AU3921478A - 3,4,5 trihydroxypiperidine derivatives - Google Patents

3,4,5 trihydroxypiperidine derivatives

Info

Publication number
AU3921478A
AU3921478A AU39214/78A AU3921478A AU3921478A AU 3921478 A AU3921478 A AU 3921478A AU 39214/78 A AU39214/78 A AU 39214/78A AU 3921478 A AU3921478 A AU 3921478A AU 3921478 A AU3921478 A AU 3921478A
Authority
AU
Australia
Prior art keywords
trihydroxypiperidine
derivatives
trihydroxypiperidine derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
AU39214/78A
Other languages
English (en)
Inventor
Bodo Junge
Hans Peter Krause
Lutz Muller
Walter Puls
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25772626&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU3921478(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from DE19772738717 external-priority patent/DE2738717A1/de
Priority claimed from DE19772758025 external-priority patent/DE2758025A1/de
Application filed by Bayer AG filed Critical Bayer AG
Publication of AU3921478A publication Critical patent/AU3921478A/en
Pending legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H9/00Compounds containing a hetero ring sharing at least two hetero atoms with a saccharide radical
    • C07H9/02Compounds containing a hetero ring sharing at least two hetero atoms with a saccharide radical the hetero ring containing only oxygen as ring hetero atoms
    • C07H9/04Cyclic acetals
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • A23K20/116Heterocyclic compounds
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • A23K20/116Heterocyclic compounds
    • A23K20/132Heterocyclic compounds containing only one nitrogen as hetero atom
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • A23K20/116Heterocyclic compounds
    • A23K20/137Heterocyclic compounds containing two hetero atoms, of which at least one is nitrogen
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K50/00Feeding-stuffs specially adapted for particular animals
    • A23K50/30Feeding-stuffs specially adapted for particular animals for swines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40Oxygen atoms
    • C07D211/44Oxygen atoms attached in position 4
    • C07D211/46Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/60Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02Acyclic radicals, not substituted by cyclic structures
    • C07H15/12Acyclic radicals, not substituted by cyclic structures attached to a nitrogen atom of the saccharide radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02Acyclic radicals, not substituted by cyclic structures
    • C07H15/14Acyclic radicals, not substituted by cyclic structures attached to a sulfur, selenium or tellurium atom of a saccharide radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/18Acyclic radicals, substituted by carbocyclic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Polymers & Plastics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Food Science & Technology (AREA)
  • Zoology (AREA)
  • Animal Husbandry (AREA)
  • Diabetes (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Birds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU39214/78A 1977-08-27 1978-08-24 3,4,5 trihydroxypiperidine derivatives Pending AU3921478A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19772738717 DE2738717A1 (de) 1977-08-27 1977-08-27 N-alkylierte derivate der 5-amino- 5-deoxy-d-glucose, verfahren zu ihrer herstellung und ihre verwendung
DE19772758025 DE2758025A1 (de) 1977-12-24 1977-12-24 Neue derivate von 3,4,5-trihydroxypiperidin, verfahren zu ihrer herstellung und ihre verwendung

Publications (1)

Publication Number Publication Date
AU3921478A true AU3921478A (en) 1980-02-28

Family

ID=25772626

Family Applications (2)

Application Number Title Priority Date Filing Date
AU39214/78A Pending AU3921478A (en) 1977-08-27 1978-08-24 3,4,5 trihydroxypiperidine derivatives
AU39304/78A Expired AU520686B2 (en) 1977-08-27 1978-08-28 3, 4, 5-trihydroxypiperidines amd their use in animal nutrition and against diabetes

Family Applications After (1)

Application Number Title Priority Date Filing Date
AU39304/78A Expired AU520686B2 (en) 1977-08-27 1978-08-28 3, 4, 5-trihydroxypiperidines amd their use in animal nutrition and against diabetes

Country Status (19)

Country Link
US (2) US4639436A (enExample)
EP (1) EP0000947B2 (enExample)
JP (1) JPS5446786A (enExample)
AT (1) AT373239B (enExample)
AU (2) AU3921478A (enExample)
CA (1) CA1123437A (enExample)
DE (1) DE2860330D1 (enExample)
DK (1) DK152753C (enExample)
ES (1) ES472838A1 (enExample)
FI (1) FI72715C (enExample)
GR (1) GR73065B (enExample)
HU (1) HU182449B (enExample)
IE (1) IE47070B1 (enExample)
IL (1) IL55423A (enExample)
IT (1) IT1111197B (enExample)
LU (1) LU90211I2 (enExample)
NL (1) NL960027I2 (enExample)
NO (1) NO154918C (enExample)
PT (1) PT68474A (enExample)

Families Citing this family (245)

* Cited by examiner, † Cited by third party
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JPS5943946B2 (ja) * 1978-04-28 1984-10-25 日本新薬株式会社 N−アルケニルモラノリン誘導体
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DE2922760A1 (de) * 1979-06-05 1980-12-11 Bayer Ag Neue derivate von 3,4,5-trihydroxypiperidin, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel sowie in der tierernaehrung
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DE2660486C2 (de) * 1975-12-29 1984-03-08 Nippon Shinyaku Co., Ltd., Kyoto Verwendung von 2-Hydroxymethyl-3,4,5-trihydroxypiperidin als Arzneimittel
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GB2020278B (en) * 1978-05-03 1983-02-23 Nippon Shinyaku Co Ltd Moranoline dervitives
JPS5943948B2 (ja) * 1978-07-06 1984-10-25 日本新薬株式会社 置換モラノリン誘導体
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JPS5943948A (ja) * 1982-09-03 1984-03-12 Toyota Motor Corp 可変ベンチユリ型気化器

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NO154918B (no) 1986-10-06
FI72715C (fi) 1987-07-10
NO154918C (no) 1987-01-14
IL55423A (en) 1982-09-30
FI782607A7 (fi) 1979-02-28
NO782713L (no) 1979-02-28
AT373239B (de) 1983-12-27
AU3930478A (en) 1980-03-06
AU520686B2 (en) 1982-02-18
EP0000947B2 (de) 1984-10-10
EP0000947A1 (de) 1979-03-07
IL55423A0 (en) 1978-10-31
FI72715B (fi) 1987-03-31
LU90211I2 (fr) 1998-04-08
US4639436A (en) 1987-01-27
JPS5446786A (en) 1979-04-12
IE47070B1 (en) 1983-12-14
ES472838A1 (es) 1979-03-16
NL960027I2 (nl) 1997-07-01
IT1111197B (it) 1986-01-13
US4260622A (en) 1981-04-07
JPS6231703B2 (enExample) 1987-07-09
NL960027I1 (nl) 1997-01-06
DK152753C (da) 1988-10-31
DE2860330D1 (en) 1981-03-12
GR73065B (enExample) 1984-01-30
HU182449B (en) 1984-01-30
IT7827067A0 (it) 1978-08-25
IE781716L (en) 1979-02-27
DK152753B (da) 1988-05-09
DK377678A (da) 1979-02-28
CA1123437A (en) 1982-05-11
ATA621778A (de) 1983-05-15
EP0000947B1 (de) 1981-01-14
PT68474A (de) 1978-09-01

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