ATE403659T1 - Camptothecine mit modifiziertem lactonring - Google Patents

Camptothecine mit modifiziertem lactonring

Info

Publication number
ATE403659T1
ATE403659T1 AT06116366T AT06116366T ATE403659T1 AT E403659 T1 ATE403659 T1 AT E403659T1 AT 06116366 T AT06116366 T AT 06116366T AT 06116366 T AT06116366 T AT 06116366T AT E403659 T1 ATE403659 T1 AT E403659T1
Authority
AT
Austria
Prior art keywords
camptothecine
lactone ring
modified lactone
modified
ring
Prior art date
Application number
AT06116366T
Other languages
German (de)
English (en)
Inventor
Mauro Marzi
Elena Marastoni
Sergio Penco
Claudio Pisano
Maria Ornella Tinti
Loredana Vesci
Franco Zunino
Domenico Vergani
Walter Cabri
Marco Alpegiani
Martin Patricio
Tamara Danelli
Original Assignee
Sigma Tau Ind Farmaceuti
Ist Naz Stud Cura Dei Tumori
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sigma Tau Ind Farmaceuti, Ist Naz Stud Cura Dei Tumori filed Critical Sigma Tau Ind Farmaceuti
Application granted granted Critical
Publication of ATE403659T1 publication Critical patent/ATE403659T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/22Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Epoxy Compounds (AREA)
AT06116366T 2002-05-31 2003-05-28 Camptothecine mit modifiziertem lactonring ATE403659T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT2002RM000305A ITRM20020305A1 (it) 2002-05-31 2002-05-31 Camptotecine con anello lattonico modificato.

Publications (1)

Publication Number Publication Date
ATE403659T1 true ATE403659T1 (de) 2008-08-15

Family

ID=11456338

Family Applications (2)

Application Number Title Priority Date Filing Date
AT06116366T ATE403659T1 (de) 2002-05-31 2003-05-28 Camptothecine mit modifiziertem lactonring
AT03730480T ATE339422T1 (de) 2002-05-31 2003-05-28 Camptothecine mit modifiziertem lactonring

Family Applications After (1)

Application Number Title Priority Date Filing Date
AT03730480T ATE339422T1 (de) 2002-05-31 2003-05-28 Camptothecine mit modifiziertem lactonring

Country Status (22)

Country Link
US (1) US7273873B2 (enExample)
EP (2) EP1719775B1 (enExample)
JP (1) JP4693410B2 (enExample)
KR (1) KR101042042B1 (enExample)
CN (1) CN1656100A (enExample)
AR (1) AR040139A1 (enExample)
AT (2) ATE403659T1 (enExample)
AU (2) AU2003241160B2 (enExample)
BR (2) BR0311333A (enExample)
CA (2) CA2485201C (enExample)
CY (2) CY1107311T1 (enExample)
DE (2) DE60322754D1 (enExample)
DK (2) DK1719775T3 (enExample)
ES (2) ES2273002T7 (enExample)
IT (1) ITRM20020305A1 (enExample)
MX (1) MXPA04011682A (enExample)
PE (1) PE20050120A1 (enExample)
PL (1) PL374346A1 (enExample)
PT (2) PT1511752E (enExample)
SI (2) SI1511752T1 (enExample)
TW (1) TWI325866B (enExample)
WO (1) WO2003101995A2 (enExample)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2852606A1 (fr) * 2003-03-18 2004-09-24 Inst Nat Sante Rech Med Moyens pour inhiber simultanement l'expression de plusieurs genes impliques dans une pathologie
ITRM20030344A1 (it) * 2003-07-14 2005-01-15 Ist Naz Stud Cura Dei Tumori 7-n-poliamminoalchil(ossi)imminometilcamptotecine recanti gruppi protettivi.
PL2170900T3 (pl) * 2007-08-01 2013-04-30 Sigma Tau Ind Farmaceuti Krystaliczna forma II 7-(dimetoksymetylo)kamptotecyny, jej zastosowanie jako związek pośredni oraz otrzymane z niej produkty
CN102746314B (zh) * 2011-04-18 2016-07-06 华东师范大学 含有稳定7元内酯环的喜树碱类化合物、制备方法和用途
CN104530066A (zh) * 2015-01-06 2015-04-22 华东师范大学 一类新型高喜树碱衍生物、制备方法和用途
CN112566666A (zh) 2018-05-14 2021-03-26 努瓦申生物公司 靶向抗癌核激素受体的化合物
AU2020274113A1 (en) 2019-05-14 2021-11-11 Nuvation Bio Inc. Anti-cancer nuclear hormone receptor-targeting compounds
TW202131930A (zh) 2019-11-13 2021-09-01 美商諾維雪碧歐公司 抗癌核荷爾蒙受體標靶化合物
IL306010A (en) 2021-03-23 2023-11-01 Nuvation Bio Inc Anticancer compounds against the nuclear hormone receptor
CA3218577A1 (en) 2021-05-03 2022-11-10 Nuvation Bio Inc. Anti-cancer nuclear hormone receptor-targeting compounds
WO2024073626A2 (en) * 2022-09-28 2024-04-04 Nuvation Bio Inc. Anti-cancer nuclear hormone receptor-targeting compounds

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57116076A (en) * 1981-01-09 1982-07-19 Yakult Honsha Co Ltd Novel camptothecin derivative and its preparation
US4399276A (en) * 1981-01-09 1983-08-16 Kabushiki Kaisha Yakult Honsha 7-Substituted camptothecin derivatives
FR2532591A1 (fr) 1982-09-02 1984-03-09 Hutchinson Nouveau dispositif de securite pour pneumatiques de vehicules ou autres engins
EP1251125B1 (fr) * 1995-06-21 2005-12-07 Société de Conseils et de Recherches d'Applications Scientifiques (S.C.R.A.S.) Nouveaux analogues de la camptoth-cine, des proc-d-s de pr-paration, leur application comme m-dicaments et les compositions pharmaceutiques les contenant
DK1044977T3 (da) * 1999-03-09 2002-07-08 Sigma Tau Ind Farmaceuti Camptothecinderivater med antitumoraktivitet

Also Published As

Publication number Publication date
ES2273002T7 (es) 2011-08-01
EP1719775B1 (en) 2008-08-06
WO2003101995A2 (en) 2003-12-11
PT1719775E (pt) 2008-09-30
SI1511752T1 (sl) 2007-02-28
EP1719775A1 (en) 2006-11-08
BR0311329A (pt) 2005-02-22
AU2009236044A1 (en) 2009-12-03
EP1511752A2 (en) 2005-03-09
ITRM20020305A1 (it) 2003-12-01
AU2003241160A1 (en) 2003-12-19
JP2005531602A (ja) 2005-10-20
CY1108793T1 (el) 2014-04-09
AU2009236044B2 (en) 2011-03-24
AU2009236044A8 (en) 2011-07-21
DE60308368T3 (de) 2010-09-16
EP1511752B3 (en) 2010-03-10
EP1511752B8 (en) 2007-04-18
ES2312090T3 (es) 2009-02-16
DE60308368D1 (de) 2006-10-26
EP1511752B1 (en) 2006-09-13
ATE339422T1 (de) 2006-10-15
AU2009236044B8 (en) 2011-07-21
PL374346A1 (en) 2005-10-17
WO2003101995A8 (en) 2004-12-23
SI1719775T1 (sl) 2009-04-30
CA2485201A1 (en) 2003-12-11
JP4693410B2 (ja) 2011-06-01
US20050154003A1 (en) 2005-07-14
DK1511752T5 (da) 2010-06-14
DE60322754D1 (de) 2008-09-18
BR0311333A (pt) 2005-03-15
PT1511752E (pt) 2007-01-31
TWI325866B (en) 2010-06-11
CY1107311T1 (el) 2012-11-21
ITRM20020305A0 (it) 2002-05-31
TW200404806A (en) 2004-04-01
CA2706635A1 (en) 2003-12-11
PE20050120A1 (es) 2005-03-04
CN1656100A (zh) 2005-08-17
KR20050036909A (ko) 2005-04-20
DE60308368T2 (de) 2007-09-06
DK1719775T3 (da) 2008-11-17
CA2485201C (en) 2010-11-02
AU2003241160B2 (en) 2009-08-20
ES2273002T3 (es) 2007-05-01
KR101042042B1 (ko) 2011-06-16
AR040139A1 (es) 2005-03-16
MXPA04011682A (es) 2005-03-31
WO2003101995A3 (en) 2004-02-19
US7273873B2 (en) 2007-09-25
DK1511752T3 (da) 2007-01-29

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