ZA792804B - New 2,6-dimethyl-4-2,3-disubstituted phenyl-1,4-dihydropyridine-3,5-dicarboxylic acid 3,5-asymmetric disters - Google Patents

New 2,6-dimethyl-4-2,3-disubstituted phenyl-1,4-dihydropyridine-3,5-dicarboxylic acid 3,5-asymmetric disters

Info

Publication number
ZA792804B
ZA792804B ZA792804A ZA792804A ZA792804B ZA 792804 B ZA792804 B ZA 792804B ZA 792804 A ZA792804 A ZA 792804A ZA 792804 A ZA792804 A ZA 792804A ZA 792804 B ZA792804 B ZA 792804B
Authority
ZA
South Africa
Prior art keywords
sub
new
disters
dihydropyridine
asymmetric
Prior art date
Application number
ZA792804A
Other languages
English (en)
Inventor
S Carlsson
P Berntsson
B Ljung
J Gaarder
Original Assignee
Haessle Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=20335348&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA792804(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Haessle Ab filed Critical Haessle Ab
Publication of ZA792804B publication Critical patent/ZA792804B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
    • C07D211/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Peptides Or Proteins (AREA)
ZA792804A 1978-06-30 1979-06-06 New 2,6-dimethyl-4-2,3-disubstituted phenyl-1,4-dihydropyridine-3,5-dicarboxylic acid 3,5-asymmetric disters ZA792804B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE7807404A SE429652B (sv) 1978-06-30 1978-06-30 2.6-dimetyl-4-(2.3-diklorfenyl)-1.4-dihydropyridin-3.5-dikarboxylsyra-3-metylester-5-etylester

Publications (1)

Publication Number Publication Date
ZA792804B true ZA792804B (en) 1980-06-25

Family

ID=20335348

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA792804A ZA792804B (en) 1978-06-30 1979-06-06 New 2,6-dimethyl-4-2,3-disubstituted phenyl-1,4-dihydropyridine-3,5-dicarboxylic acid 3,5-asymmetric disters

Country Status (24)

Country Link
US (1) US4264611A (es)
EP (1) EP0007293B1 (es)
JP (1) JPS559083A (es)
AT (1) ATE1237T1 (es)
AU (1) AU529116B2 (es)
BG (1) BG61420B2 (es)
CA (1) CA1117530A (es)
CS (1) CS241021B2 (es)
CY (1) CY1299A (es)
DD (1) DD144667A5 (es)
DE (1) DE2963150D1 (es)
DK (1) DK148978C (es)
FI (1) FI70573C (es)
HK (1) HK60585A (es)
HU (1) HU178568B (es)
IE (1) IE48650B1 (es)
LU (2) LU88666I2 (es)
NL (2) NL930054I2 (es)
NO (3) NO151965C (es)
NZ (1) NZ190809A (es)
SE (1) SE429652B (es)
SG (1) SG26085G (es)
SU (2) SU856380A3 (es)
ZA (1) ZA792804B (es)

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US6653481B2 (en) * 2000-12-29 2003-11-25 Synthon Bv Process for making amlodipine
JP4625637B2 (ja) 2002-02-22 2011-02-02 シャイア エルエルシー 活性物質送達系及び活性物質を保護し投与する方法
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US7741317B2 (en) 2005-10-21 2010-06-22 Bristol-Myers Squibb Company LXR modulators
ATE551059T1 (de) * 2005-10-26 2012-04-15 Asahi Kasei Pharma Corp Fasudil in kombination mit bosentan zur behandlung von pulmonaler arterieller hypertonie
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CN102827068A (zh) * 2011-06-17 2012-12-19 张锐豪 一种4-(2, 3-二氯苯基)-2, 6-二甲基-1, 4-二氢-5-甲氧基羰基-3-吡啶羧酸的制备方法
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JP2016516804A (ja) 2013-04-17 2016-06-09 ファイザー・インク 心血管疾患を治療するためのｎ−ピペリジン−３−イルベンズアミド誘導体
CN104177286A (zh) * 2014-08-11 2014-12-03 广东东阳光药业有限公司 一种地平类药物的制备方法
WO2016055901A1 (en) 2014-10-08 2016-04-14 Pfizer Inc. Substituted amide compounds
KR101824982B1 (ko) 2015-10-07 2018-02-02 엘지전자 주식회사 차량 및 그 제어방법
CN107952483B (zh) * 2017-12-18 2020-07-28 万华化学集团股份有限公司 一种催化剂，使用该催化剂的反应器，以及一种制备β-苯乙醇的方法
CN108840819B (zh) * 2018-04-02 2021-07-30 常州瑞明药业有限公司 一种非洛地平的制备方法
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US3441648A (en) * 1967-02-07 1969-04-29 Smithkline Corp Compositions and methods for lowering blood pressure with 1,4-dihydropyridines
DE1670824C3 (de) * 1967-03-20 1978-08-03 Bayer Ag, 5090 Leverkusen 1,4-Dihydropyridin-33-dicarbonsäurealkylester
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Also Published As

Publication number Publication date
HK60585A (en) 1985-08-23
LU88306I2 (fr) 1994-05-04
DK275079A (da) 1979-12-31
FI70573B (fi) 1986-06-06
US4264611B1 (es) 1984-07-17
SG26085G (en) 1986-01-24
JPS559083A (en) 1980-01-22
EP0007293A1 (en) 1980-01-23
FI70573C (fi) 1986-09-24
DK148978B (da) 1985-12-09
NL940012I1 (nl) 1994-08-01
NO1994026I1 (no) 1994-12-21
AU529116B2 (en) 1983-05-26
SE7807404L (sv) 1979-12-31
DD144667A5 (de) 1980-10-29
US4264611A (en) 1981-04-28
CS241021B2 (en) 1986-03-13
DK148978C (da) 1986-08-18
SE429652B (sv) 1983-09-19
NO151965B (no) 1985-04-01
NO792112L (no) 1980-01-03
DE2963150D1 (en) 1982-08-12
BG61420B2 (bg) 1997-07-31
ATE1237T1 (de) 1982-07-15
EP0007293B1 (en) 1982-06-23
IE791217L (en) 1979-12-30
AU4831679A (en) 1980-02-07
CA1117530A (en) 1982-02-02
NL930054I1 (nl) 1993-09-01
NO1996006I1 (no) 1996-06-24
NL930054I2 (nl) 1994-02-16
IE48650B1 (en) 1985-04-03
NZ190809A (en) 1982-03-09
HU178568B (en) 1982-05-28
CY1299A (en) 1985-10-18
SU856380A3 (ru) 1981-08-15
JPS6121550B2 (es) 1986-05-27
SU915799A3 (en) 1982-03-23
NO151965C (no) 1985-07-10
LU88666I2 (fr) 1996-02-01
FI792058A (fi) 1979-12-31

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