ZA200304810B - Pharmaceutical formulation. - Google Patents
Pharmaceutical formulation. Download PDFInfo
- Publication number
- ZA200304810B ZA200304810B ZA200304810A ZA200304810A ZA200304810B ZA 200304810 B ZA200304810 B ZA 200304810B ZA 200304810 A ZA200304810 A ZA 200304810A ZA 200304810 A ZA200304810 A ZA 200304810A ZA 200304810 B ZA200304810 B ZA 200304810B
- Authority
- ZA
- South Africa
- Prior art keywords
- eudragit
- capsule
- dosage form
- sub
- compartment
- Prior art date
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- 239000008194 pharmaceutical composition Substances 0.000 title claims description 9
- 239000002775 capsule Substances 0.000 claims description 203
- 239000000203 mixture Substances 0.000 claims description 131
- 239000002552 dosage form Substances 0.000 claims description 125
- GLDOVTGHNKAZLK-UHFFFAOYSA-N octadecan-1-ol Chemical group CCCCCCCCCCCCCCCCCCO GLDOVTGHNKAZLK-UHFFFAOYSA-N 0.000 claims description 99
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- 239000000546 pharmaceutical excipient Substances 0.000 claims description 59
- NEDGUIRITORSKL-UHFFFAOYSA-N butyl 2-methylprop-2-enoate;2-(dimethylamino)ethyl 2-methylprop-2-enoate;methyl 2-methylprop-2-enoate Chemical compound COC(=O)C(C)=C.CCCCOC(=O)C(C)=C.CN(C)CCOC(=O)C(C)=C NEDGUIRITORSKL-UHFFFAOYSA-N 0.000 claims description 56
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- 238000004090 dissolution Methods 0.000 claims description 49
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- 229940088679 drug related substance Drugs 0.000 claims description 48
- 239000008186 active pharmaceutical agent Substances 0.000 claims description 40
- 239000007924 injection Substances 0.000 claims description 40
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- FCZYGJBVLGLYQU-UHFFFAOYSA-M sodium;2-[2-[2-[4-(2,4,4-trimethylpentan-2-yl)phenoxy]ethoxy]ethoxy]ethanesulfonate Chemical compound [Na+].CC(C)(C)CC(C)(C)C1=CC=C(OCCOCCOCCS([O-])(=O)=O)C=C1 FCZYGJBVLGLYQU-UHFFFAOYSA-M 0.000 description 1
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4816—Wall or shell material
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4808—Preparations in capsules, e.g. of gelatin, of chocolate characterised by the form of the capsule or the structure of the filling; Capsules containing small tablets; Capsules with outer layer for immediate drug release
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
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GBGB0102342.3A GB0102342D0 (en) | 2001-01-30 | 2001-01-30 | Pharmaceutical formulation |
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ZA200305045A ZA200305045B (en) | 2001-01-30 | 2003-06-27 | Pharmaceutical formulation. |
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ZA200305045A ZA200305045B (en) | 2001-01-30 | 2003-06-27 | Pharmaceutical formulation. |
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CZ (2) | CZ20031980A3 (cs) |
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TW (2) | TWI257871B (cs) |
WO (2) | WO2002060385A2 (cs) |
ZA (2) | ZA200304810B (cs) |
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