BG63121B1 - Таксоиди, тяхното получаване и фармацевтични състави, които ги съдържат - Google Patents
Таксоиди, тяхното получаване и фармацевтични състави, които ги съдържат Download PDFInfo
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- BG63121B1 BG63121B1 BG101918A BG10191897A BG63121B1 BG 63121 B1 BG63121 B1 BG 63121B1 BG 101918 A BG101918 A BG 101918A BG 10191897 A BG10191897 A BG 10191897A BG 63121 B1 BG63121 B1 BG 63121B1
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Epoxy Compounds (AREA)
- Medicines Containing Plant Substances (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9503545A FR2732340B1 (fr) | 1995-03-27 | 1995-03-27 | Nouveaux taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent |
| FR9515381A FR2742754B1 (fr) | 1995-12-22 | 1995-12-22 | Procede de preparation de taxoides |
| PCT/FR1996/000441 WO1996030356A1 (fr) | 1995-03-27 | 1996-03-25 | Nouveaux taxoïdes, leur preparation et les compositions pharmaceutiques qui les contiennent |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BG101918A BG101918A (en) | 1998-10-30 |
| BG63121B1 true BG63121B1 (bg) | 2001-04-30 |
Family
ID=26231838
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG101918A BG63121B1 (bg) | 1995-03-27 | 1997-09-25 | Таксоиди, тяхното получаване и фармацевтични състави, които ги съдържат |
| BG101917A BG63009B1 (bg) | 1995-03-27 | 1997-09-25 | Таксоиди,тяхното получаване и фармацевтични състави, които ги съдържат |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG101917A BG63009B1 (bg) | 1995-03-27 | 1997-09-25 | Таксоиди,тяхното получаване и фармацевтични състави, които ги съдържат |
Country Status (41)
| Country | Link |
|---|---|
| US (3) | US5889043A (cs) |
| EP (2) | EP0817780B1 (cs) |
| JP (2) | JP2941951B2 (cs) |
| KR (2) | KR100297196B1 (cs) |
| CN (2) | CN1213042C (cs) |
| AP (2) | AP753A (cs) |
| AR (1) | AR001440A1 (cs) |
| AT (2) | ATE188471T1 (cs) |
| AU (2) | AU711227B2 (cs) |
| BG (2) | BG63121B1 (cs) |
| BR (2) | BR9607929A (cs) |
| CA (2) | CA2214319C (cs) |
| CO (1) | CO4700576A1 (cs) |
| CZ (2) | CZ287468B6 (cs) |
| DE (2) | DE69604653T2 (cs) |
| DK (2) | DK0817780T3 (cs) |
| DZ (1) | DZ2009A1 (cs) |
| EA (2) | EA000709B1 (cs) |
| EE (2) | EE03609B1 (cs) |
| ES (2) | ES2140075T3 (cs) |
| GE (2) | GEP20002188B (cs) |
| GR (2) | GR3031526T3 (cs) |
| HU (2) | HU223732B1 (cs) |
| IL (1) | IL117636A (cs) |
| IS (2) | IS2058B (cs) |
| MA (1) | MA23823A1 (cs) |
| MY (1) | MY121225A (cs) |
| NO (2) | NO316607B1 (cs) |
| NZ (2) | NZ304901A (cs) |
| OA (2) | OA10514A (cs) |
| PE (1) | PE51097A1 (cs) |
| PL (2) | PL188284B1 (cs) |
| PT (1) | PT817779E (cs) |
| RO (2) | RO115878B1 (cs) |
| SK (2) | SK281928B6 (cs) |
| TN (1) | TNSN96043A1 (cs) |
| TR (2) | TR199701040T1 (cs) |
| TW (1) | TW394765B (cs) |
| UY (2) | UY24192A1 (cs) |
| WO (2) | WO1996030356A1 (cs) |
| ZA (1) | ZA962399B (cs) |
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| US6500858B2 (en) | 1994-10-28 | 2002-12-31 | The Research Foundation Of The State University Of New York | Taxoid anti-tumor agents and pharmaceutical compositions thereof |
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| US5811452A (en) * | 1997-01-08 | 1998-09-22 | The Research Foundation Of State University Of New York | Taxoid reversal agents for drug-resistance in cancer chemotherapy and pharmaceutical compositions thereof |
| US7288665B1 (en) * | 1997-08-18 | 2007-10-30 | Florida State University | Process for selective derivatization of taxanes |
| FR2771092B1 (fr) * | 1997-11-18 | 1999-12-17 | Rhone Poulenc Rorer Sa | Procede de preparation de derives de la classe des taxoides |
| US6346543B1 (en) * | 1998-08-17 | 2002-02-12 | Aventis Pharma S.A. | Use of a taxoid to treat abnormal cell proliferation in the brain |
| EP0982027A1 (en) * | 1998-08-17 | 2000-03-01 | Aventis Pharma S.A. | Taxoid derivatives for treating abnormal cell proliferation of the brain |
| KR20010079665A (ko) * | 1998-08-20 | 2001-08-22 | 추후제출 | 탁소이드 유도체의 신규 용도 |
| EP0982028A1 (en) * | 1998-08-20 | 2000-03-01 | Aventis Pharma S.A. | New use of taxoid derivatives |
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| US8147816B2 (en) * | 2000-08-16 | 2012-04-03 | Encore Health, Llc | Presbyopia treatment by lens alteration |
| HUP0302599A3 (en) | 2000-09-22 | 2005-05-30 | Bristol Myers Squibb Co | Method for reducing toxicity of combined chemotherapic compositions |
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| US6593334B1 (en) | 2002-05-02 | 2003-07-15 | The University Of North Carolina At Chapel Hill | Camptothecin-taxoid conjugates as antimitotic and antitumor agents |
| KR102008768B1 (ko) | 2002-09-06 | 2019-08-08 | 인설트 테라페틱스, 인코퍼레이티드 | 공유결합된 치료제 전달을 위한 사이클로덱스트린-기초 중합체 |
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| SG10201810928SA (en) | 2009-10-29 | 2019-01-30 | Aventis Pharma Sa | Novel antitumoral use of cabazitaxel |
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| US10894087B2 (en) | 2010-12-22 | 2021-01-19 | Nektar Therapeutics | Multi-arm polymeric prodrug conjugates of cabazitaxel-based compounds |
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| EA023950B1 (ru) | 2011-04-12 | 2016-07-29 | Тева Фармасьютикалз Интернэшнл Гмбх | Твердофазные формы кабазитаксела и способы их получения |
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| JP6025861B2 (ja) | 2011-12-13 | 2016-11-16 | アベンティス・ファーマ・ソシエテ・アノニム | カバジタキセルの結晶形およびこれを調製するための方法 |
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| EP2743264A1 (en) | 2012-12-13 | 2014-06-18 | INDENA S.p.A. | New crystalline form of cabazitaxel, process for the preparation and pharmaceutical compositions thereof |
| EP2815749A1 (en) | 2013-06-20 | 2014-12-24 | IP Gesellschaft für Management mbH | Solid form of 4-amino-2-(2,6-dioxopiperidine-3-yl)isoindoline-1,3-dione having specified X-ray diffraction pattern |
| EP2865674A1 (en) | 2013-10-23 | 2015-04-29 | INDENA S.p.A. | Crystalline solvate forms of Cabazitaxel |
| EP2865675A1 (en) * | 2013-10-23 | 2015-04-29 | INDENA S.p.A. | A crystalline anhydrous form of Cabazitaxel, process for the preparation and pharmaceutical compositions thereof |
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| PL3258931T3 (pl) | 2015-02-17 | 2020-12-28 | Erasmus University Medical Center Rotterdam | Zastosowanie kabazitakselu w leczeniu nowotworu złośliwego prostaty |
| EP3093014A1 (en) * | 2015-05-13 | 2016-11-16 | Aventis Pharma S.A. | Cabazitaxel and its use for treating cancer |
| WO2020249507A1 (en) | 2019-06-11 | 2020-12-17 | Indena S.P.A. | Anhydrous crystalline form of cabazitaxel, a process for its preparation and pharmaceutical compositions containing it |
| TWI857119B (zh) | 2019-08-08 | 2024-10-01 | 香港商來凱有限公司 | 治療癌症之方法 |
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| FR2629819B1 (fr) | 1988-04-06 | 1990-11-16 | Rhone Poulenc Sante | Procede de preparation de derives de la baccatine iii et de la desacetyl-10 baccatine iii |
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| US5489601A (en) | 1991-09-23 | 1996-02-06 | Florida State University | Taxanes having a pyridyl substituted side-chain and pharmaceutical compositions containing them |
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| EP0767786B1 (en) | 1994-06-28 | 1998-09-16 | PHARMACIA & UPJOHN COMPANY | 7-ether-taxol analogs, antineoplastic use and pharmaceutical compositions containing them |
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1996
- 1996-03-08 MA MA24180A patent/MA23823A1/fr unknown
- 1996-03-19 PE PE1996000181A patent/PE51097A1/es not_active IP Right Cessation
- 1996-03-24 IL IL11763696A patent/IL117636A/en active Protection Beyond IP Right Term
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- 1996-03-25 HU HU9801204A patent/HU223732B1/hu active IP Right Grant
- 1996-03-25 CA CA002214321A patent/CA2214321C/fr not_active Expired - Fee Related
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- 1996-03-25 EE EE9700315A patent/EE03608B1/xx unknown
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- 1996-03-25 TR TR97/01042T patent/TR199701042T1/xx unknown
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- 1996-03-25 WO PCT/FR1996/000441 patent/WO1996030356A1/fr not_active Ceased
- 1996-03-25 ES ES96909192T patent/ES2143187T3/es not_active Expired - Lifetime
- 1996-03-25 GE GEAP19963956A patent/GEP20002188B/en unknown
- 1996-03-25 WO PCT/FR1996/000440 patent/WO1996030355A1/fr not_active Ceased
- 1996-03-25 CN CNB961928840A patent/CN1152870C/zh not_active Expired - Fee Related
- 1996-03-25 CZ CZ19973030A patent/CZ287326B6/cs not_active IP Right Cessation
- 1996-03-25 EP EP96909192A patent/EP0817779B1/fr not_active Expired - Lifetime
- 1996-03-25 GE GEAP19963957A patent/GEP20002211B/en unknown
- 1996-03-25 KR KR1019970706762A patent/KR100485309B1/ko not_active Expired - Fee Related
- 1996-03-25 BR BR9607930A patent/BR9607930A/pt not_active IP Right Cessation
- 1996-03-26 TN TNTNSN96043A patent/TNSN96043A1/fr unknown
- 1996-03-26 ZA ZA962399A patent/ZA962399B/xx unknown
- 1996-03-26 TW TW085103611A patent/TW394765B/zh not_active IP Right Cessation
- 1996-03-26 MY MYPI96001132A patent/MY121225A/en unknown
- 1996-03-26 DZ DZ960050A patent/DZ2009A1/fr active
- 1996-03-27 AR AR33592996A patent/AR001440A1/es active IP Right Grant
- 1996-03-27 UY UY24192A patent/UY24192A1/es not_active IP Right Cessation
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- 1996-11-20 UY UY24370A patent/UY24370A1/es not_active IP Right Cessation
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1997
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- 1997-08-26 NO NO973923A patent/NO316607B1/no not_active IP Right Cessation
- 1997-08-26 NO NO19973922A patent/NO316379B1/no not_active IP Right Cessation
- 1997-09-23 IS IS4567A patent/IS2056B/is unknown
- 1997-09-25 BG BG101918A patent/BG63121B1/bg unknown
- 1997-09-25 BG BG101917A patent/BG63009B1/bg unknown
- 1997-09-26 OA OA70087A patent/OA10514A/fr unknown
- 1997-09-26 OA OA70086A patent/OA10513A/fr unknown
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1998
- 1998-04-28 US US09/066,929 patent/US6331635B1/en not_active Expired - Lifetime
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1999
- 1999-10-14 GR GR990402228T patent/GR3031526T3/el unknown
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2000
- 2000-01-07 GR GR990402501T patent/GR3032316T3/el unknown
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2001
- 2001-09-25 US US09/985,956 patent/US6387946B1/en not_active Expired - Lifetime
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2007
- 2007-09-11 PL PL96322499A patent/PL188987B1/pl unknown
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