AR049583A2 - Compuesto derivado de pirazolo-pirimidina, composicion farmaceutica y el uso de dicho compuesto en la fabricacion de medicamentos - Google Patents

Compuesto derivado de pirazolo-pirimidina, composicion farmaceutica y el uso de dicho compuesto en la fabricacion de medicamentos

Info

Publication number
AR049583A2
AR049583A2 ARP050102868A ARP050102868A AR049583A2 AR 049583 A2 AR049583 A2 AR 049583A2 AR P050102868 A ARP050102868 A AR P050102868A AR P050102868 A ARP050102868 A AR P050102868A AR 049583 A2 AR049583 A2 AR 049583A2
Authority
AR
Argentina
Prior art keywords
alkyl
cycloalkyl
haloalkyl
optionally substituted
case
Prior art date
Application number
ARP050102868A
Other languages
English (en)
Spanish (es)
Inventor
Liqi He
Paul Joseph Gilligan
Argyrios Georgios Arvanitis
Original Assignee
Bristol Myers Squibb Pharma Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/899,242 external-priority patent/US6124289A/en
Application filed by Bristol Myers Squibb Pharma Co filed Critical Bristol Myers Squibb Pharma Co
Publication of AR049583A2 publication Critical patent/AR049583A2/es

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Detergent Compositions (AREA)
  • Coloring (AREA)
ARP050102868A 1996-07-24 2005-07-11 Compuesto derivado de pirazolo-pirimidina, composicion farmaceutica y el uso de dicho compuesto en la fabricacion de medicamentos AR049583A2 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US68604796A 1996-07-24 1996-07-24
US2329096P 1996-07-24 1996-07-24
US08/899,242 US6124289A (en) 1996-07-24 1997-07-23 Azolo triazines and pyrimidines

Publications (1)

Publication Number Publication Date
AR049583A2 true AR049583A2 (es) 2006-08-16

Family

ID=27362048

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP050102868A AR049583A2 (es) 1996-07-24 2005-07-11 Compuesto derivado de pirazolo-pirimidina, composicion farmaceutica y el uso de dicho compuesto en la fabricacion de medicamentos

Country Status (15)

Country Link
JP (2) JP4704521B2 (pt)
CN (3) CN1104432C (pt)
AR (1) AR049583A2 (pt)
BR (1) BR9710544A (pt)
CA (1) CA2259583C (pt)
CZ (1) CZ299451B6 (pt)
EA (1) EA004403B1 (pt)
EE (1) EE04316B1 (pt)
HR (1) HRP970413A2 (pt)
IL (4) IL127871A0 (pt)
NO (1) NO315610B1 (pt)
NZ (1) NZ333777A (pt)
PL (1) PL195762B1 (pt)
SI (1) SI9720045B (pt)
SK (1) SK286461B6 (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4549630B2 (ja) * 2001-03-13 2010-09-22 ブリストル−マイヤーズ スクイブ ファーマ カンパニー コルチコトロピン放出因子受容体リガンドとしての、4−(2−ブチルアミノ)−2,7−ジメチル−8−(2−メチル−6−メトキシピリド−3−イル)ピラゾロ−[1,5−a]−1,3,5−トリアジン、その鏡像異性体および薬学的に許容できる塩類
WO2004110454A1 (ja) * 2003-06-13 2004-12-23 Ishihara Sangyo Kaisha, Ltd. アデノシンA2a受容体アゴニストの投与が必要な疾患を治療又は予防するための組成物
US7329662B2 (en) * 2003-10-03 2008-02-12 Hoffmann-La Roche Inc. Pyrazolo-pyridine
GB0519957D0 (en) * 2005-09-30 2005-11-09 Sb Pharmco Inc Chemical compound
CA2663511C (en) * 2006-09-20 2012-12-04 Eli Lilly And Company Thiazole pyrazolopyrimidines as crf1 receptor antagonists
CN103694242B (zh) * 2013-12-10 2016-01-06 昆明翔昊科技有限公司 吡唑并嘧啶类化合物及其药物组合物和其在制药中的应用
CN112608316B (zh) * 2019-07-30 2022-10-21 厦门宝太生物科技股份有限公司 一种吡唑并三嗪类腺苷受体拮抗剂
AU2021324839B2 (en) 2020-08-12 2024-02-29 Spruce Biosciences, Inc. Methods and compositions for treating polycystic ovary syndrome
US11708372B2 (en) 2021-11-19 2023-07-25 Spruce Biosciences, Inc. Crystalline composition of tildacerfont and methods of use and preparation thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3995039A (en) * 1975-05-27 1976-11-30 Merck & Co., Inc. Pyrazolo [1,5-a] [1,3,5] triazines
JPS6157587A (ja) * 1984-08-29 1986-03-24 Shionogi & Co Ltd 縮合複素環誘導体および抗潰瘍剤
US4824834A (en) * 1986-10-31 1989-04-25 Otsuka Pharmaceutical Company, Limited Pyrazolotriazine compounds
JP2691317B2 (ja) * 1989-08-25 1997-12-17 株式会社大塚製薬工場 4―ヒドロキシ―8―(3―低級アルコキシ―4―フェニルスルフィニルフェニル)ピラゾロ〔1,5―a〕―1,3,5―トリアジン光学活性体の塩類及びその製造方法
AU639615B2 (en) * 1990-10-09 1993-07-29 Otsuka Pharmaceutical Co., Ltd. Pyrimidine derivative, production thereof, and androgen inhibitor
CA2107479C (en) * 1991-04-22 1997-12-16 Makoto Inoue Pyrazolo[1,5-a]pyrimidine derivatives and anti-inflammatory agent containing the same
US5356897A (en) * 1991-09-09 1994-10-18 Fujisawa Pharmaceutical Co., Ltd. 3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines

Also Published As

Publication number Publication date
JP2002513382A (ja) 2002-05-08
SI9720045A (sl) 1999-10-31
CN1250223C (zh) 2006-04-12
EE9900019A (et) 1999-08-16
JP4704521B2 (ja) 2011-06-15
JP4194539B2 (ja) 2008-12-10
SI9720045B (sl) 2008-02-29
PL195762B1 (pl) 2007-10-31
CZ299451B6 (cs) 2008-07-30
NZ333777A (en) 2000-07-28
CN1388126A (zh) 2003-01-01
NO315610B3 (no) 2003-09-29
EA004403B1 (ru) 2004-04-29
CN1225637A (zh) 1999-08-11
IL164513A (en) 2010-04-29
HRP970413A2 (en) 1998-10-31
PL331523A1 (en) 1999-07-19
IL164513A0 (en) 2005-12-18
CN1104432C (zh) 2003-04-02
SK286461B6 (sk) 2008-10-07
IL127871A0 (en) 1999-10-28
CA2259583C (en) 2009-11-17
NO990264L (no) 1999-03-10
NO315610B1 (no) 2003-09-29
EE04316B1 (et) 2004-06-15
EA199900158A1 (ru) 1999-10-28
CZ18499A3 (cs) 1999-11-17
BR9710544A (pt) 1999-08-17
NO990264D0 (no) 1999-01-21
CA2259583A1 (en) 1998-01-29
IL150163A (en) 2010-12-30
IL127871A (en) 2010-04-29
SK9799A3 (sk) 2005-04-01
CN1327793A (zh) 2001-12-26
JP2005097257A (ja) 2005-04-14

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