AR067024A1 - Metabolitos del inhibidor de janus quinasa (r)-3-(4-(7h-pirrolo(2,3-d)pirimidin-4-il)-1h-pirazol-1-il)-3-ciclopentilpropanonitrilo - Google Patents

Metabolitos del inhibidor de janus quinasa (r)-3-(4-(7h-pirrolo(2,3-d)pirimidin-4-il)-1h-pirazol-1-il)-3-ciclopentilpropanonitrilo

Info

Publication number
AR067024A1
AR067024A1 ARP080102565A ARP080102565A AR067024A1 AR 067024 A1 AR067024 A1 AR 067024A1 AR P080102565 A ARP080102565 A AR P080102565A AR P080102565 A ARP080102565 A AR P080102565A AR 067024 A1 AR067024 A1 AR 067024A1
Authority
AR
Argentina
Prior art keywords
pyrrolo
pyrazol
pyrimidin
janus
metabolites
Prior art date
Application number
ARP080102565A
Other languages
English (en)
Spanish (es)
Inventor
James D Rodgers
Argyrios G Arvanitis
Sung-Hyuk Shin
Original Assignee
Incyte Corp
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Publication date
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Publication of AR067024A1 publication Critical patent/AR067024A1/es

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Transplantation (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Genetics & Genomics (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Biomedical Technology (AREA)
  • Microbiology (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • General Engineering & Computer Science (AREA)
ARP080102565A 2007-06-13 2008-06-17 Metabolitos del inhibidor de janus quinasa (r)-3-(4-(7h-pirrolo(2,3-d)pirimidin-4-il)-1h-pirazol-1-il)-3-ciclopentilpropanonitrilo AR067024A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US94369507P 2007-06-13 2007-06-13

Publications (1)

Publication Number Publication Date
AR067024A1 true AR067024A1 (es) 2009-09-30

Family

ID=40029276

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP080102565A AR067024A1 (es) 2007-06-13 2008-06-17 Metabolitos del inhibidor de janus quinasa (r)-3-(4-(7h-pirrolo(2,3-d)pirimidin-4-il)-1h-pirazol-1-il)-3-ciclopentilpropanonitrilo

Country Status (25)

Country Link
US (5) US7834022B2 (OSRAM)
EP (1) EP2173751B1 (OSRAM)
JP (1) JP5479331B2 (OSRAM)
KR (1) KR20100049008A (OSRAM)
CN (1) CN101815717B (OSRAM)
AR (1) AR067024A1 (OSRAM)
AU (1) AU2008266182B8 (OSRAM)
BR (1) BRPI0812563A2 (OSRAM)
CA (1) CA2689158C (OSRAM)
CL (1) CL2008001709A1 (OSRAM)
CO (1) CO6251255A2 (OSRAM)
CR (1) CR11149A (OSRAM)
EA (1) EA017790B1 (OSRAM)
EC (1) ECSP099821A (OSRAM)
ES (1) ES2448868T3 (OSRAM)
GE (1) GEP20125534B (OSRAM)
IL (1) IL202429A0 (OSRAM)
MX (2) MX339139B (OSRAM)
NZ (1) NZ581801A (OSRAM)
PL (1) PL2173751T3 (OSRAM)
PT (1) PT2173751E (OSRAM)
TW (1) TWI426911B (OSRAM)
UA (1) UA99465C2 (OSRAM)
WO (1) WO2008157207A2 (OSRAM)
ZA (1) ZA200908820B (OSRAM)

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