ZA200605587B - Novel phenylalanine derivative - Google Patents
Novel phenylalanine derivative Download PDFInfo
- Publication number
- ZA200605587B ZA200605587B ZA200605587A ZA200605587A ZA200605587B ZA 200605587 B ZA200605587 B ZA 200605587B ZA 200605587 A ZA200605587 A ZA 200605587A ZA 200605587 A ZA200605587 A ZA 200605587A ZA 200605587 B ZA200605587 B ZA 200605587B
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- ZA
- South Africa
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- pharmaceutically acceptable
- acceptable salts
- carbon atoms
- hydrogen atom
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Classifications
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
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Landscapes
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- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (4)
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| JP2003425347 | 2003-12-22 | ||
| JP2004074943 | 2004-03-16 | ||
| JP2004159919 | 2004-05-28 | ||
| JP2004260319 | 2004-09-07 |
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| EP (3) | EP2803667A1 (de) |
| JP (1) | JP4743659B2 (de) |
| KR (2) | KR101194176B1 (de) |
| CN (2) | CN1917881B (de) |
| AU (1) | AU2004303696B2 (de) |
| BR (1) | BRPI0418026A (de) |
| CA (1) | CA2550843C (de) |
| ES (1) | ES2548853T3 (de) |
| IL (1) | IL176469A (de) |
| NO (1) | NO337628B1 (de) |
| NZ (1) | NZ548420A (de) |
| RU (1) | RU2390520C2 (de) |
| WO (1) | WO2005061466A1 (de) |
| ZA (1) | ZA200605587B (de) |
Families Citing this family (36)
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| BRPI0113331B8 (pt) | 2000-08-18 | 2021-05-25 | Ajinomoto Kk | derivados de fenilalanina ou seus sais parmaceuticamente aceitáveis, antagonista de integrina alfa 4, agente terapêutico ou agente preventivo para doenças inflamatórias, e, composição farmacêutica |
| AU2001290303A1 (en) * | 2000-09-29 | 2002-04-15 | Ajinomoto Co., Inc. | Novel phenylalanine derivatives |
| JP4470219B2 (ja) * | 2002-02-20 | 2010-06-02 | 味の素株式会社 | 新規フェニルアラニン誘導体 |
| EP1595870B1 (de) * | 2003-02-20 | 2015-09-23 | Ajinomoto Co., Inc. | Verfahren zur herstellung eines phenylalaninderivats mit chinazolindionskelett und zwischenprodukt dafür |
| WO2005046697A1 (ja) * | 2003-11-14 | 2005-05-26 | Ajinomoto Co., Inc. | フェニルアラニン誘導体の徐放性経口投与製剤 |
| CN100563658C (zh) * | 2003-11-14 | 2009-12-02 | 味之素株式会社 | 苯丙氨酸衍生物的固体分散体或固体分散体医药制剂 |
| JP4748449B2 (ja) * | 2003-11-27 | 2011-08-17 | 味の素株式会社 | フェニルアラニン誘導体の結晶及びその製造方法 |
| KR101194176B1 (ko) * | 2003-12-22 | 2012-10-24 | 아지노모토 가부시키가이샤 | 신규한 페닐알라닌 유도체 |
| CN101243056B (zh) * | 2005-06-21 | 2013-03-27 | 味之素株式会社 | 苯基丙氨酸衍生物的结晶、其制备方法及其应用 |
| WO2007028789A1 (en) * | 2005-09-07 | 2007-03-15 | Istituto Di Ricerche Di Biologia Molecolare P. Angeletti Spa | Quinazoline derivatives as antiviral agents |
| CN101360736A (zh) * | 2005-11-23 | 2009-02-04 | 阿斯利康(瑞典)有限公司 | L-丙氨酸衍生物 |
| ES2684821T3 (es) | 2005-12-29 | 2018-10-04 | Lexicon Pharmaceuticals, Inc. | Derivados de aminoácidos multicíclicos y métodos de su uso |
| US7834050B2 (en) * | 2006-03-29 | 2010-11-16 | Duke University | Small molecule insulin mimetics absent quinones |
| US20080045521A1 (en) * | 2006-06-09 | 2008-02-21 | Astrazeneca Ab | Phenylalanine derivatives |
| MX297306B (es) * | 2006-11-22 | 2012-03-22 | Ajinomoto Kk | Procedimiento para la produccion de derivados de fenilalanina que tienen estructuras de base de quinazolinodiona e intermediarios para la produccion. |
| WO2008093065A1 (en) * | 2007-01-29 | 2008-08-07 | Astrazeneca Ab | L-ALANINE DERIVATIVES AS α5βL ANTAGONISTS |
| WO2008125811A1 (en) * | 2007-04-11 | 2008-10-23 | Astrazeneca Ab | N-[HETEROARYLCARBONYL]-S-THIENYL-L-ALANINE DERIVATIVES AS α5β1 ANTAGONISTS |
| WO2008133155A1 (ja) | 2007-04-19 | 2008-11-06 | Astellas Pharma Inc. | 二環式ヘテロ環化合物 |
| WO2011094890A1 (en) * | 2010-02-02 | 2011-08-11 | Argusina Inc. | Phenylalanine derivatives and their use as non-peptide glp-1 receptor modulators |
| JP6109568B2 (ja) | 2010-03-29 | 2017-04-05 | Ｅａファーマ株式会社 | フェニルアラニン誘導体の塩の結晶 |
| JP2013530963A (ja) | 2010-06-09 | 2013-08-01 | レセプトス インコーポレイテッド | 新規のｇｌｐ−１受容体安定化薬および調節薬 |
| US9278910B2 (en) | 2011-05-31 | 2016-03-08 | Receptos, Inc. | GLP-1 receptor stabilizers and modulators |
| MX365923B (es) * | 2011-12-12 | 2019-06-20 | Celgene Int Ii Sarl | Derivados de acido carboxilico que comprenden cuatro ciclos, que actuan como moduladores del receptor del peptido 1 similar al glucagon (glp-1) para terapia de enfermedades como la diabetes. |
| US9533985B2 (en) | 2012-04-24 | 2017-01-03 | Ea Pharma Co., Ltd. | Sulfonamide derivative and medicinal use thereof |
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- 2004-12-22 US US11/018,226 patent/US7345049B2/en not_active Expired - Fee Related
- 2004-12-22 ZA ZA200605587A patent/ZA200605587B/en unknown
- 2004-12-22 BR BRPI0418026-7A patent/BRPI0418026A/pt not_active IP Right Cessation
- 2004-12-22 EP EP04808055.0A patent/EP1700850B1/de active Active
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- 2004-12-22 RU RU2006126651/04A patent/RU2390520C2/ru not_active IP Right Cessation
- 2004-12-22 AU AU2004303696A patent/AU2004303696B2/en not_active Ceased
- 2004-12-22 KR KR1020117019338A patent/KR20110098980A/ko not_active Application Discontinuation
- 2004-12-22 EP EP13152904.2A patent/EP2615087A3/de not_active Withdrawn
- 2004-12-22 CN CN201410016206.3A patent/CN103784458B/zh not_active Expired - Fee Related
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