BE892357A - Nouveaux derives de l'erythromycine a, procede pour leur preparation et leur utilisation comme substances anti-bacteriennes - Google Patents

Nouveaux derives de l'erythromycine a, procede pour leur preparation et leur utilisation comme substances anti-bacteriennes

Info

Publication number
BE892357A
BE892357A BE0/207464A BE207464A BE892357A BE 892357 A BE892357 A BE 892357A BE 0/207464 A BE0/207464 A BE 0/207464A BE 207464 A BE207464 A BE 207464A BE 892357 A BE892357 A BE 892357A
Authority
BE
Belgium
Prior art keywords
derivatives
preparation
bacterial substances
novel erythromycin
erythromycin
Prior art date
Application number
BE0/207464A
Other languages
English (en)
Original Assignee
Pliva Pharm & Chem Works
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25550598&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BE892357(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pliva Pharm & Chem Works filed Critical Pliva Pharm & Chem Works
Publication of BE892357A publication Critical patent/BE892357A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
BE0/207464A 1981-03-06 1982-03-04 Nouveaux derives de l'erythromycine a, procede pour leur preparation et leur utilisation comme substances anti-bacteriennes BE892357A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
YU592/81A YU43006B (en) 1981-03-06 1981-03-06 Process for preparing n-methyl-11-aza-10-deoxo-10-dihydro erythromycin and derivatives thereof

Publications (1)

Publication Number Publication Date
BE892357A true BE892357A (fr) 1982-07-01

Family

ID=25550598

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/207464A BE892357A (fr) 1981-03-06 1982-03-04 Nouveaux derives de l'erythromycine a, procede pour leur preparation et leur utilisation comme substances anti-bacteriennes

Country Status (19)

Country Link
US (1) US4517359A (fr)
JP (1) JPS5858357B2 (fr)
AT (1) AT375945B (fr)
BE (1) BE892357A (fr)
CA (1) CA1191843A (fr)
CH (1) CH655728A5 (fr)
CZ (1) CZ418991A3 (fr)
DD (1) DD202437A5 (fr)
DE (1) DE3140449C2 (fr)
FR (1) FR2501212B1 (fr)
GB (1) GB2094293B (fr)
HU (1) HU186845B (fr)
IT (1) IT1200960B (fr)
PL (2) PL133764B1 (fr)
SE (1) SE457084B (fr)
SI (1) SI8110592A8 (fr)
SK (1) SK418991A3 (fr)
SU (1) SU1287755A3 (fr)
YU (1) YU43006B (fr)

Cited By (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4464527A (en) * 1983-06-30 1984-08-07 Pfizer Inc. Antibacterial 9-deoxo-9a-alkyl-9a-aza-9a-homoerythromycin A derivatives and intermediates therefore
US4474768A (en) * 1982-07-19 1984-10-02 Pfizer Inc. N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor
WO1999020639A3 (fr) * 1997-10-16 1999-07-08 Pliva Pharm & Chem Works NOUVEAUX 3,6-HEMICETALS APPARTENANT A LA CLASSE DES 9a-AZALIDES
BG64600B1 (bg) * 1998-04-06 2005-08-31 Pliva, Farmaceutska Industrija, Dionicko Drustvo Кетолиди от класа на 15-членни лактами с антибактериална активност
US7419961B2 (en) 2002-10-29 2008-09-02 Zambon S.P.A. 9a-azalides with anti-inflammatory activity
US9700564B2 (en) 2009-09-04 2017-07-11 Horizon Orphan Llc Use of aerosolized levofloxacin for treating cystic fibrosis
US9717738B2 (en) 2008-10-07 2017-08-01 Horizon Orphan Llc Aerosol fluoroquinolone formulations for improved pharmacokinetics
US10987357B2 (en) 2005-05-18 2021-04-27 Horizon Orphan, LLC Aerosolized fluoroquinolones and uses thereof
WO2021209563A1 (fr) 2020-04-16 2021-10-21 Som Innovation Biotech, S.A. Composés destinés à être utilisés dans le traitement d'infections virales par un coronavirus associé au syndrome respiratoire

Families Citing this family (140)

* Cited by examiner, † Cited by third party
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US4526889A (en) * 1982-11-15 1985-07-02 Pfizer Inc. Epimeric azahomoerythromycin A derivative, intermediates and method of use
US4492688A (en) * 1983-11-25 1985-01-08 Pfizer Inc. Antibacterial cyclic ethers of 9-deoxo-9a-aza-9a-homoerythromycin A and intermediates therefor
JPS59225198A (ja) * 1983-05-23 1984-12-18 フアイザ−・インコ−ポレ−テツド 抗菌性を有する９―デオキソ―９ａ―アザ―９ａ―ホモエリスロマイシンＡ，その製造方法および組成物
DE3461803D1 (en) * 1983-05-23 1987-02-05 Pfizer Antibacterial cyclic ethers of 9-deoxo-9a-aza-9a-homoerythromycin a and intermediates therefor
GR80277B (en) * 1983-09-06 1985-01-04 Pfizer Azahomoerythromycin b derivatives and intermediates therefor
US4465674A (en) * 1983-09-06 1984-08-14 Pfizer Inc. Azahomoerythromycin D derivative and intermediates therefor
US4518590A (en) * 1984-04-13 1985-05-21 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
US4512982A (en) * 1984-04-13 1985-04-23 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical composition and therapeutic method
US4921947A (en) * 1986-03-31 1990-05-01 Eli Lilly And Company Process for preparing macrolide derivatives
RU2066324C1 (ru) 1987-07-09 1996-09-10 Пфайзер Инк. Кристаллический дигидрат азитромицина и способ его получения
WO1989002271A1 (fr) * 1987-09-10 1989-03-23 Pfizer Azithromycine et derives utilises comme agents anti-protozoaires
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US6017894A (en) * 1988-08-03 2000-01-25 Schering Corporation Actinomadura fulva subsp uruguayensis and antimicrobial complex and antimicrobial compounds isolated therefrom
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US5985844A (en) * 1992-03-26 1999-11-16 Merck & Co., Inc. Homoerythromycin A derivatives modified at the 4"-and 8A-positions
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US5215980A (en) * 1992-01-17 1993-06-01 Merck & Co., Inc. 10-AZA-9-deoxo-11-deoxy-erythromycin A and derivatives thereof
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CA2245398C (fr) * 1998-08-21 2002-01-29 Apotex Inc. Clathrate d'isopropanol monohydrate d'azithromycine et methodes d'obtention
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AR085286A1 (es) 2011-02-21 2013-09-18 Taisho Pharmaceutical Co Ltd Derivado de macrolido sustituido en la posicion c-4
JP5718488B2 (ja) 2011-03-01 2015-05-13 ウォックハート リミテッド ケトライド中間体の調製方法
EP2688900B1 (fr) 2011-03-22 2016-09-28 Wockhardt Limited Procédé de préparation de composés de cétolides
WO2013088274A1 (fr) 2011-12-14 2013-06-20 Wockhardt Limited Composition d'azithromycine amorphe anhydre dépourvue de dihydrate d'azithromycine
MX2015008146A (es) 2012-12-24 2016-01-20 Univ Ramot Agentes para tratar enfermedades geneticas derivadas de mutaciones sin sentido y metodos para identificarlas.
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AR102810A1 (es) 2014-08-18 2017-03-29 Taisho Pharmaceutical Co Ltd Derivado de macrólido sustituido en la posición c-4
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US4474768A (en) * 1982-07-19 1984-10-02 Pfizer Inc. N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor
US4464527A (en) * 1983-06-30 1984-08-07 Pfizer Inc. Antibacterial 9-deoxo-9a-alkyl-9a-aza-9a-homoerythromycin A derivatives and intermediates therefore
WO1999020639A3 (fr) * 1997-10-16 1999-07-08 Pliva Pharm & Chem Works NOUVEAUX 3,6-HEMICETALS APPARTENANT A LA CLASSE DES 9a-AZALIDES
BG64600B1 (bg) * 1998-04-06 2005-08-31 Pliva, Farmaceutska Industrija, Dionicko Drustvo Кетолиди от класа на 15-членни лактами с антибактериална активност
US7419961B2 (en) 2002-10-29 2008-09-02 Zambon S.P.A. 9a-azalides with anti-inflammatory activity
US10987357B2 (en) 2005-05-18 2021-04-27 Horizon Orphan, LLC Aerosolized fluoroquinolones and uses thereof
US9717738B2 (en) 2008-10-07 2017-08-01 Horizon Orphan Llc Aerosol fluoroquinolone formulations for improved pharmacokinetics
US10149854B2 (en) 2008-10-07 2018-12-11 Horizon Orphan Llc Aerosol fluoroquinolone formulations for improved pharmacokinetics
US10722519B2 (en) 2008-10-07 2020-07-28 Horizon Orphan Llc Aerosol fluoroquinolone formulations for improved pharmacokinetics
US9700564B2 (en) 2009-09-04 2017-07-11 Horizon Orphan Llc Use of aerosolized levofloxacin for treating cystic fibrosis
US10231975B2 (en) 2009-09-04 2019-03-19 Horizon Orphan Llc Use of aerosolized levofloxacin for treating cystic fibrosis
WO2021209563A1 (fr) 2020-04-16 2021-10-21 Som Innovation Biotech, S.A. Composés destinés à être utilisés dans le traitement d'infections virales par un coronavirus associé au syndrome respiratoire

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CA1191843A (fr) 1985-08-13
CZ418991A3 (en) 1993-01-13
PL235329A1 (fr) 1982-09-27
YU43006B (en) 1989-02-28
FR2501212A1 (fr) 1982-09-10
AT375945B (de) 1984-09-25
JPS57158798A (en) 1982-09-30
PL131784B1 (en) 1985-01-31
ATA440081A (de) 1984-02-15
SE457084B (sv) 1988-11-28
FR2501212B1 (fr) 1985-08-09
SU1287755A3 (ru) 1987-01-30
PL133764B1 (en) 1985-06-29
SK418991A3 (en) 1995-07-11
YU59281A (en) 1983-06-30
GB2094293A (en) 1982-09-15
IT1200960B (it) 1989-01-27
HU186845B (en) 1985-09-30
GB2094293B (en) 1985-12-18
US4517359A (en) 1985-05-14
DE3140449A1 (de) 1983-10-13
DD202437A5 (de) 1983-09-14
IT8267263A0 (it) 1982-03-05
JPS5858357B2 (ja) 1983-12-24
SI8110592A8 (en) 1996-06-30
SE8201311L (sv) 1982-09-07
CH655728A5 (de) 1986-05-15
DE3140449C2 (de) 1984-06-20

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