MX2009006540A - Derivados de ester y amida de indazolilo para el tratamiento de enfermedades mediadas por un receptor de glucocorticoides. - Google Patents
Derivados de ester y amida de indazolilo para el tratamiento de enfermedades mediadas por un receptor de glucocorticoides.Info
- Publication number
- MX2009006540A MX2009006540A MX2009006540A MX2009006540A MX2009006540A MX 2009006540 A MX2009006540 A MX 2009006540A MX 2009006540 A MX2009006540 A MX 2009006540A MX 2009006540 A MX2009006540 A MX 2009006540A MX 2009006540 A MX2009006540 A MX 2009006540A
- Authority
- MX
- Mexico
- Prior art keywords
- treatment
- amide derivatives
- glucocorticoid receptor
- receptor mediated
- mediated disorders
- Prior art date
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- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
- C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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Abstract
La presente invención se relaciona con nuevos derivados éster o amida de indazolilo, composiciones farmacéuticas que comprenden los derivados, procesos para preparar los nuevos derivados y el uso de los derivados como medicamento (por ejemplo en el tratamiento de un estado de enfermedad inflamatoria).
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
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US87118406P | 2006-12-21 | 2006-12-21 | |
US94174507P | 2007-06-04 | 2007-06-04 | |
US97852607P | 2007-10-09 | 2007-10-09 | |
PCT/SE2007/001136 WO2008076048A1 (en) | 2006-12-21 | 2007-12-20 | Indazolyl ester and amide derivatives for the treatment of glucocorticoid receptor mediated disorders |
Publications (1)
Publication Number | Publication Date |
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MX2009006540A true MX2009006540A (es) | 2009-06-30 |
Family
ID=39536557
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2009006540A MX2009006540A (es) | 2006-12-21 | 2007-12-20 | Derivados de ester y amida de indazolilo para el tratamiento de enfermedades mediadas por un receptor de glucocorticoides. |
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US (4) | US7728030B2 (es) |
EP (1) | EP2102169B1 (es) |
JP (2) | JP5119267B2 (es) |
KR (1) | KR20090091354A (es) |
CN (1) | CN101611015B (es) |
AR (1) | AR064505A1 (es) |
AU (1) | AU2007334659B2 (es) |
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CR (1) | CR10875A (es) |
CY (1) | CY1113269T1 (es) |
DK (1) | DK2102169T3 (es) |
DO (1) | DOP2009000148A (es) |
EA (1) | EA016895B1 (es) |
EC (1) | ECSP099452A (es) |
ES (1) | ES2387584T3 (es) |
GT (1) | GT200900175A (es) |
HK (2) | HK1133651A1 (es) |
HR (1) | HRP20120656T1 (es) |
IL (1) | IL198880A (es) |
JO (1) | JO2754B1 (es) |
MA (1) | MA31087B1 (es) |
MX (1) | MX2009006540A (es) |
MY (1) | MY153270A (es) |
NO (1) | NO20092723L (es) |
NZ (1) | NZ577186A (es) |
PE (1) | PE20081838A1 (es) |
PL (1) | PL2102169T3 (es) |
PT (1) | PT2102169E (es) |
RS (1) | RS52411B (es) |
SA (1) | SA07280740B1 (es) |
SV (1) | SV2009003305A (es) |
TN (1) | TN2009000250A1 (es) |
TW (1) | TWI417094B (es) |
UY (1) | UY30824A1 (es) |
WO (1) | WO2008076048A1 (es) |
ZA (1) | ZA200903654B (es) |
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