YU97583A - Process for obtaining new piperidine derivatives - Google Patents

Process for obtaining new piperidine derivatives

Info

Publication number
YU97583A
YU97583A YU00975/83A YU97583A YU97583A YU 97583 A YU97583 A YU 97583A YU 00975/83 A YU00975/83 A YU 00975/83A YU 97583 A YU97583 A YU 97583A YU 97583 A YU97583 A YU 97583A
Authority
YU
Yugoslavia
Prior art keywords
piperidine derivatives
obtaining new
new piperidine
obtaining
derivatives
Prior art date
Application number
YU00975/83A
Other languages
English (en)
Inventor
J L Archibald
T J Ward
Original Assignee
Wyeth John & Brother Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth John & Brother Ltd filed Critical Wyeth John & Brother Ltd
Publication of YU97583A publication Critical patent/YU97583A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms
    • C07D211/58—Nitrogen atoms attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
YU00975/83A 1980-03-01 1983-05-04 Process for obtaining new piperidine derivatives YU97583A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8007048 1980-03-01
GB8027435 1980-08-22

Publications (1)

Publication Number Publication Date
YU97583A true YU97583A (en) 1983-10-31

Family

ID=26274662

Family Applications (4)

Application Number Title Priority Date Filing Date
YU00473/81A YU47381A (en) 1980-03-01 1981-02-24 Process for obtaining new piperidine derivatives
YU00973/83A YU97383A (en) 1980-03-01 1983-05-04 Process for obtaining new piperidine derivatives
YU00974/83A YU97483A (en) 1980-03-01 1983-05-04 Process for obtaining new piperidine derivatives
YU00975/83A YU97583A (en) 1980-03-01 1983-05-04 Process for obtaining new piperidine derivatives

Family Applications Before (3)

Application Number Title Priority Date Filing Date
YU00473/81A YU47381A (en) 1980-03-01 1981-02-24 Process for obtaining new piperidine derivatives
YU00973/83A YU97383A (en) 1980-03-01 1983-05-04 Process for obtaining new piperidine derivatives
YU00974/83A YU97483A (en) 1980-03-01 1983-05-04 Process for obtaining new piperidine derivatives

Country Status (20)

Country Link
US (2) US4426387A (xx)
EP (1) EP0035374B1 (xx)
KR (4) KR850000630B1 (xx)
AU (1) AU542950B2 (xx)
CA (1) CA1173037A (xx)
DE (1) DE3168564D1 (xx)
DK (1) DK164546C (xx)
EG (1) EG16004A (xx)
ES (4) ES8203840A1 (xx)
FI (1) FI77231C (xx)
GR (1) GR73576B (xx)
HU (1) HU187768B (xx)
IE (1) IE52014B1 (xx)
IL (1) IL62200A (xx)
NO (1) NO156864C (xx)
NZ (1) NZ196324A (xx)
PH (1) PH17019A (xx)
PL (4) PL128409B1 (xx)
PT (1) PT72562B (xx)
YU (4) YU47381A (xx)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8528235D0 (en) * 1985-11-15 1985-12-18 Wyeth John & Brother Ltd Heterocyclic compounds
US4508722A (en) * 1981-05-18 1985-04-02 Eli Lilly And Company 1-Benzoyl-3-(arylpyridyl)urea compounds
ATE27152T1 (de) * 1982-04-07 1987-05-15 Ici Plc Chinolin-derivate.
DE3377796D1 (en) * 1982-05-04 1988-09-29 Ici Plc Quinoline derivatives
FR2527205A1 (fr) * 1982-05-18 1983-11-25 Bouchara Emile Nouvelles phenyloxoalcoyl piperidines, leurs procedes d'obtention et les compositions pharmaceutiques en renfermant
EP0157762B1 (fr) * 1983-09-19 1990-08-08 Bouchara S.A. Nouvelles piperidinoguanidines substituees, leur procede de preparation et les compositions pharmaceutiques en renfermant
US4569933A (en) * 1984-04-13 1986-02-11 Cornu Pierre Jean Antihypertensive substituted derivatives of 2,5-diamino 1,4-diazole
GB8528234D0 (en) * 1985-11-15 1985-12-18 Wyeth John & Brother Ltd Heterocyclic compounds
US4709094A (en) * 1986-07-10 1987-11-24 State Of Oregon, Acting By And Through The Oregon State Board Of Higher Education, Acting For And On Behalf Of The Oregon Health Sciences University And The University Of Oregon Sigma brain receptor ligands and their use
US5502255A (en) * 1986-07-10 1996-03-26 State Of Oregon Acting By And Through The Oregon State Board Of Higher Education, Acting For And On Behalf Of The Oregon Health Sciences University And The University Of Oregon Substituted guanidines having high binding to the sigma receptor and the use thereof
US5312840A (en) * 1986-07-10 1994-05-17 State Of Oregon, Acting By And Through The Oregon State Board Of Higher Education Substituted guanidines having high binding to the sigma receptor and the use thereof
EP0343307A1 (en) * 1988-05-26 1989-11-29 Fabrica Espanola De Productos Quimicos Y Farmaceuticos, S.A. 4-Piperidinealkanamine derivatives
GR1000662B (el) * 1988-07-01 1992-09-25 Janssen Pharmaceutica Nv Μεθοδος παρασκευης cis-ν-(3-μεθοξυ-4-πιπεριδινυλο)βενζαμιδιων.
DK0517852T3 (da) 1990-03-02 2002-10-07 Oregon State Tri- og tetrasubstituerede guanidinerog disses anvendelse som excitatoriske aminosyre-antagonister
US5262568A (en) * 1990-03-02 1993-11-16 State Of Oregon Tri- and tetra-substituted guanidines and their use as excitatory amino acid antagonists
FR2662162B1 (fr) * 1990-05-18 1995-01-20 Adir Nouveaux derives de l'amino piperidine, de l'amino pyrrolidine et de l'amino perhydroazepine, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent.
EP0532642A1 (en) * 1990-05-25 1993-03-24 STATE OF OREGON, acting through OREGON STATE BOARD OF HIGHER EDUCATION, acting for OREGON HEALTH SC. UNIV. AND UNIV. OF OREGON Substituted guanidines having high binding to the sigma receptor and the use thereof
US5403861A (en) * 1991-02-08 1995-04-04 Cambridge Neuroscience, Inc. Substituted guanidines and derivatives thereof as modulators of neurotransmitter release and novel methodology for identifying neurotransmitter release blockers
US5847006A (en) * 1991-02-08 1998-12-08 Cambridge Neuroscience, Inc. Therapeutic guanidines
US5741661A (en) * 1991-02-08 1998-04-21 Cambridge Neuroscience, Inc. Substituted guanidines and derivatives thereof as modulators of neurotransmitter release and novel methodology for identifying neurotransmitter release blockers
FR2690158B1 (fr) * 1992-04-17 1994-07-22 Sanofi Elf Nouveau derive arylpiperidinique, procede pour sa preparation et compositions pharmaceutiques le contenant.
KR20030097618A (ko) * 1993-05-27 2003-12-31 캠브리지 뉴로사이언스, 인코포레이티드 치료용 치환 구아니딘류
US5739135A (en) * 1993-09-03 1998-04-14 Bristol-Myers Squibb Company Inhibitors of microsomal triglyceride transfer protein and method
WO1995014461A1 (en) * 1993-11-23 1995-06-01 Cambridge Neuroscience, Inc. Therapeutic substituted guanidines
CA2182302A1 (en) 1994-02-03 1995-08-10 Stanley M. Goldin Therapeutic guanidines
US6143791A (en) * 1994-02-03 2000-11-07 Cambridge Neuroscience, Inc. Therapeutic guanidines
US7351743B1 (en) 1994-02-03 2008-04-01 Wyeth Therapeutic guanidines
US6787569B1 (en) 1994-02-03 2004-09-07 Cambridge Neuroscience, Inc. Therapeutic guanidines
US6025355A (en) 1997-05-19 2000-02-15 Cambridge Neuroscience, Inc. Pharmaceutically active compounds and methods of use
US6242198B1 (en) 1996-07-25 2001-06-05 Cambridge Neuroscience, Inc. Methods of treatment of eye trauma and disorders
US6756389B2 (en) 1996-08-09 2004-06-29 Cambridge Neuroscience, Inc. Pharmaceutically active compounds and methods of use
DE19824470A1 (de) 1998-05-30 1999-12-02 Boehringer Ingelheim Pharma Neue Neurokininantagonisten, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3072663A (en) * 1961-09-25 1963-01-08 Warner Lambert Pharmaceutical Polyalkyl substituted-4-guanidopiperidines
US3171838A (en) * 1961-10-10 1965-03-02 Res Lab Dr C Janssen N V Aroylalkyl and hydroxyaralkyl derivatives of 4-(n-arylalkanamido)-piperidines and related compounds
US3161637A (en) * 1961-10-10 1964-12-15 Res Lab Dr C Janssen N V 1-(gamma-aroyl-propyl)-4-(nu-arylcarbonyl amino) piperidines and related compounds
GB1411782A (en) * 1972-02-24 1975-10-29 Wyeth John & Brother Ltd Piperidine derivatives
GB1411783A (en) * 1972-02-24 1975-10-29 Wyeth John & Brother Ltd Piperidine derivatives
US3910930A (en) * 1973-01-04 1975-10-07 Janssen Pharmaceutica Nv 1-{55 1-{8 2-(1,4-Benzodioxan-2-yl)-2-hydroxyethyl{9 -4-piperidyl{56 -2-benzimidazolinones
US4177279A (en) * 1973-10-10 1979-12-04 John Wyeth & Brother Ltd. 1-[(3-Indolyl)-alkyl]-piperidyl ureas and hypotensive compositions
GB1459506A (en) * 1974-02-18 1976-12-22 Wyeth John & Brother Ltd Piperidine derivatives
JPS5152176A (xx) * 1974-10-12 1976-05-08 Yoshitomi Pharmaceutical
AU500990B2 (en) * 1975-07-25 1979-06-07 John Wyeth & Brother Limited Piperidine derivatives
JPS6039680B2 (ja) * 1975-12-22 1985-09-06 日本化薬株式会社 ３‐（メチルメルカプト）プロピルアミノブレオマイシンの製造法
JPS5285174A (en) * 1976-01-05 1977-07-15 Yoshitomi Pharmaceut Ind Ltd Novel urea or thiourea derivatives
GB1582239A (en) * 1976-12-11 1981-01-07 Wyeth John & Brother Ltd Piperidin-4-yl ureas and thioureas
GB1561023A (en) * 1977-04-22 1980-02-13 Beecham Group Ltd 2-methoxy - 5 - chloro aniline derivatives
IN148482B (xx) * 1977-06-03 1981-03-07 Pfizer
EP0000485A1 (de) * 1977-07-08 1979-02-07 Ciba-Geigy Ag Piperidino-propanole, ihre Herstellung und pharmazeutische Präparate die diese enthalten
US4281132A (en) * 1977-10-29 1981-07-28 John Wyeth & Brother Limited Piperidino ureas and thioureas
GB1586817A (en) * 1977-12-01 1981-03-25 Wyeth John & Brother Ltd Indole derivatives
US4169202A (en) * 1978-06-05 1979-09-25 American Home Products Corporation Process for preparing 4,5-dihydro-4-oxofuran-2-carboxylic acid derivatives
GB2034305B (en) * 1978-10-24 1982-12-22 Wyeth John & Brother Ltd Preparation of piperidine derivatives

Also Published As

Publication number Publication date
PL135545B1 (en) 1985-11-30
ES499716A0 (es) 1982-05-01
ES509163A0 (es) 1983-02-01
NO810610L (no) 1981-09-02
DE3168564D1 (en) 1985-03-14
EG16004A (en) 1986-12-30
NZ196324A (en) 1983-09-02
KR850000631B1 (ko) 1985-05-06
IL62200A0 (en) 1981-03-31
PL229830A1 (xx) 1982-11-22
DK164546C (da) 1992-11-30
HU187768B (en) 1986-02-28
IL62200A (en) 1984-09-30
KR830005140A (ko) 1983-08-03
YU97483A (en) 1983-10-31
IE810392L (en) 1981-09-01
DK164546B (da) 1992-07-13
PT72562A (en) 1981-03-01
ES8302658A1 (es) 1983-02-01
NO156864B (no) 1987-08-31
EP0035374B1 (en) 1985-01-30
PL234318A1 (xx) 1982-08-16
FI77231C (fi) 1989-02-10
FI810587L (fi) 1981-09-02
ES509165A0 (es) 1983-02-01
ES8302657A1 (es) 1983-02-01
KR850002008A (ko) 1985-04-10
KR850002009A (ko) 1985-04-10
EP0035374A3 (en) 1981-11-11
KR850001035B1 (ko) 1985-07-19
AU542950B2 (en) 1985-03-28
ES509164A0 (es) 1983-02-01
IE52014B1 (en) 1987-05-27
PL128510B1 (en) 1984-02-29
ES8302656A1 (es) 1983-02-01
PH17019A (en) 1984-05-11
PL128409B1 (en) 1984-01-31
PL234317A1 (xx) 1982-08-16
DK87881A (da) 1981-09-02
US4563466A (en) 1986-01-07
PT72562B (en) 1982-06-20
FI77231B (fi) 1988-10-31
PL129174B1 (en) 1984-04-30
AU6761481A (en) 1981-09-10
EP0035374A2 (en) 1981-09-09
YU97383A (en) 1983-10-31
ES8203840A1 (es) 1982-05-01
KR850000630B1 (ko) 1985-05-06
KR850002007A (ko) 1985-05-06
GR73576B (xx) 1984-03-20
KR850001063B1 (ko) 1985-07-25
PL234316A1 (en) 1983-11-07
YU47381A (en) 1983-10-31
NO156864C (no) 1987-12-09
US4426387A (en) 1984-01-17
CA1173037A (en) 1984-08-21

Similar Documents

Publication Publication Date Title
YU97583A (en) Process for obtaining new piperidine derivatives
YU221681A (en) Process for obtaining n-arylbenzamide derivatives
YU281081A (en) Process for preparing 1-sulfo-2-oxo-azetidine derivatives
YU144288A (en) Process for obtaining new substituted pyrimidins
YU227181A (en) Process for obtaining 3-aryl-5-isothiazole derivatives
PT73186B (en) Process for preparing pyrazolopyrydazine derivatives
YU126281A (en) Process for obtaining new pyridoxine derivatives
YU98081A (en) Process for obtaining imidosulfamide derivatives
DE3160156D1 (en) Process for preparing vinylphosphonic-acid derivatives
YU45076B (en) Process for obtaining new alphasulphonyloxiketone-acethale
YU42734B (en) Process for obtaining new imidazolyl-pyridine
YU42592B (en) Process for preparing 3-amino-propoxyphenyl derivatives
YU42236B (en) Process for obtaining new 1-(4-aryl-cyclohexyl)piperidine derivatives
YU81181A (en) Process for obtaining substituted derivatives
YU277781A (en) Process for obtaining new acylcarbamides
HU182341B (en) Process for preparing new substituted phenoxy-amino-propanol derivatives
YU252981A (en) Process for obtaining 11-dodecene-1-yl derivatives
PT74153B (en) Process for preparing oxadiazolopyrimidine derivatives
YU159481A (en) Process for preparing dibenzindole derivatives
YU73179A (en) Process for obtaining substituted n-iminomethyl piperidine
PT73457A (en) Process for preparing heteroprostaglandin derivatives
YU42413B (en) Process for obtaining dephenylether derivatives
YU70881A (en) New process for obtaining new 2-haloacetamides
SG65486G (en) Process for preparing 16-hydroxy-17-aminoprepnane derivatives
YU246381A (en) Process for obtaining cephalexine derivatives