AR048939A1 - Derivados de fenol y tiofenol 3 - o 4 - monosustituidos utiles como ligandos de h3; composiciones farmaceuticas que los contienen y su uso en la fabricacion de medicamentos para el tratamiento de trastornos neurologicos e inflamatorios. - Google Patents

Derivados de fenol y tiofenol 3 - o 4 - monosustituidos utiles como ligandos de h3; composiciones farmaceuticas que los contienen y su uso en la fabricacion de medicamentos para el tratamiento de trastornos neurologicos e inflamatorios.

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Publication number
AR048939A1
AR048939A1 ARP050101824A ARP050101824A AR048939A1 AR 048939 A1 AR048939 A1 AR 048939A1 AR P050101824 A ARP050101824 A AR P050101824A AR P050101824 A ARP050101824 A AR P050101824A AR 048939 A1 AR048939 A1 AR 048939A1
Authority
AR
Argentina
Prior art keywords
alkyl
optionally substituted
alkoxy
amino
cycloalkyl
Prior art date
Application number
ARP050101824A
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English (en)
Spanish (es)
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP04291187A external-priority patent/EP1593679A1/en
Priority claimed from GB0504564A external-priority patent/GB0504564D0/en
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of AR048939A1 publication Critical patent/AR048939A1/es

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    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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ARP050101824A 2004-05-07 2005-05-05 Derivados de fenol y tiofenol 3 - o 4 - monosustituidos utiles como ligandos de h3; composiciones farmaceuticas que los contienen y su uso en la fabricacion de medicamentos para el tratamiento de trastornos neurologicos e inflamatorios. AR048939A1 (es)

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EP04291187A EP1593679A1 (en) 2004-05-07 2004-05-07 3- Or 4-monosubstituted phenol derivatives useful as H3 ligands
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WO2007045989A1 (en) * 2005-10-20 2007-04-26 Pfizer Limited Pyridyl derivatives useful as h3 ligands
JP5432526B2 (ja) 2006-01-06 2014-03-05 サノビオン ファーマシューティカルズ インク モノアミン再取り込み阻害剤としてのシクロアルキルアミン
CA2636275C (en) 2006-01-06 2013-02-12 Sepracor Inc. Tetralone-based monoamine reuptake inhibitors
US8097760B2 (en) 2006-03-31 2012-01-17 Sunovion Pharmacuticals Inc. Preparation of chiral amides and amines
EP2007723A2 (en) 2006-04-11 2008-12-31 Novartis AG Organic compounds
KR20090024811A (ko) 2006-06-23 2009-03-09 아보트 러보러터리즈 히스타민 ｈ3 수용체 조절제로서의 사이클로프로필 아민 유도체
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PA8632201A1 (es) 2006-09-22
AU2005240846A1 (en) 2005-11-17
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JP4173191B2 (ja) 2008-10-29
KR20060133091A (ko) 2006-12-22
CA2565852C (en) 2010-08-10
CN1950351A (zh) 2007-04-18
DE602005022062D1 (de) 2010-08-12
TW200607494A (en) 2006-03-01
BRPI0510664A (pt) 2007-12-04
DK1747210T3 (da) 2010-09-27
ES2346665T3 (es) 2010-10-19
ATE472540T1 (de) 2010-07-15
EP1747210B1 (en) 2010-06-30
TW200815412A (en) 2008-04-01
CR8729A (es) 2006-11-30
HK1100823A1 (en) 2007-09-28
CA2565852A1 (en) 2005-11-17
TWI346549B (en) 2011-08-11
PL1747210T3 (pl) 2010-11-30
MY144634A (en) 2011-10-14
PT1747210E (pt) 2010-08-31
CY1110735T1 (el) 2015-06-10
AP2006003772A0 (en) 2006-10-31
RS51403B (sr) 2011-02-28
NZ550769A (en) 2010-06-25
SI1747210T1 (sl) 2010-09-30
AP2353A (en) 2012-02-16
EA011161B1 (ru) 2009-02-27
JP2007536365A (ja) 2007-12-13
KR100843848B1 (ko) 2008-07-03
GT200500107A (es) 2006-01-10
JP2008050365A (ja) 2008-03-06
PE20060237A1 (es) 2006-04-01
HRP20100469T1 (hr) 2010-10-31
IL178433A0 (en) 2007-02-11
EP1747210A1 (en) 2007-01-31
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MA28634B1 (fr) 2007-06-01
BRPI0510664B8 (pt) 2021-05-25
CN1950351B (zh) 2012-01-18
WO2005108384A1 (en) 2005-11-17
GEP20094826B (en) 2009-11-10
BRPI0510664B1 (pt) 2020-04-07
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