ZA200900070B - Hydroxylated and methoxylated cyclopenta [D] pyrimidines as AKT protein kinase inhibitors - Google Patents

Hydroxylated and methoxylated cyclopenta [D] pyrimidines as AKT protein kinase inhibitors

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Publication number
ZA200900070B
ZA200900070B ZA200900070A ZA200900070A ZA200900070B ZA 200900070 B ZA200900070 B ZA 200900070B ZA 200900070 A ZA200900070 A ZA 200900070A ZA 200900070 A ZA200900070 A ZA 200900070A ZA 200900070 B ZA200900070 B ZA 200900070B
Authority
ZA
South Africa
Prior art keywords
pyrimidines
hydroxylated
protein kinase
kinase inhibitors
akt protein
Prior art date
Application number
ZA200900070A
Other languages
English (en)
Inventor
Ian S Mitchell
James F Blake
Rui Xu
Nicholas C Kallan
Dengming Xiao
Keith Lee Spencer
Josef R Bencsik
Jun Liang
Brian Safina
Birong Zhang
Christine Chabot
Steven Do
Eli M Wallace
Anna L Banka
Stephen T Schlachter
Original Assignee
Array Biopharma Inc
Genentech Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38686743&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA200900070(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Array Biopharma Inc, Genentech Inc filed Critical Array Biopharma Inc
Publication of ZA200900070B publication Critical patent/ZA200900070B/xx

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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ZA200900070A 2006-07-06 2009-01-05 Hydroxylated and methoxylated cyclopenta [D] pyrimidines as AKT protein kinase inhibitors ZA200900070B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US81871806P 2006-07-06 2006-07-06

Publications (1)

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ZA200900070B true ZA200900070B (en) 2010-03-31

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ID=38686743

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ZA200900070A ZA200900070B (en) 2006-07-06 2009-01-05 Hydroxylated and methoxylated cyclopenta [D] pyrimidines as AKT protein kinase inhibitors

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