AR020029A1 - Procedimiento para preparar 2-fenil-3-aminopiridina, derivados fenilo sustituidos de la misma. - Google Patents
Procedimiento para preparar 2-fenil-3-aminopiridina, derivados fenilo sustituidos de la misma.Info
- Publication number
- AR020029A1 AR020029A1 ARP000102332A ARP000102332A AR020029A1 AR 020029 A1 AR020029 A1 AR 020029A1 AR P000102332 A ARP000102332 A AR P000102332A AR P000102332 A ARP000102332 A AR P000102332A AR 020029 A1 AR020029 A1 AR 020029A1
- Authority
- AR
- Argentina
- Prior art keywords
- compound
- phenyl
- formula
- aminopiridine
- prepare
- Prior art date
Links
- CIUQDSCDWFSTQR-UHFFFAOYSA-N [C]1=CC=CC=C1 Chemical class [C]1=CC=CC=C1 CIUQDSCDWFSTQR-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 9
- KDLHZDBZIXYQEI-UHFFFAOYSA-N Palladium Chemical compound [Pd] KDLHZDBZIXYQEI-UHFFFAOYSA-N 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 239000002904 solvent Substances 0.000 abstract 2
- XTHJCITVHCRQRD-UHFFFAOYSA-N 2-phenylpyridin-3-amine Chemical compound NC1=CC=CN=C1C1=CC=CC=C1 XTHJCITVHCRQRD-UHFFFAOYSA-N 0.000 abstract 1
- 239000011260 aqueous acid Substances 0.000 abstract 1
- 239000003054 catalyst Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 229910052763 palladium Inorganic materials 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/73—Unsubstituted amino or imino radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pyridine Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US13455999P | 1999-05-17 | 1999-05-17 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR020029A1 true AR020029A1 (es) | 2002-03-27 |
Family
ID=22463902
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP000102332A AR020029A1 (es) | 1999-05-17 | 2000-05-15 | Procedimiento para preparar 2-fenil-3-aminopiridina, derivados fenilo sustituidos de la misma. |
Country Status (25)
| Country | Link |
|---|---|
| US (1) | US6316632B1 (show.php) |
| EP (1) | EP1054002B1 (show.php) |
| JP (1) | JP3837011B2 (show.php) |
| KR (1) | KR100386226B1 (show.php) |
| CN (1) | CN1216865C (show.php) |
| AR (1) | AR020029A1 (show.php) |
| AT (1) | ATE306474T1 (show.php) |
| AU (1) | AU775947B2 (show.php) |
| BR (1) | BR0001773A (show.php) |
| CA (1) | CA2308817C (show.php) |
| CZ (1) | CZ299474B6 (show.php) |
| DE (1) | DE60023063T2 (show.php) |
| DK (1) | DK1054002T3 (show.php) |
| ES (1) | ES2248017T3 (show.php) |
| HU (1) | HUP0001928A3 (show.php) |
| ID (1) | ID26061A (show.php) |
| IL (1) | IL136105A (show.php) |
| IN (1) | IN192341B (show.php) |
| MX (1) | MXPA00004790A (show.php) |
| PL (1) | PL198153B1 (show.php) |
| RS (1) | RS49964B (show.php) |
| RU (1) | RU2181120C2 (show.php) |
| TR (1) | TR200001403A2 (show.php) |
| TW (1) | TWI286133B (show.php) |
| ZA (1) | ZA200002375B (show.php) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2021094247A1 (en) | 2019-11-15 | 2021-05-20 | KaNDy Therapeutics Limited | New chemical process for making 6-chloro-4-(4-fluoro-2-methylphenyl)pyridin-3-amine a key intermediate of nt-814 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5232929A (en) * | 1990-11-28 | 1993-08-03 | Pfizer Inc. | 3-aminopiperidine derivatives and related nitrogen containing heterocycles and pharmaceutical compositions and use |
| US5364943A (en) * | 1991-11-27 | 1994-11-15 | Pfizer Inc. | Preparation of substituted piperidines |
| DK0532515T3 (da) * | 1990-05-31 | 1997-04-21 | Pfizer | Fremstilling af substituerede piperidiner |
| CZ289960B6 (cs) | 1991-03-26 | 2002-05-15 | Pfizer Inc. | Způsob přípravy substituovaných piperidinů |
| BR9206161A (pt) | 1991-06-20 | 1995-10-31 | Pfizer | Derivados fluoroalcoxibenzilamino de heterociclos contendo nitrogénio |
| US6180647B1 (en) | 1995-07-07 | 2001-01-30 | Pfizer Inc. | Substituted benzolactam compounds as substance P antagonists |
| TW340842B (en) | 1995-08-24 | 1998-09-21 | Pfizer | Substituted benzylaminopiperidine compounds |
| AU734860B2 (en) | 1996-12-02 | 2001-06-21 | Merck Sharp & Dohme Limited | Use of NK-1 receptor antagonists for treating cognitive disorders |
| TW426667B (en) | 1997-11-19 | 2001-03-21 | Pfizer | Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance P antagonists |
-
2000
- 2000-04-03 RS YUP-196/00A patent/RS49964B/sr unknown
- 2000-04-07 CN CN001064517A patent/CN1216865C/zh not_active Expired - Fee Related
- 2000-04-11 AU AU27662/00A patent/AU775947B2/en not_active Ceased
- 2000-05-09 ES ES00303889T patent/ES2248017T3/es not_active Expired - Lifetime
- 2000-05-09 AT AT00303889T patent/ATE306474T1/de not_active IP Right Cessation
- 2000-05-09 DK DK00303889T patent/DK1054002T3/da active
- 2000-05-09 EP EP00303889A patent/EP1054002B1/en not_active Expired - Lifetime
- 2000-05-09 JP JP2000136185A patent/JP3837011B2/ja not_active Expired - Fee Related
- 2000-05-09 DE DE60023063T patent/DE60023063T2/de not_active Expired - Fee Related
- 2000-05-11 US US09/569,010 patent/US6316632B1/en not_active Expired - Fee Related
- 2000-05-11 IN IN506DE2000 patent/IN192341B/en unknown
- 2000-05-11 TW TW089109033A patent/TWI286133B/zh not_active IP Right Cessation
- 2000-05-12 IL IL136105A patent/IL136105A/en not_active IP Right Cessation
- 2000-05-15 ID IDP20000406A patent/ID26061A/id unknown
- 2000-05-15 CA CA002308817A patent/CA2308817C/en not_active Expired - Fee Related
- 2000-05-15 ZA ZA200002375A patent/ZA200002375B/xx unknown
- 2000-05-15 AR ARP000102332A patent/AR020029A1/es active IP Right Grant
- 2000-05-16 BR BR0001773-6A patent/BR0001773A/pt not_active Application Discontinuation
- 2000-05-16 RU RU2000112354/04A patent/RU2181120C2/ru not_active IP Right Cessation
- 2000-05-16 MX MXPA00004790A patent/MXPA00004790A/es unknown
- 2000-05-16 KR KR10-2000-0025978A patent/KR100386226B1/ko not_active Expired - Fee Related
- 2000-05-16 HU HU0001928A patent/HUP0001928A3/hu unknown
- 2000-05-16 CZ CZ20001800A patent/CZ299474B6/cs not_active IP Right Cessation
- 2000-05-17 PL PL340157A patent/PL198153B1/pl unknown
- 2000-05-17 TR TR2000/01403A patent/TR200001403A2/xx unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant, registration |