ZA200903654B - Indazolyl ester and amide derivatives for the treatment of glucocorticoid receptor mediated disorders - Google Patents
Indazolyl ester and amide derivatives for the treatment of glucocorticoid receptor mediated disordersInfo
- Publication number
- ZA200903654B ZA200903654B ZA2009/03654A ZA200903654A ZA200903654B ZA 200903654 B ZA200903654 B ZA 200903654B ZA 2009/03654 A ZA2009/03654 A ZA 2009/03654A ZA 200903654 A ZA200903654 A ZA 200903654A ZA 200903654 B ZA200903654 B ZA 200903654B
- Authority
- ZA
- South Africa
- Prior art keywords
- treatment
- glucocorticoid receptor
- amide derivatives
- receptor mediated
- mediated disorders
- Prior art date
Links
- 102000003676 Glucocorticoid Receptors Human genes 0.000 title 1
- 108090000079 Glucocorticoid Receptors Proteins 0.000 title 1
- -1 Indazolyl ester Chemical class 0.000 title 1
- 150000001408 amides Chemical class 0.000 title 1
- 230000001404 mediated effect Effects 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
- C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US87118406P | 2006-12-21 | 2006-12-21 | |
| US94174507P | 2007-06-04 | 2007-06-04 | |
| US97852607P | 2007-10-09 | 2007-10-09 | |
| PCT/SE2007/001136 WO2008076048A1 (en) | 2006-12-21 | 2007-12-20 | Indazolyl ester and amide derivatives for the treatment of glucocorticoid receptor mediated disorders |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200903654B true ZA200903654B (en) | 2010-09-29 |
Family
ID=39536557
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA2009/03654A ZA200903654B (en) | 2006-12-21 | 2009-05-26 | Indazolyl ester and amide derivatives for the treatment of glucocorticoid receptor mediated disorders |
Country Status (36)
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| TN (1) | TN2009000250A1 (OSRAM) |
| TW (1) | TWI417094B (OSRAM) |
| UY (1) | UY30824A1 (OSRAM) |
| WO (1) | WO2008076048A1 (OSRAM) |
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| JPH081035Y2 (ja) | 1993-06-30 | 1996-01-17 | 伸夫 高橋 | 家庭用雑排水の処理装置 |
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| BR112017000418A2 (pt) | 2014-07-31 | 2017-11-07 | Dow Agrosciences Llc | processo para a preparação de 3-(3-cloro-1h-pirazol-1-il)piridina |
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