BR0107246A - Agentes diazabicìclicos ativos no sistema nervoso central - Google Patents

Agentes diazabicìclicos ativos no sistema nervoso central

Info

Publication number
BR0107246A
BR0107246A BR0107246-3A BR0107246A BR0107246A BR 0107246 A BR0107246 A BR 0107246A BR 0107246 A BR0107246 A BR 0107246A BR 0107246 A BR0107246 A BR 0107246A
Authority
BR
Brazil
Prior art keywords
diazabicyclic
nervous system
central nervous
agents active
compounds
Prior art date
Application number
BR0107246-3A
Other languages
English (en)
Portuguese (pt)
Inventor
Michael R Schrimpf
Karin R Tietje
Richard B Toupence
Jianguo Ji
Anwer Basha
William H Bunnelle
Jerome F Daanen
Jennifer M Pace
Kevin B Sippy
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US09/833,914 external-priority patent/US6809105B2/en
Application filed by Abbott Lab filed Critical Abbott Lab
Publication of BR0107246A publication Critical patent/BR0107246A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/34—Tobacco-abuse
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Addiction (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Anesthesiology (AREA)
  • Urology & Nephrology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BR0107246-3A 2000-04-27 2001-04-27 Agentes diazabicìclicos ativos no sistema nervoso central BR0107246A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US55994300A 2000-04-27 2000-04-27
US09/833,914 US6809105B2 (en) 2000-04-27 2001-04-12 Diazabicyclic central nervous system active agents
PCT/US2001/013798 WO2001081347A2 (en) 2000-04-27 2001-04-27 Diazabicyclic central nervous system active agents

Publications (1)

Publication Number Publication Date
BR0107246A true BR0107246A (pt) 2002-10-01

Family

ID=27072208

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0107246-3A BR0107246A (pt) 2000-04-27 2001-04-27 Agentes diazabicìclicos ativos no sistema nervoso central

Country Status (22)

Country Link
EP (3) EP2295437A1 (enExample)
JP (2) JP4981232B2 (enExample)
KR (4) KR100947188B1 (enExample)
CN (3) CN102863441A (enExample)
AR (1) AR030421A1 (enExample)
AU (2) AU2001266559C1 (enExample)
BG (2) BG66151B1 (enExample)
BR (1) BR0107246A (enExample)
CA (2) CA2407094C (enExample)
CZ (4) CZ302038B6 (enExample)
HK (1) HK1054375A1 (enExample)
HU (1) HUP0300602A3 (enExample)
IL (3) IL152231A0 (enExample)
MX (1) MXPA02010594A (enExample)
MY (3) MY137020A (enExample)
NO (1) NO324250B1 (enExample)
NZ (1) NZ521734A (enExample)
PE (1) PE20011305A1 (enExample)
PL (2) PL398491A1 (enExample)
SK (2) SK287658B6 (enExample)
TW (4) TWI311137B (enExample)
WO (1) WO2001081347A2 (enExample)

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CN107108597B (zh) 2014-10-31 2020-04-17 英立维尔英国有限公司 多巴胺d3受体拮抗剂化合物
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Also Published As

Publication number Publication date
CN101935322A (zh) 2011-01-05
TW200909432A (en) 2009-03-01
TWI357903B (en) 2012-02-11
KR20090013833A (ko) 2009-02-05
KR20090071654A (ko) 2009-07-01
CZ301324B6 (cs) 2010-01-13
CZ302795B6 (cs) 2011-11-16
TW200617013A (en) 2006-06-01
CN1440410A (zh) 2003-09-03
WO2001081347A3 (en) 2002-01-31
JP4981232B2 (ja) 2012-07-18
BG66151B1 (bg) 2011-08-31
EP2298775A1 (en) 2011-03-23
CZ20023765A3 (cs) 2003-02-12
AU2001266559B2 (en) 2005-03-03
SK16812002A3 (sk) 2003-04-01
HUP0300602A2 (hu) 2003-06-28
PL358340A1 (en) 2004-08-09
EP2295437A1 (en) 2011-03-16
MXPA02010594A (es) 2003-05-14
IL177316A0 (en) 2006-12-10
CN100430398C (zh) 2008-11-05
CA2407094A1 (en) 2001-11-01
SK287658B6 (sk) 2011-05-06
PE20011305A1 (es) 2001-12-31
TW201141871A (en) 2011-12-01
CA2407094C (en) 2009-11-17
MY168244A (en) 2018-10-15
CN102863441A (zh) 2013-01-09
KR100961406B1 (ko) 2010-06-09
IL152231A0 (en) 2003-05-29
CZ302072B6 (cs) 2010-09-29
NO20025107L (no) 2002-12-19
AU6655901A (en) 2001-11-07
SK287273B6 (sk) 2010-05-07
KR100947188B1 (ko) 2010-03-12
BG110620A (bg) 2010-07-30
BG107303A (bg) 2003-07-31
NZ521734A (en) 2004-10-29
HK1054375A1 (zh) 2003-11-28
IL203035A (en) 2010-12-30
PL398491A1 (pl) 2012-06-04
AU2001266559C1 (en) 2005-11-17
MY137020A (en) 2008-12-31
KR100899950B1 (ko) 2009-05-28
JP2003531210A (ja) 2003-10-21
NO324250B1 (no) 2007-09-17
NO20025107D0 (no) 2002-10-24
HUP0300602A3 (en) 2005-12-28
KR100947187B1 (ko) 2010-03-12
CA2683045A1 (en) 2001-11-01
JP2012041349A (ja) 2012-03-01
WO2001081347A2 (en) 2001-11-01
IL177316A (en) 2010-06-30
CZ302038B6 (cs) 2010-09-15
KR20090121385A (ko) 2009-11-25
AR030421A1 (es) 2003-08-20
KR20020093955A (ko) 2002-12-16
TWI311137B (en) 2009-06-21
EP1284976A2 (en) 2003-02-26
MY145722A (en) 2012-03-30
TWI323733B (en) 2010-04-21

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