TW200815412A - A pharmaceutical combination comprising 3-or 4-monosubstituted phenol and thiophenol derivatives - Google Patents

A pharmaceutical combination comprising 3-or 4-monosubstituted phenol and thiophenol derivatives Download PDF

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Publication number
TW200815412A
TW200815412A TW096139294A TW96139294A TW200815412A TW 200815412 A TW200815412 A TW 200815412A TW 096139294 A TW096139294 A TW 096139294A TW 96139294 A TW96139294 A TW 96139294A TW 200815412 A TW200815412 A TW 200815412A
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Taiwan
Prior art keywords
group
phenyl
etoac
mmol
alkyl
Prior art date
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TW096139294A
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English (en)
Chinese (zh)
Inventor
Patrick Bernardelli
Andrew Michael Cronin
Alexis Denis
Stephen Martin Denton
Henry Jacobelli
Mark Ian Kemp
Edwige Lorthiois
Fiona Rousseau
Delphine Serradeil-Civit
Fabrice Vergne
Original Assignee
Warner Lambert Co
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Priority claimed from EP04291187A external-priority patent/EP1593679A1/en
Priority claimed from GB0504564A external-priority patent/GB0504564D0/en
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of TW200815412A publication Critical patent/TW200815412A/zh

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    • C07D309/04—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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WO2007045989A1 (en) * 2005-10-20 2007-04-26 Pfizer Limited Pyridyl derivatives useful as h3 ligands
JP5432526B2 (ja) 2006-01-06 2014-03-05 サノビオン ファーマシューティカルズ インク モノアミン再取り込み阻害剤としてのシクロアルキルアミン
CA2636275C (en) 2006-01-06 2013-02-12 Sepracor Inc. Tetralone-based monoamine reuptake inhibitors
US8097760B2 (en) 2006-03-31 2012-01-17 Sunovion Pharmacuticals Inc. Preparation of chiral amides and amines
EP2007723A2 (en) 2006-04-11 2008-12-31 Novartis AG Organic compounds
KR20090024811A (ko) 2006-06-23 2009-03-09 아보트 러보러터리즈 히스타민 ｈ3 수용체 조절제로서의 사이클로프로필 아민 유도체
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CA2565852C (en) 2010-08-10
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CR8729A (es) 2006-11-30
HK1100823A1 (en) 2007-09-28
CA2565852A1 (en) 2005-11-17
TWI346549B (en) 2011-08-11
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MY144634A (en) 2011-10-14
PT1747210E (pt) 2010-08-31
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RS51403B (sr) 2011-02-28
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