BE1000158A4 - Nouveaux anthracycline glycosides, leur procede de preparation et leur application comme agents antitumoraux. - Google Patents

Nouveaux anthracycline glycosides, leur procede de preparation et leur application comme agents antitumoraux. Download PDF

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Publication number
BE1000158A4
BE1000158A4 BE8700645A BE8700645A BE1000158A4 BE 1000158 A4 BE1000158 A4 BE 1000158A4 BE 8700645 A BE8700645 A BE 8700645A BE 8700645 A BE8700645 A BE 8700645A BE 1000158 A4 BE1000158 A4 BE 1000158A4
Authority
BE
Belgium
Prior art keywords
glycoside
formula
group
epi
salicylidene
Prior art date
Application number
BE8700645A
Other languages
English (en)
French (fr)
Inventor
Suarato Antonino
Caruso Michele
Penco Sergio
Giuliani Fernando
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Application granted granted Critical
Publication of BE1000158A4 publication Critical patent/BE1000158A4/fr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/24—Condensed ring systems having three or more rings
    • C07H15/252—Naphthacene radicals, e.g. daunomycins, adriamycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
BE8700645A 1986-06-12 1987-06-10 Nouveaux anthracycline glycosides, leur procede de preparation et leur application comme agents antitumoraux. BE1000158A4 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB868614323A GB8614323D0 (en) 1986-06-12 1986-06-12 Anthracyclines

Publications (1)

Publication Number Publication Date
BE1000158A4 true BE1000158A4 (fr) 1988-06-28

Family

ID=10599357

Family Applications (1)

Application Number Title Priority Date Filing Date
BE8700645A BE1000158A4 (fr) 1986-06-12 1987-06-10 Nouveaux anthracycline glycosides, leur procede de preparation et leur application comme agents antitumoraux.

Country Status (24)

Country Link
JP (1) JP2516769B2 (fi)
KR (1) KR950004897B1 (fi)
AT (1) AT392793B (fi)
AU (1) AU595328B2 (fi)
BE (1) BE1000158A4 (fi)
CA (1) CA1291122C (fi)
CH (1) CH676985A5 (fi)
DE (1) DE3719377C2 (fi)
DK (1) DK169076B1 (fi)
ES (1) ES2006488A6 (fi)
FI (1) FI84075C (fi)
FR (1) FR2600066B1 (fi)
GB (2) GB8614323D0 (fi)
GR (1) GR870909B (fi)
HU (1) HU196220B (fi)
IE (1) IE60412B1 (fi)
IL (1) IL82820A0 (fi)
IT (1) IT1215552B (fi)
NL (1) NL8701349A (fi)
NZ (1) NZ220604A (fi)
PT (1) PT85056B (fi)
SE (1) SE500732C2 (fi)
SU (1) SU1590045A3 (fi)
ZA (1) ZA874202B (fi)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3842836A1 (de) * 1988-12-20 1990-06-21 Behringwerke Ag Rhodomycine mit einer modifizierten kohlenhydrat-einheit
GB9325417D0 (en) * 1993-12-13 1994-02-16 Erba Carlo Spa 3'- aziridino-anthracycline derivatives
IT1275953B1 (it) * 1995-03-22 1997-10-24 Sicor Spa Procedimento per la preparazione di antibiotici della classe delle antracicline
GB9808027D0 (en) * 1998-04-15 1998-06-17 Pharmacia & Upjohn Spa 13-dihydro-3' aziridino anthracyclines
AU2343900A (en) * 1998-11-02 2000-05-22 Board Of Regents, The University Of Texas System Methods and compositions for the manufacture of highly potent anthracycline-based antitumor agents
GB0114654D0 (en) * 2001-06-15 2001-08-08 Pharmacia & Upjohn Spa Anti-tumor compound
CN110483871A (zh) * 2019-08-15 2019-11-22 陈全明 一种抗压耐磨的hdpe双壁波纹管

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0051280A1 (en) * 1980-11-01 1982-05-12 FARMITALIA CARLO ERBA S.p.A. Anthracycline glycosides, process for the preparation thereof, intermediate compounds and their preparation and pharmaceutical compositions
EP0199920A1 (en) * 1985-03-28 1986-11-05 FARMITALIA CARLO ERBA S.r.l. New antitumor anthracyclines

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3803124A (en) * 1968-04-12 1974-04-09 Farmaceutici It Soc Process for the preparation of adriamycin and adriamycinone and adriamycin derivatives

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0051280A1 (en) * 1980-11-01 1982-05-12 FARMITALIA CARLO ERBA S.p.A. Anthracycline glycosides, process for the preparation thereof, intermediate compounds and their preparation and pharmaceutical compositions
EP0199920A1 (en) * 1985-03-28 1986-11-05 FARMITALIA CARLO ERBA S.r.l. New antitumor anthracyclines

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
ANTHRACYCLINE ANTIBIOTICS, 1982, pages 197-224, Academic Press, Inc.; D. HORTON et al.: "Glycon- and C-14-modified, antitumor doxorubicin analogs" *

Also Published As

Publication number Publication date
PT85056B (pt) 1990-03-30
GB2195998A (en) 1988-04-20
DK169076B1 (da) 1994-08-08
FI84075C (fi) 1991-10-10
DE3719377A1 (de) 1987-12-17
FI872571A (fi) 1987-12-13
DK298787D0 (da) 1987-06-11
JP2516769B2 (ja) 1996-07-24
GB8713443D0 (en) 1987-07-15
NL8701349A (nl) 1988-01-04
AU7410887A (en) 1987-12-17
IT1215552B (it) 1990-02-14
IT8720834A0 (it) 1987-06-09
AT392793B (de) 1991-06-10
SU1590045A3 (ru) 1990-08-30
SE8702409D0 (sv) 1987-06-10
HUT43866A (en) 1987-12-28
FR2600066B1 (fr) 1992-05-15
NZ220604A (en) 1989-10-27
ATA144987A (de) 1990-11-15
HU196220B (en) 1988-10-28
GR870909B (en) 1987-10-12
ZA874202B (en) 1988-02-24
SE500732C2 (sv) 1994-08-15
AU595328B2 (en) 1990-03-29
IL82820A0 (en) 1987-12-20
FI84075B (fi) 1991-06-28
PT85056A (en) 1987-07-01
IE60412B1 (en) 1994-07-13
IE871538L (en) 1987-12-13
FR2600066A1 (fr) 1987-12-18
SE8702409L (sv) 1987-12-13
GB2195998B (en) 1990-02-14
DK298787A (da) 1987-12-13
DE3719377C2 (de) 1995-09-28
FI872571A0 (fi) 1987-06-09
KR950004897B1 (ko) 1995-05-15
CH676985A5 (fi) 1991-03-28
GB8614323D0 (en) 1986-07-16
ES2006488A6 (es) 1989-05-01
KR880000459A (ko) 1988-03-26
CA1291122C (en) 1991-10-22
JPS62292793A (ja) 1987-12-19

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: FARMITALIA CARLO ERBA S.P.A.

Effective date: 19960630