CY1113269T1 - Παραγωγα ινδαζολυλ αμιδιου για τη θεραπευτικη αγωγη διαταραχων διαμεσολαβουμενων υπο υποδοχεα γλυκοκορτικοειδων - Google Patents

Παραγωγα ινδαζολυλ αμιδιου για τη θεραπευτικη αγωγη διαταραχων διαμεσολαβουμενων υπο υποδοχεα γλυκοκορτικοειδων

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Publication number
CY1113269T1
CY1113269T1 CY20121100730T CY121100730T CY1113269T1 CY 1113269 T1 CY1113269 T1 CY 1113269T1 CY 20121100730 T CY20121100730 T CY 20121100730T CY 121100730 T CY121100730 T CY 121100730T CY 1113269 T1 CY1113269 T1 CY 1113269T1
Authority
CY
Cyprus
Prior art keywords
indiazolyl
gluccortic
amid
medicines
product
Prior art date
Application number
CY20121100730T
Other languages
English (en)
Inventor
Markus Berger
Jan Dahmén
Anders Eriksson
Balint Gabos
Thomas Hansson
Martin Hemmerling
Krister Henriksson
Svetlana Ivanova
Matti Lepistö
Darren Mckerrecher
af Rosenschöld Magnus Munck
Stinabritt Nilsson
Hartmut Rehwinkel
Camilla Taflin
Karl Edman
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of CY1113269T1 publication Critical patent/CY1113269T1/el

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    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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Abstract

Ενώσεις του τύπου (Ι): Η παρούσα εφεύρεση αφορά νέα παράγωγα ινδαζολυλ εστέρα ή αμιδίου, φαρμακευτικές συνθέσεις που περιλαμβάνουν τέτοια παράγωγα, διεργασίες για την παρασκευή τέτοιων νέων παραγώγων και τη χρήση τέτοιων παραγώγων ως φαρμάκων.
CY20121100730T 2006-12-21 2012-08-13 Παραγωγα ινδαζολυλ αμιδιου για τη θεραπευτικη αγωγη διαταραχων διαμεσολαβουμενων υπο υποδοχεα γλυκοκορτικοειδων CY1113269T1 (el)

Applications Claiming Priority (4)

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US87118406P 2006-12-21 2006-12-21
US94174507P 2007-06-04 2007-06-04
US97852607P 2007-10-09 2007-10-09
EP07852132A EP2102169B1 (en) 2006-12-21 2007-12-20 Indazolyl amide derivatives for the treatment of glucocorticoid receptor mediated disorders

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CY1113269T1 true CY1113269T1 (el) 2016-04-13

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EP2102169A4 (en) 2011-01-05
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ECSP099452A (es) 2009-07-31
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CR10875A (es) 2009-07-20
IL198880A (en) 2013-10-31
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PE20081838A1 (es) 2009-03-14
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CN101611015B (zh) 2012-09-26
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JO2754B1 (en) 2014-03-15
AR064505A1 (es) 2009-04-08
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SV2009003305A (es) 2010-06-09
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