UA128210C2 - Аналог glp-1 - Google Patents

Аналог glp-1 Download PDF

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Publication number
UA128210C2
UA128210C2 UAA202006178A UAA202006178A UA128210C2 UA 128210 C2 UA128210 C2 UA 128210C2 UA A202006178 A UAA202006178 A UA A202006178A UA A202006178 A UAA202006178 A UA A202006178A UA 128210 C2 UA128210 C2 UA 128210C2
Authority
UA
Ukraine
Prior art keywords
ethoxy
resin
tert
amino
acid
Prior art date
Application number
UAA202006178A
Other languages
English (en)
Ukrainian (uk)
Inventor
Раджаманнар Тхеннаті
Раджаманнар Тхеннати
Нішітх Чатурведі
Нишитх Чатурведи
Вінод Сампатрао Бураде
Винод Сампатрао Бураде
Прадіп Дінеш Шахі
Прадип Динеш Шахи
Мутхукумаран Натараджан
Равішанкара Мадаваті Нагараджа
Равишанкара Мадавати Нагараджа
Рішіт Мансухлал Залавадія
Ришит Мансухлал Залавадия
Кунал Пандья
Бріджешкумар Пател
Бриджешкумар Пател
Дхірен Рамешчандра Джоші
Дхирен Рамешчандра Джоши
Крунал Харішбхай Соні
Крунал Харишбхай Сони
Абхішек Тіварі
Абхишек Тивари
Віпулкумар Шанкарбхай Пател
Випулкумар Шанкарбхай Пател
Original Assignee
Сан Фармасьютікал Індастріз Лімітед
Сан Фармасьютикал Индастриз Лимитед
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Сан Фармасьютікал Індастріз Лімітед, Сан Фармасьютикал Индастриз Лимитед filed Critical Сан Фармасьютікал Індастріз Лімітед
Publication of UA128210C2 publication Critical patent/UA128210C2/uk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/605—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/26—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Endocrinology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Obesity (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Zoology (AREA)
  • Biophysics (AREA)
  • Epidemiology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Toxicology (AREA)
  • Biochemistry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Immunology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Transmission And Conversion Of Sensor Element Output (AREA)
UAA202006178A 2018-04-05 2019-04-05 Аналог glp-1 UA128210C2 (uk)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
IN201821013109 2018-04-05
IN201821040474 2018-10-26
IN201821040468 2018-10-26
PCT/IB2019/052835 WO2019193576A1 (en) 2018-04-05 2019-04-05 Novel glp-1 analogues

Publications (1)

Publication Number Publication Date
UA128210C2 true UA128210C2 (uk) 2024-05-08

Family

ID=66589592

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA202006178A UA128210C2 (uk) 2018-04-05 2019-04-05 Аналог glp-1

Country Status (33)

Country Link
US (7) US11447535B2 (https=)
EP (3) EP4364751A3 (https=)
JP (2) JP7250814B2 (https=)
KR (2) KR20250065720A (https=)
CN (3) CN117964735A (https=)
AU (3) AU2019247936C1 (https=)
BR (1) BR112020020419A2 (https=)
CA (1) CA3095988A1 (https=)
CL (1) CL2020002574A1 (https=)
CO (1) CO2020012425A2 (https=)
CY (1) CY1125528T1 (https=)
DK (2) DK3774862T3 (https=)
EC (1) ECSP20070185A (https=)
ES (2) ES2925678T3 (https=)
FI (1) FI4122954T3 (https=)
HR (2) HRP20240749T1 (https=)
HU (2) HUE060135T2 (https=)
IL (1) IL277483B1 (https=)
JO (1) JOP20200251B1 (https=)
LT (2) LT3774862T (https=)
MX (2) MX2020010505A (https=)
MY (1) MY202560A (https=)
PE (1) PE20211417A1 (https=)
PH (1) PH12020551591A1 (https=)
PL (2) PL4122954T3 (https=)
PT (2) PT4122954T (https=)
RS (2) RS65639B1 (https=)
SG (1) SG11202009467YA (https=)
SI (2) SI3774862T1 (https=)
SM (2) SMT202400241T1 (https=)
UA (1) UA128210C2 (https=)
WO (1) WO2019193576A1 (https=)
ZA (1) ZA202306729B (https=)

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WO2020180534A1 (en) 2019-03-01 2020-09-10 President And Fellows Of Harvard College Methods and compositions for protein delivery
TW202216746A (zh) * 2020-06-22 2022-05-01 印度商太陽製藥工業有限公司 長效型ｇｌｐ－１／ｇｉｐ雙重促效劑
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CN114685646B (zh) * 2020-12-31 2023-04-07 厦门赛诺邦格生物科技股份有限公司 一种多肽侧链类似物的制备方法及其应用
CA3204051A1 (en) 2021-01-20 2022-07-28 Brian Lian Compositions and methods for the treatment of metabolic and liver disorders
JP7642830B2 (ja) 2021-09-15 2025-03-10 バイキング・セラピューティクス・インコーポレイテッド 代謝及び肝臓障害の処置のための組成物及び方法
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Also Published As

Publication number Publication date
RS65639B1 (sr) 2024-07-31
JOP20200251A1 (ar) 2020-10-04
BR112020020419A2 (pt) 2021-01-19
CN112236444A (zh) 2021-01-15
EP3774862A1 (en) 2021-02-17
JP2023078367A (ja) 2023-06-06
PT3774862T (pt) 2022-09-05
SMT202200352T1 (it) 2022-09-14
EP4122954B1 (en) 2024-04-03
RS63523B1 (sr) 2022-09-30
PT4122954T (pt) 2024-06-05
CN120554480A (zh) 2025-08-29
US20220402992A1 (en) 2022-12-22
ZA202306729B (en) 2024-03-27
CL2020002574A1 (es) 2021-06-04
US20240199718A1 (en) 2024-06-20
US11866477B2 (en) 2024-01-09
AU2019247936B2 (en) 2023-03-02
MY202560A (en) 2024-05-08
SG11202009467YA (en) 2020-10-29
SI4122954T1 (sl) 2024-07-31
AU2023203430B2 (en) 2025-07-03
KR20200141469A (ko) 2020-12-18
JP2021520346A (ja) 2021-08-19
US20240376175A1 (en) 2024-11-14
US20200362007A1 (en) 2020-11-19
AU2019247936C1 (en) 2023-06-15
KR20250065720A (ko) 2025-05-13
EP4122954A1 (en) 2023-01-25
KR102801994B1 (ko) 2025-04-30
CN117964735A (zh) 2024-05-03
CN112236444B (zh) 2025-09-19
PH12020551591A1 (en) 2021-08-16
HUE067499T2 (hu) 2024-10-28
FI4122954T3 (fi) 2024-06-18
IL277483B1 (en) 2026-01-01
US11447535B2 (en) 2022-09-20
WO2019193576A1 (en) 2019-10-10
PL4122954T3 (pl) 2024-08-12
MX2020010505A (es) 2021-01-15
CO2020012425A2 (es) 2020-12-21
JP7250814B2 (ja) 2023-04-03
ES2980707T3 (es) 2024-10-02
JOP20200251B1 (ar) 2024-04-18
IL277483A (en) 2020-11-30
HRP20240749T1 (hr) 2024-09-13
NZ768446A (en) 2025-10-31
AU2023203430A1 (en) 2023-06-29
EP3774862B1 (en) 2022-06-08
CA3095988A1 (en) 2019-10-10
LT3774862T (lt) 2022-09-12
DK4122954T3 (da) 2024-06-10
AU2019247936A1 (en) 2020-10-15
MX2024007688A (es) 2024-07-09
SI3774862T1 (sl) 2022-10-28
US11242373B2 (en) 2022-02-08
ES2925678T3 (es) 2022-10-19
PL3774862T3 (pl) 2022-10-03
PE20211417A1 (es) 2021-08-02
AU2025242190A1 (en) 2025-10-23
ECSP20070185A (es) 2021-01-29
CY1125528T1 (el) 2026-02-25
US11873328B2 (en) 2024-01-16
US12421289B2 (en) 2025-09-23
EP4364751A2 (en) 2024-05-08
LT4122954T (lt) 2024-06-25
US11485766B2 (en) 2022-11-01
US20190309040A1 (en) 2019-10-10
US20210206823A1 (en) 2021-07-08
SMT202400241T1 (it) 2024-07-09
HRP20221054T1 (hr) 2022-11-11
HUE060135T2 (hu) 2023-02-28
DK3774862T3 (da) 2022-09-05
US20220402991A1 (en) 2022-12-22
EP4364751A3 (en) 2024-06-26

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