502932T1 (de) 2011-04-15
EP1087960A4 (en) 2004-12-01
US6365759B1 (en) 2002-04-02
DE69943296D1 (de) 2011-05-05
KR20010083050A (ko) 2001-08-31
CA2335300C (en) 2008-10-07
US20110172446A1 (en) 2011-07-14
PT1087960E (pt) 2011-06-17
EP2272839B1 (en) 2012-08-22
EP2277873B1 (en) 2012-05-30
US6214865B1 (en) 2001-04-10
EP2272839A1 (en) 2011-01-12
NO2011026I2 (no) 2012-06-11
HU227912B1 (en) 2012-05-29
NO331183B1 (no) 2011-10-24
BE2011C028I2 (en) 2018-08-24
EP2272840A1 (en) 2011-01-12
JP2002518384A (ja) 2002-06-25
CN1312804A (zh) 2001-09-12
KR100798600B1 (ko) 2008-01-28
CA2335300A1 (en) 1999-12-23
ZA200007159B (en) 2001-12-04
LU91854I2 (fr) 2011-10-17
CY2011010I2 (el) 2014-04-09
BR9911326A (pt) 2001-04-03
NO2011018I1 (no) 2011-09-26

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