TWI389878B - 新穎化合物，其製備及用途 - Google Patents

新穎化合物，其製備及用途 Download PDF

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Publication number
TWI389878B
TWI389878B TW095148358A TW95148358A TWI389878B TW I389878 B TWI389878 B TW I389878B TW 095148358 A TW095148358 A TW 095148358A TW 95148358 A TW95148358 A TW 95148358A TW I389878 B TWI389878 B TW I389878B
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Taiwan
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compound
alkyl
phenyl
group
methyl
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TW095148358A
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English (en)
Chinese (zh)
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TW200745004A (en
Inventor
Per Sauerberg
Pavel Pihera
Miroslav Havranek
Ingrid Pettersson
John Patrick Mogensen
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High Point Pharmaceuticals Llc
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    • C07C69/66—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety
    • C07C69/73—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of unsaturated acids
    • C07C69/734—Ethers
    • C07C69/736—Ethers the hydroxy group of the ester being etherified with a hydroxy compound having the hydroxy group bound to a carbon atom of a six-membered aromatic ring
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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