TWI410406B - 吡咯烷化合物 - Google Patents

吡咯烷化合物 Download PDF

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Publication number
TWI410406B
TWI410406B TW095116220A TW95116220A TWI410406B TW I410406 B TWI410406 B TW I410406B TW 095116220 A TW095116220 A TW 095116220A TW 95116220 A TW95116220 A TW 95116220A TW I410406 B TWI410406 B TW I410406B
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TW
Taiwan
Prior art keywords
group
alkyl
phenyl
pyrrolidin
fluorophenyl
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TW095116220A
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English (en)
Chinese (zh)
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TW200720249A (en
Inventor
Muneaki Kurimura
Shinichi Taira
Takahiro Tomoyasu
Nobuaki Ito
Kuninori Tai
Noriaki Takemura
Takayuki Matsuzaki
Yasuhiro Menjo
Shin Miyamura
Yohji Sakurai
Akihito Watanabe
Yasuyo Sakata
Takumi Masumoto
Kohei Akazawa
Haruhiko Sugino
Naoki Amada
Satoshi Ohashi
Tomoichi Shinohara
Hirofumi Sasaki
Chisako Morita
Junko Yamashita
Satoko Nakajima
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Otsuka Pharma Co Ltd
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Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of TW200720249A publication Critical patent/TW200720249A/zh
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Publication of TWI410406B publication Critical patent/TWI410406B/zh

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  • Life Sciences & Earth Sciences (AREA)
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  • Diabetes (AREA)
  • Psychiatry (AREA)
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  • Psychology (AREA)
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  • Child & Adolescent Psychology (AREA)
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TW095116220A 2005-05-13 2006-05-08 吡咯烷化合物 TWI410406B (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2005141230 2005-05-13

Publications (2)

Publication Number Publication Date
TW200720249A TW200720249A (en) 2007-06-01
TWI410406B true TWI410406B (zh) 2013-10-01

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Family Applications (3)

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TW095116220A TWI410406B (zh) 2005-05-13 2006-05-08 吡咯烷化合物
TW102143870A TWI449692B (zh) 2005-05-13 2006-05-08 吡咯烷化合物(三)
TW102101997A TWI439452B (zh) 2005-05-13 2006-05-08 吡咯烷化合物(二)

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TW102143870A TWI449692B (zh) 2005-05-13 2006-05-08 吡咯烷化合物(三)
TW102101997A TWI439452B (zh) 2005-05-13 2006-05-08 吡咯烷化合物(二)

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US (6) US8084442B2 (enExample)
EP (2) EP1881975B8 (enExample)
JP (1) JP4776631B2 (enExample)
KR (2) KR20100038453A (enExample)
CN (3) CN103613527B (enExample)
AR (1) AR054191A1 (enExample)
AU (2) AU2006244851B2 (enExample)
BR (1) BRPI0610279A2 (enExample)
CA (1) CA2608184C (enExample)
CY (1) CY1114767T1 (enExample)
DK (1) DK2407451T3 (enExample)
ES (2) ES2446375T3 (enExample)
IL (1) IL187311A (enExample)
IN (1) IN2012DN00758A (enExample)
MX (1) MX2007014252A (enExample)
MY (1) MY148653A (enExample)
PL (1) PL2407451T3 (enExample)
PT (1) PT2407451E (enExample)
RU (1) RU2414454C2 (enExample)
SG (1) SG162722A1 (enExample)
SI (1) SI2407451T1 (enExample)
TW (3) TWI410406B (enExample)
WO (1) WO2006121218A1 (enExample)
ZA (1) ZA200709691B (enExample)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2507501C (en) 2002-11-27 2011-10-04 Incyte Corporation 3-aminopyrrolidine derivatives as modulators of chemokine receptors
TWI410406B (zh) 2005-05-13 2013-10-01 Otsuka Pharma Co Ltd 吡咯烷化合物
EP1954133A4 (en) * 2005-11-30 2010-11-24 Glaxosmithkline Llc PYRROLIDINANILINE
EP1960355A1 (en) * 2005-11-30 2008-08-27 F.Hoffmann-La Roche Ag 3-amino-1-arylpropyl indoles and aza-substituted indoles
JP5219465B2 (ja) * 2006-11-10 2013-06-26 大塚製薬株式会社 医薬
ATE522519T1 (de) * 2008-03-20 2011-09-15 Hoffmann La Roche Pyrrolidinylderivate und anwendungen davon
JP5827627B2 (ja) * 2009-11-07 2015-12-02 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングMerck Patent Gesellschaft mit beschraenkter Haftung TGF−β受容体キナーゼ阻害剤としてのヘテロアリールアミノキノリン
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