UY29686A1 - Proceso para producir 3-oxo-pregn-4-eno-21, 17-carbolactonas por oxidación libre de metales de 17-(3-hidroxipropil)-3,17-dihidroxiandrostanos. - Google Patents

Proceso para producir 3-oxo-pregn-4-eno-21, 17-carbolactonas por oxidación libre de metales de 17-(3-hidroxipropil)-3,17-dihidroxiandrostanos.

Info

Publication number
UY29686A1
UY29686A1 UY29686A UY29686A UY29686A1 UY 29686 A1 UY29686 A1 UY 29686A1 UY 29686 A UY29686 A UY 29686A UY 29686 A UY29686 A UY 29686A UY 29686 A1 UY29686 A1 UY 29686A1
Authority
UY
Uruguay
Prior art keywords
oxo
carbolactones
pregn
eno
produce
Prior art date
Application number
UY29686A
Other languages
English (en)
Spanish (es)
Inventor
Carsten Seilz
Hartmut Seba
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35744678&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY29686(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Ag filed Critical Schering Ag
Publication of UY29686A1 publication Critical patent/UY29686A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002—Carbocyclic rings fused
    • C07J53/004—3 membered carbocyclic rings
    • C07J53/008—3 membered carbocyclic rings in position 15/16

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
UY29686A 2005-07-21 2006-07-20 Proceso para producir 3-oxo-pregn-4-eno-21, 17-carbolactonas por oxidación libre de metales de 17-(3-hidroxipropil)-3,17-dihidroxiandrostanos. UY29686A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP05090214.7A EP1746101B2 (de) 2005-07-21 2005-07-21 Verfahren zur Herstellung von 3-Oxo-pregn-4-en-21,17-carbolactonen durch die metallfreie Oxidation von 17-(3-hydroxypropyl)-3,17-dihydroxyandrostanen

Publications (1)

Publication Number Publication Date
UY29686A1 true UY29686A1 (es) 2007-02-28

Family

ID=35744678

Family Applications (1)

Application Number Title Priority Date Filing Date
UY29686A UY29686A1 (es) 2005-07-21 2006-07-20 Proceso para producir 3-oxo-pregn-4-eno-21, 17-carbolactonas por oxidación libre de metales de 17-(3-hidroxipropil)-3,17-dihidroxiandrostanos.

Country Status (22)

Country Link
US (2) US20070049747A1 (cg-RX-API-DMAC7.html)
EP (1) EP1746101B2 (cg-RX-API-DMAC7.html)
JP (2) JP5345843B2 (cg-RX-API-DMAC7.html)
CN (1) CN101223186B (cg-RX-API-DMAC7.html)
AR (1) AR055993A1 (cg-RX-API-DMAC7.html)
AT (1) ATE403668T1 (cg-RX-API-DMAC7.html)
CY (1) CY1110411T1 (cg-RX-API-DMAC7.html)
DE (1) DE502005004948D1 (cg-RX-API-DMAC7.html)
DK (1) DK1746101T4 (cg-RX-API-DMAC7.html)
DO (1) DOP2006000172A (cg-RX-API-DMAC7.html)
ES (1) ES2311927T5 (cg-RX-API-DMAC7.html)
GT (1) GT200600321A (cg-RX-API-DMAC7.html)
MY (1) MY147795A (cg-RX-API-DMAC7.html)
PE (2) PE20070215A1 (cg-RX-API-DMAC7.html)
PL (1) PL1746101T5 (cg-RX-API-DMAC7.html)
PT (1) PT1746101E (cg-RX-API-DMAC7.html)
SI (1) SI1746101T2 (cg-RX-API-DMAC7.html)
SV (1) SV2007002621A (cg-RX-API-DMAC7.html)
TW (1) TWI392683B (cg-RX-API-DMAC7.html)
UA (1) UA100092C2 (cg-RX-API-DMAC7.html)
UY (1) UY29686A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA200801674B (cg-RX-API-DMAC7.html)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI1746101T2 (sl) * 2005-07-21 2014-09-30 Bayer Pharma Aktiengesellschaft Postopek za pripravo 3-okso-pregn-4-en-21,17-karbolaktonov z oksidacijo 17-(3-hidroksipropil)-3,17-dihidroksiandrostanov brez uporabe kovine
EP2265629B1 (en) * 2008-03-05 2015-06-24 Evestra, Inc. Bismethylene-17 carbolactones and related uses
DE102008026793A1 (de) * 2008-06-02 2009-12-03 Bayer Schering Pharma Aktiengesellschaft C-Ring-substituierte Pregn-4-en-21,17-carbolactone, sowie diese enthaltende pharmazeutische Präparate
US8222237B2 (en) * 2008-11-25 2012-07-17 Evestra, Inc. Progestational 3-(6,6-ethylene-17B-hydroxy-3-oxo-17A-pregna-4-ene-17A-yl)propionic acid G-lactones
US8334375B2 (en) * 2009-04-10 2012-12-18 Evestra, Inc. Methods for the preparation of drospirenone
ES2432063T3 (es) 2009-06-16 2013-11-29 Crystal Pharma, S.A.U. Procedimiento para la obtención de 17-espirolactonas en esteroides
CN101775057B (zh) * 2010-02-09 2014-07-16 浙江仙琚制药股份有限公司 屈螺酮及其中间体的制备方法
CN101830959B (zh) * 2010-05-27 2012-07-18 杭州龙山化工有限公司 一种曲螺酮的合成方法
AR081670A1 (es) 2010-06-29 2012-10-10 Leon Farma Sa Lab Composicion farmaceutica que comprende drospirenona y kit anticonceptivo
US10849857B2 (en) 2010-07-28 2020-12-01 Laboratorios Leon Farma Sa Pharmaceutical compositions comprising active drugs, contraceptive kits comprising active drugs, and methods of administering the same
US11351122B1 (en) 2010-07-28 2022-06-07 Laboratorios Leon Farma Sa Synthetic progestogens and pharmaceutical compositions comprising the same
WO2012107513A1 (en) 2011-02-10 2012-08-16 Crystal Pharma, S.A.U. Process for obtaining drospirenone
CN102746370A (zh) * 2011-04-22 2012-10-24 天津金耀集团有限公司 一种氧化合成孕甾11位酮基的新工艺
KR101672109B1 (ko) * 2012-01-13 2016-11-02 쌩-고벵 글래스 프랑스 단열 창유리 유닛용 스페이서
CN102887934B (zh) * 2012-09-20 2015-05-27 杭州福斯特药业有限公司 一种屈螺酮的制备方法
WO2014167386A1 (en) * 2013-04-12 2014-10-16 Industriale Chimica S.R.L. Process for the preparation of drospirenone
CN104163846A (zh) * 2013-05-17 2014-11-26 上海创诺制药有限公司 一种制备曲螺酮的方法
KR20160095128A (ko) 2013-12-12 2016-08-10 쌩-고벵 글래스 프랑스 개선된 밀봉을 갖는 이중 글레이징
WO2015086459A1 (de) 2013-12-12 2015-06-18 Saint-Gobain Glass France Abstandshalter für isolierverglasungen mit extrudiertem dichtprofil
CN104788524B (zh) * 2014-01-16 2016-07-06 浙江仙居君业药业有限公司 一种19-去甲-4-雄甾烯-3,17-二酮的制备方法
WO2015197491A1 (de) 2014-06-27 2015-12-30 Saint-Gobain Glass France Isolierverglasung mit abstandhalter und verfahren zur herstellung
PL3161237T3 (pl) 2014-06-27 2018-12-31 Saint-Gobain Glass France Oszklenie zespolone z elementem dystansowym i sposób wytwarzania takiego oszklenia oraz jego zastosowanie jako oszklenia budynku
BR112017003684B1 (pt) 2014-09-25 2022-04-05 Saint-Gobain Glass France Espaçador para unidades de envidraçamento isolantes
KR20170109616A (ko) 2015-03-02 2017-09-29 쌩-고벵 글래스 프랑스 절연 글레이징용 유리 섬유-강화 스페이서
CN113750108B (zh) 2015-06-23 2025-08-19 莱昂实验室制药股份有限公司 用于过重女性患者的基于屈螺酮的避孕药
EP3108889A1 (en) 2015-06-23 2016-12-28 Philippe Perrin Drospirenone-based contraceptive for a female patient affected with excess weight

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4069219A (en) 1976-12-27 1978-01-17 G. D. Searle & Co. 7ξ-(Alkoxycarbonyl)-6ξ-alkyl/halo-17-hydroxy-3-oxo-17α-pregn-4-ene-21-carboxylic acid γ-lactones and corresponding 21-carboxylic acids, their salts, and esters
DE3026783C2 (de) 1980-07-11 1982-07-29 Schering Ag, 1000 Berlin Und 4619 Bergkamen Verfahren zur Herstellung von 5β-Hydroxy-δ↑6↑-steroiden
DE3042136A1 (de) 1980-11-03 1982-06-09 Schering Ag, 1000 Berlin Und 4619 Bergkamen Verfahren zur herstellung von 3 (beta), 7 (beta) -dihydroxy- (delta) (pfeil hoch)5(pfeil hoch) -steroiden
ATE15206T1 (de) 1981-09-21 1985-09-15 Schering Ag 3-beta,7-beta,15-alpha-trihydroxy-5-androsten-1 - one, ihre 3,15-trimethylessigsaeure-ester und ihre herstellung.
US5106995A (en) 1989-05-05 1992-04-21 Isp Investments Inc. Production of lactones from diols
DE3916112A1 (de) * 1989-05-16 1990-11-22 Schering Ag Dihydrospirorenon als antiandrogen
DE19633685C1 (de) * 1996-08-12 1997-10-09 Schering Ag Verfahren zur Herstellung von Drospirenon (6beta,7beta;15 beta,16beta-Dimethyl-en-3-oxo-17alpha-pregn-4-en-21,17-carbolacton, DRSP) sowie 7alpha-(3-Hydroxy-1-propyl)-6beta,7beta;15beta, 16beta-dimethylen-5beta-androstan-3beta,5,17beta-triol (ZK 92836) und 6beta,7beta;15beta,16beta-dimethylen-5beta-hydroxy-3-oxo-17alpha-androstan-21,17-carbolacton (90965) als Zwischenprodukte des Verfahrens
WO2004016640A2 (en) * 2002-08-16 2004-02-26 Pharmacia & Upjohn Company Llc 5 ANDROSTEN-3β-OL STEROID INTERMEDIATES AND PROCESSES FOR THEIR PREPARATION
JP2005027184A (ja) * 2003-07-04 2005-01-27 Seiko Epson Corp 高周波複合部品
ITMI20040367A1 (it) * 2004-03-01 2004-06-01 Ind Chimica Srl Processo per la preparazione di drospirenone
ITMI20042338A1 (it) * 2004-12-06 2005-03-06 Ind Chimica Srl Processo per la preparazione di drospirenone
US7319154B2 (en) * 2005-07-21 2008-01-15 Bayer Schering Pharma Ag Process for the production of 3-oxo-pregn-4-ene-21, 17-carbolactones by the metal free oxidation of 17-(3-hydroxypropyl)-3, 17-dihydroxyandrostanes
SI1746101T2 (sl) * 2005-07-21 2014-09-30 Bayer Pharma Aktiengesellschaft Postopek za pripravo 3-okso-pregn-4-en-21,17-karbolaktonov z oksidacijo 17-(3-hidroksipropil)-3,17-dihidroksiandrostanov brez uporabe kovine
US20080032147A1 (en) * 2005-08-26 2008-02-07 Thomas Neel Medium density fibreboard

Also Published As

Publication number Publication date
MY147795A (en) 2013-01-31
CN101223186B (zh) 2012-09-05
EP1746101B2 (de) 2014-05-14
ZA200801674B (en) 2009-08-26
PE20131303A1 (es) 2013-11-27
UA100092C2 (en) 2012-11-12
CN101223186A (zh) 2008-07-16
CY1110411T1 (el) 2015-04-29
US8658788B2 (en) 2014-02-25
PL1746101T5 (pl) 2014-11-28
PT1746101E (pt) 2008-10-27
DK1746101T4 (da) 2014-08-11
ES2311927T5 (es) 2014-09-08
SI1746101T1 (sl) 2009-02-28
ATE403668T1 (de) 2008-08-15
PL1746101T3 (pl) 2009-01-30
EP1746101B1 (de) 2008-08-06
DE502005004948D1 (de) 2008-09-18
US20070049747A1 (en) 2007-03-01
DK1746101T3 (da) 2008-11-24
JP2013177450A (ja) 2013-09-09
ES2311927T3 (es) 2009-02-16
GT200600321A (es) 2007-02-23
DOP2006000172A (es) 2007-02-15
PE20070215A1 (es) 2007-04-11
TWI392683B (zh) 2013-04-11
AR055993A1 (es) 2007-09-12
US20110275796A1 (en) 2011-11-10
TW200716660A (en) 2007-05-01
JP5345843B2 (ja) 2013-11-20
SI1746101T2 (sl) 2014-09-30
SV2007002621A (es) 2007-12-12
EP1746101A1 (de) 2007-01-24
JP2009501753A (ja) 2009-01-22

Similar Documents

Publication Publication Date Title
UY29686A1 (es) Proceso para producir 3-oxo-pregn-4-eno-21, 17-carbolactonas por oxidación libre de metales de 17-(3-hidroxipropil)-3,17-dihidroxiandrostanos.
IN2012DN00580A (cg-RX-API-DMAC7.html)
AR066773A1 (es) Proceso para preparar alcoxidos de metales alcalinos
UA103794C2 (en) Liposome composition
MX2009005813A (es) Procedimiento para la preparacion de betamimeticos.
BRPI1015572A2 (pt) material de adição para a brasagem de chapas.
CU23757B7 (es) Bencilaminas, un proceso para su producción y su uso como agentes anti-inflamatorios
ECSP088124A (es) Proceso para producir 3-oxo-pregn-4-eno-21,17-carbolactonas por oxidación libre de metales de 17-(3-hidroxipropil)-3,17-dihidroxiandrostanos
TW200714632A (en) Manufacture of polytrimethylene ether glycol
TW200640914A (en) Novel processes for the preparation of a benzofuran
EP1860103A4 (en) ANTICANCER COMPOUND, ITS INTERMEDIATE AND METHODS OF PRODUCTION
CU23609B7 (es) Proceso para producir 3-oxo-pregn-4-eno-21,17-carbolactonas por oxidación libre de metales de 17-(3-hidroxipropil)-3,17-dihidroxiandrostanos
ATE496923T1 (de) Neues verfahren für die zubereitung von 3-methyl- 4-phenylisoxazoloä3,4-düpyridazin-7(6h)-on
MX2009008093A (es) Procedimientos para la preparacion de compuestos de urea sustituidos con piperidinilo.
MY151052A (en) Cu-zn-al catalyst promoted with palladium for hydrogen production from methanol
TW200740739A (en) Process for preparing ethylcyclohexane by selectively hydrogenating 4-vinylcyclohexene
TH86966A (th) กรรมวิธีสำหรับการผลิต 3-ออกโซ-เพรกน-4-อีน-21,17-คาร์โบแลคโตน โดยเมทาล-ฟรี ออกซิเดชั่น ของ 17-(3-ไฮดรอกซีโพรพิล)-3,17-ไดไฮดรอกซีแอนโดรสเตน
MX2009003196A (es) Proceso para la preparacion de y-butirolactonas.
MX2009014191A (es) Procedimiento para la preparacion de derivados de dioxazina.
SG155231A1 (en) Process for synthesis of dialkoxyorganoboranes
MY166606A (en) Mo-ni-cu catalyst on y-al2o3 support for hydrogen production from methanol
RU2006116621A (ru) Сплав на основе молибдена

Legal Events

Date Code Title Description
110 Patent granted

Effective date: 20181213