ZA200605587B - Novel phenylalanine derivative - Google Patents
Novel phenylalanine derivative Download PDFInfo
- Publication number
- ZA200605587B ZA200605587B ZA200605587A ZA200605587A ZA200605587B ZA 200605587 B ZA200605587 B ZA 200605587B ZA 200605587 A ZA200605587 A ZA 200605587A ZA 200605587 A ZA200605587 A ZA 200605587A ZA 200605587 B ZA200605587 B ZA 200605587B
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- ZA
- South Africa
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- pharmaceutically acceptable
- acceptable salts
- carbon atoms
- hydrogen atom
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Classifications
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- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
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- C07—ORGANIC CHEMISTRY
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- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
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Landscapes
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- General Health & Medical Sciences (AREA)
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- Life Sciences & Earth Sciences (AREA)
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- Bioinformatics & Cheminformatics (AREA)
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- Transplantation (AREA)
- Dermatology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
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| JP2003425347 | 2003-12-22 | ||
| JP2004074943 | 2004-03-16 | ||
| JP2004159919 | 2004-05-28 | ||
| JP2004260319 | 2004-09-07 |
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| ZA200605587B true ZA200605587B (en) | 2008-02-27 |
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| Application Number | Title | Priority Date | Filing Date |
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| ZA200605587A ZA200605587B (en) | 2003-12-22 | 2004-12-22 | Novel phenylalanine derivative |
Country Status (15)
| Country | Link |
|---|---|
| US (2) | US7345049B2 (de) |
| EP (3) | EP1700850B1 (de) |
| JP (1) | JP4743659B2 (de) |
| KR (2) | KR20110098980A (de) |
| CN (2) | CN103784458B (de) |
| AU (1) | AU2004303696B2 (de) |
| BR (1) | BRPI0418026A (de) |
| CA (1) | CA2550843C (de) |
| ES (1) | ES2548853T3 (de) |
| IL (1) | IL176469A (de) |
| NO (1) | NO337628B1 (de) |
| NZ (1) | NZ548420A (de) |
| RU (1) | RU2390520C2 (de) |
| WO (1) | WO2005061466A1 (de) |
| ZA (1) | ZA200605587B (de) |
Families Citing this family (36)
| Publication number | Priority date | Publication date | Assignee | Title |
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| YU12203A (sh) * | 2000-08-18 | 2006-03-03 | Ajinomoto Co.Inc. | Novi derivati fenilalanina |
| ATE345127T1 (de) * | 2000-09-29 | 2006-12-15 | Ajinomoto Kk | Neue phenylalanin-derivate |
| AU2003211560A1 (en) * | 2002-02-20 | 2003-09-09 | Ajinomoto Co., Inc. | Novel phenylalanine derivative |
| CN100436429C (zh) * | 2003-02-20 | 2008-11-26 | 味之素株式会社 | 具有喹唑二酮骨架的苯丙氨酸衍生物的制造方法及制造中间体 |
| EP1683525B1 (de) * | 2003-11-14 | 2017-05-17 | EA Pharma Co., Ltd. | Phenylalanin-derivat-präparat mit verzögerter freisetzung zur oralen verabreichung |
| DK1683524T3 (da) * | 2003-11-14 | 2011-03-14 | Ajinomoto Kk | Dispergering på fast form eller medicinsk præparat på fast form af phenyalaninderivat |
| JP4748449B2 (ja) * | 2003-11-27 | 2011-08-17 | 味の素株式会社 | フェニルアラニン誘導体の結晶及びその製造方法 |
| KR20110098980A (ko) * | 2003-12-22 | 2011-09-02 | 아지노모토 가부시키가이샤 | 신규한 페닐알라닌 유도체 |
| ES2416354T3 (es) | 2005-06-21 | 2013-07-31 | Ajinomoto Co., Inc. | Cristal de derivado de fenilalanina, método de producción del mismo y uso del mismo |
| WO2007028789A1 (en) * | 2005-09-07 | 2007-03-15 | Istituto Di Ricerche Di Biologia Molecolare P. Angeletti Spa | Quinazoline derivatives as antiviral agents |
| JP2009516730A (ja) * | 2005-11-23 | 2009-04-23 | アストラゼネカ アクチボラグ | Ｌ−アラニン誘導体 |
| AU2006337137B2 (en) * | 2005-12-29 | 2012-06-14 | Tersera Therapeutics Llc | Multicyclic amino acid derivatives and methods of their use |
| US7834050B2 (en) | 2006-03-29 | 2010-11-16 | Duke University | Small molecule insulin mimetics absent quinones |
| JP2009539815A (ja) * | 2006-06-09 | 2009-11-19 | アストラゼネカ アクチボラグ | 固形腫瘍の治療用のａ５ｂ１アンタゴニストとしてのＮ−（ベンゾイル）−Ｏ−［２−（ピリジン−２−イルアミノ）エチル］−Ｌ−チロシン誘導体と関連化合物 |
| MX297306B (es) * | 2006-11-22 | 2012-03-22 | Ajinomoto Kk | Procedimiento para la produccion de derivados de fenilalanina que tienen estructuras de base de quinazolinodiona e intermediarios para la produccion. |
| WO2008093065A1 (en) * | 2007-01-29 | 2008-08-07 | Astrazeneca Ab | L-ALANINE DERIVATIVES AS α5βL ANTAGONISTS |
| WO2008125811A1 (en) * | 2007-04-11 | 2008-10-23 | Astrazeneca Ab | N-[HETEROARYLCARBONYL]-S-THIENYL-L-ALANINE DERIVATIVES AS α5β1 ANTAGONISTS |
| JPWO2008133155A1 (ja) * | 2007-04-19 | 2010-07-22 | アステラス製薬株式会社 | 二環式ヘテロ環化合物 |
| WO2011094890A1 (en) * | 2010-02-02 | 2011-08-11 | Argusina Inc. | Phenylalanine derivatives and their use as non-peptide glp-1 receptor modulators |
| EP2554542B1 (de) | 2010-03-29 | 2015-10-07 | Ajinomoto Co., Inc. | Phenylalaninderivat-hydrochlorid-salzkristall |
| WO2011156655A2 (en) | 2010-06-09 | 2011-12-15 | Receptos, Inc. | Novel glp-1 receptor stabilizers and modulators |
| EP2713722B1 (de) | 2011-05-31 | 2017-03-15 | Receptos, LLC | Neue glp-1-rezeptor-stabilisatoren und -modulatoren |
| CN104080767A (zh) * | 2011-12-12 | 2014-10-01 | 瑞塞普托斯公司 | 新的glp-1受体调节剂 |
| CA2871464C (en) * | 2012-04-24 | 2017-09-26 | Ajinomoto Co., Inc. | Sulfonamide derivatives and their use in the inhibition of .alpha.4.beta.7 integrin-dependent process |
| CN102993105B (zh) * | 2012-12-19 | 2014-06-11 | 西南大学 | 1-甲基-2,4-喹唑啉二酮衍生物及其制备方法和应用 |
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2004
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- 2004-12-22 EP EP04808055.0A patent/EP1700850B1/de active Active
- 2004-12-22 US US11/018,226 patent/US7345049B2/en not_active Expired - Fee Related
- 2004-12-22 EP EP14181015.0A patent/EP2803667A1/de not_active Withdrawn
- 2004-12-22 WO PCT/JP2004/019704 patent/WO2005061466A1/ja active Application Filing
- 2004-12-22 ZA ZA200605587A patent/ZA200605587B/en unknown
- 2004-12-22 EP EP13152904.2A patent/EP2615087A3/de not_active Withdrawn
- 2004-12-22 CN CN201410016206.3A patent/CN103784458B/zh not_active Expired - Fee Related
- 2004-12-22 KR KR1020067014754A patent/KR101194176B1/ko active IP Right Grant
- 2004-12-22 NZ NZ548420A patent/NZ548420A/en not_active IP Right Cessation
- 2004-12-22 CN CN200480041967.9A patent/CN1917881B/zh not_active Expired - Fee Related
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- 2004-12-22 RU RU2006126651/04A patent/RU2390520C2/ru not_active IP Right Cessation
- 2004-12-22 ES ES04808055.0T patent/ES2548853T3/es active Active
- 2004-12-22 AU AU2004303696A patent/AU2004303696B2/en not_active Ceased
- 2004-12-22 JP JP2005516537A patent/JP4743659B2/ja not_active Expired - Fee Related
- 2004-12-22 BR BRPI0418026-7A patent/BRPI0418026A/pt not_active IP Right Cessation
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2006
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- 2006-07-20 NO NO20063372A patent/NO337628B1/no not_active IP Right Cessation
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2007
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