AP762A - Substituted 6,5-hetero-bicyclic derivatives. - Google Patents
Substituted 6,5-hetero-bicyclic derivatives. Download PDFInfo
- Publication number
- AP762A AP762A APAP/P/1997/001077A AP9701077A AP762A AP 762 A AP762 A AP 762A AP 9701077 A AP9701077 A AP 9701077A AP 762 A AP762 A AP 762A
- Authority
- AP
- ARIPO
- Prior art keywords
- alkyl
- phenyl
- trimethyl
- methyl
- ethyl
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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- A61P11/06—Antiasthmatics
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US2503996P | 1996-08-28 | 1996-08-28 |
Publications (2)
Publication Number | Publication Date |
---|---|
AP9701077A0 AP9701077A0 (en) | 1997-10-31 |
AP762A true AP762A (en) | 1999-09-13 |
Family
ID=21823717
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
APAP/P/1997/001077A AP762A (en) | 1996-08-28 | 1997-08-21 | Substituted 6,5-hetero-bicyclic derivatives. |
Country Status (36)
Country | Link |
---|---|
EP (1) | EP0923582B1 (ja) |
JP (2) | JP3621706B2 (ja) |
KR (1) | KR20000035934A (ja) |
CN (1) | CN1227554A (ja) |
AP (1) | AP762A (ja) |
AR (1) | AR015103A1 (ja) |
AT (1) | ATE340176T1 (ja) |
AU (1) | AU735401B2 (ja) |
BG (1) | BG103189A (ja) |
BR (1) | BR9711970A (ja) |
CA (1) | CA2263566C (ja) |
CO (1) | CO4600634A1 (ja) |
CZ (1) | CZ68199A3 (ja) |
DE (1) | DE69736711T2 (ja) |
DZ (1) | DZ2300A1 (ja) |
EA (1) | EA002769B1 (ja) |
ES (1) | ES2273369T3 (ja) |
GT (1) | GT199700095A (ja) |
HR (1) | HRP970454B1 (ja) |
HU (1) | HUP9903965A3 (ja) |
ID (1) | ID18249A (ja) |
IL (1) | IL127566A0 (ja) |
IS (1) | IS4963A (ja) |
MA (1) | MA26438A1 (ja) |
NO (1) | NO313636B1 (ja) |
NZ (1) | NZ333302A (ja) |
OA (1) | OA10977A (ja) |
PA (1) | PA8436201A1 (ja) |
PE (1) | PE108898A1 (ja) |
PL (1) | PL332040A1 (ja) |
SK (1) | SK23399A3 (ja) |
TN (1) | TNSN97145A1 (ja) |
TR (1) | TR199900389T2 (ja) |
TW (1) | TW575573B (ja) |
WO (1) | WO1998008847A1 (ja) |
ZA (1) | ZA977687B (ja) |
Families Citing this family (147)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1996035689A1 (en) | 1995-05-12 | 1996-11-14 | Neurogen Corporation | Novel deazapurine derivatives; a new class of crf1 specific ligands |
US6060478A (en) * | 1996-07-24 | 2000-05-09 | Dupont Pharmaceuticals | Azolo triazines and pyrimidines |
US6191131B1 (en) | 1997-07-23 | 2001-02-20 | Dupont Pharmaceuticals Company | Azolo triazines and pyrimidines |
US6124289A (en) * | 1996-07-24 | 2000-09-26 | Dupont Pharmaceuticals Co. | Azolo triazines and pyrimidines |
US7094782B1 (en) | 1996-07-24 | 2006-08-22 | Bristol-Myers Squibb Company | Azolo triazines and pyrimidines |
US6313124B1 (en) | 1997-07-23 | 2001-11-06 | Dupont Pharmaceuticals Company | Tetrazine bicyclic compounds |
WO1998035967A2 (en) * | 1997-02-18 | 1998-08-20 | Neurocrine Biosciences, Inc. | Biazacyclic crf antagonists |
NZ335823A (en) * | 1997-04-22 | 2001-06-29 | Neurocrine Biosciences Inc | Thiophenopyridines, preparation as CRF receptor antagonists |
WO1999001454A1 (en) * | 1997-07-03 | 1999-01-14 | Du Pont Pharmaceuticals Company | Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders |
DE69916578T2 (de) * | 1998-01-28 | 2005-03-31 | Bristol-Myers Squibb Pharma Co. | Pyrazolotriazine als crf-antagonisten |
US6187777B1 (en) | 1998-02-06 | 2001-02-13 | Amgen Inc. | Compounds and methods which modulate feeding behavior and related diseases |
US6472402B1 (en) | 1998-04-02 | 2002-10-29 | Neurogen Corporation | Aminoalkyl substituted 5,6,7,8-Tetrahydro-9H-Pyridino [2,3-B]indole derivatives |
CA2326319A1 (en) | 1998-04-02 | 1999-10-14 | Neurogen Corporation | Aminoalkyl substituted 5,6,7,8-tetrahydro-9h pyrimidino[2,3-b]indole and 5,6,7,8-tetrahydro-9h-pyrimidino[4,5-b]indole derivatives: crf1 specific ligands |
CA2326884A1 (en) * | 1998-04-03 | 1999-10-14 | Dupont Pharmaceuticals Company | Thiazolo¬4,5-d|pyrimidines and pyridines as corticotropin releasing factor (crf) antagonists |
ATE239019T1 (de) * | 1998-06-09 | 2003-05-15 | Neurogen Corp | Pyrido(2,3-b)indolizinderivate und aza analoge: crf1 spezifische liganden |
US6509338B1 (en) | 1998-06-22 | 2003-01-21 | Bristol-Myers Squibb Company | Pyrazolo[1,5-A]triazine corticotropin releasing factor antagonists |
WO2000011003A1 (en) * | 1998-08-21 | 2000-03-02 | Du Pont Pharmaceuticals Company | ISOXAZOLO[4,5-d]PYRIMIDINES AS CRF ANTAGONISTS |
ATE240958T1 (de) * | 1998-11-12 | 2003-06-15 | Neurocrine Biosciences Inc | Crf rezeptor-antagonisten und darauf bezogene methoden |
JP2002529465A (ja) * | 1998-11-12 | 2002-09-10 | ニューロクライン バイオサイエンシーズ, インコーポレイテッド | Crfレセプターアンタゴニストおよびcrfレセプターアンタゴニストに関する方法 |
US6531475B1 (en) * | 1998-11-12 | 2003-03-11 | Neurocrine Biosciences, Inc. | CRF receptor antagonists and methods relating thereto |
WO2000044754A1 (fr) * | 1999-01-29 | 2000-08-03 | Sumitomo Chemical Company, Limited | Agents inhibiteurs d'accumulation de graisse |
EP1040831A3 (en) * | 1999-04-02 | 2003-05-02 | Pfizer Products Inc. | Use of corticotropin releasing factor (CRF) antagonists to prevent sudden death |
WO2000059908A2 (en) | 1999-04-06 | 2000-10-12 | Du Pont Pharmaceuticals Company | Pyrazolopyrimidines as crf antagonists |
AU4331500A (en) | 1999-04-06 | 2000-10-23 | Du Pont Pharmaceuticals Company | Pyrazolotriazines as crf antagonists |
US6982265B1 (en) | 1999-05-21 | 2006-01-03 | Bristol Myers Squibb Company | Pyrrolotriazine inhibitors of kinases |
EP1669071B1 (en) * | 1999-05-21 | 2009-07-22 | Bristol-Myers Squibb Company | Pyrrolotriazine inhibitors of kinases |
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- 2004-09-21 JP JP2004273978A patent/JP2005047930A/ja not_active Withdrawn
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1995033750A1 (en) * | 1994-06-08 | 1995-12-14 | Pfizer Inc. | Corticotropin releasing factor antagonists |
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