TWI275591B - Opiod and opioid-like coumpounds and uses thereof - Google Patents
Opiod and opioid-like coumpounds and uses thereof Download PDFInfo
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- TWI275591B TWI275591B TWOPIOIDANA TW92132155A TWI275591B TW I275591 B TWI275591 B TW I275591B TW OPIOIDAN A TWOPIOIDAN A TW OPIOIDANA TW 92132155 A TW92132155 A TW 92132155A TW I275591 B TWI275591 B TW I275591B
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Classifications
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
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Landscapes
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- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Plural Heterocyclic Compounds (AREA)
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| JP2521914Y2 (ja) | 1988-12-23 | 1997-01-08 | エヌティエヌ株式会社 | 大型転がり軸受 |
| US7923454B2 (en) * | 2002-05-17 | 2011-04-12 | Jenken Biosciences, Inc. | Opioid and opioid-like compounds and uses thereof |
| US20040204862A1 (en) | 2003-04-11 | 2004-10-14 | Wainer Irving W. | Computer-based model for identification and characterization for non-competitive inhibitors of nicotinic acetylcholine receptors and related ligand-gated ion channel receptors |
| AU2005244852B2 (en) * | 2004-05-12 | 2011-09-22 | The Government Of The United States Of America, As Represented By The Secretary, Department Of Health And Human Services | Methods related to the treatment of neurodegenerative and inflammatory conditions |
| AU2005244401B2 (en) | 2004-05-14 | 2009-01-22 | Green Cross Corp. | Neuroprotective properties of dextrorotatory morphinans |
| SA07280459B1 (ar) * | 2006-08-25 | 2011-07-20 | بيورديو فارما إل. بي. | أشكال جرعة صيدلانية للتناول عن طريق الفم مقاومة للعبث تشتمل على مسكن شبه أفيوني |
| PT2357183E (pt) | 2007-05-01 | 2015-09-28 | Concert Pharmaceuticals Inc | Compostos de morfinano |
| US8329897B2 (en) | 2007-07-26 | 2012-12-11 | Vitae Pharmaceuticals, Inc. | Synthesis of inhibitors of 11β-hydroxysteroid dehydrogenase type 1 |
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| CA2704628C (en) | 2007-11-16 | 2016-11-29 | Boehringer Ingelheim International Gmbh | Aryl- and heteroarylcarbonyl derivatives of benzomorphanes and related scaffolds, medicaments containing such compounds and their use |
| PL2596784T3 (pl) * | 2007-11-23 | 2017-06-30 | Grünenthal GmbH | Kompozycje tapentadolu |
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| TW200934490A (en) | 2008-01-07 | 2009-08-16 | Vitae Pharmaceuticals Inc | Lactam inhibitors of 11 &abgr;-hydroxysteroid dehydrogenase 1 |
| JP5490020B2 (ja) | 2008-01-24 | 2014-05-14 | ヴァイティー ファーマシューティカルズ,インコーポレイテッド | 11β−ヒドロキシステロイドデヒドロゲナーゼ1の環状カルバゼート及びセミカルバジドインヒビター |
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| CA2723034A1 (en) | 2008-05-01 | 2009-11-05 | Vitae Pharmaceuticals, Inc. | Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1 |
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| JP5379160B2 (ja) | 2008-07-25 | 2013-12-25 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 11β−ヒドロキシステロイドデヒドロゲナーゼ1の環状インヒビター |
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| MA33216B1 (fr) | 2009-04-30 | 2012-04-02 | Boehringer Ingelheim Int | Inhibiteurs cycliques de la 11béta-hydroxysteroïde déshydrogénase 1 |
| JP5656986B2 (ja) | 2009-06-11 | 2015-01-21 | ヴァイティー ファーマシューティカルズ,インコーポレイテッド | 1,3−オキサジナン−2−オン構造に基づく11β−ヒドロキシステロイドデヒドロゲナーゼ1の環状阻害剤 |
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| TWI531571B (zh) | 2009-11-06 | 2016-05-01 | 維它藥物公司 | 六氫茚并吡啶及八氫苯并喹啉之芳基-及雜芳基羰基衍生物 |
| AU2011250485B2 (en) * | 2010-05-03 | 2016-07-07 | Tsh Biopharm Corporation, Limited | Pharmaceutical composition and method for treating hypertension |
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| JP5813106B2 (ja) | 2010-06-25 | 2015-11-17 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 代謝障害の処置のための11−β−HSD1のインヒビターとしてのアザスピロヘキサノン |
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| TWI537258B (zh) | 2010-11-05 | 2016-06-11 | 百靈佳殷格翰國際股份有限公司 | 六氫茚并吡啶及八氫苯并喹啉之芳基-及雜環芳基羰基衍生物 |
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| JP6248711B2 (ja) | 2014-03-06 | 2017-12-20 | 株式会社デンソー | 回転電機の固定子 |
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| RU2717677C1 (ru) | 2016-04-22 | 2020-03-25 | Тайваньж Фармасьютикалс Со., Лтд. | Налмефен, налтрексон или их производные для применения в лечении (не)алкогольного стеатогепатита или неалкогольной жировой болезни печени |
| CN110290792A (zh) * | 2017-01-05 | 2019-09-27 | 景凯生物科技股份有限公司 | 吗啡喃衍生物和其用于治疗自体免疫、发炎或感染相关的障碍的组合物 |
| CN107157998A (zh) * | 2017-05-26 | 2017-09-15 | 张灏 | 右美沙芬的新用途 |
| WO2020172248A1 (en) * | 2019-02-19 | 2020-08-27 | Robert Barsotti | Solutions and methods for organ preservation |
| CN119977886B (zh) * | 2025-02-13 | 2025-08-22 | 安徽益普克医药科技发展有限公司 | 一种葡萄糖酸喷他佐辛苯甲酸酯及其制备方法与用途 |
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| AUPQ968300A0 (en) * | 2000-08-25 | 2000-09-21 | Glaxo Wellcome Australia Ltd | Chemical methods |
| DE60109960T2 (de) * | 2000-10-31 | 2006-02-16 | Rensselaer Polytechnic Institute | 8-substituierte 2,6-methano-3-benzazocine und 3-substituierte morphinane als opioidrezeptorbindende agenzien |
| US20030144312A1 (en) * | 2001-10-30 | 2003-07-31 | Schoenhard Grant L. | Inhibitors of ABC drug transporters in multidrug resistant cancer cells |
-
2003
- 2003-05-16 MX MXPA04011327A patent/MXPA04011327A/es not_active Application Discontinuation
- 2003-05-16 CN CN201310094981.6A patent/CN103405431B/zh not_active Expired - Lifetime
- 2003-05-16 CN CN038112396A patent/CN1653050B/zh not_active Expired - Lifetime
- 2003-05-16 JP JP2004505341A patent/JP5438250B2/ja not_active Expired - Fee Related
- 2003-05-16 CA CA2486157A patent/CA2486157C/en not_active Expired - Fee Related
- 2003-05-16 AU AU2003234621A patent/AU2003234621A1/en not_active Abandoned
- 2003-05-16 WO PCT/US2003/015461 patent/WO2003097608A2/en not_active Ceased
- 2003-05-16 EP EP03728964.2A patent/EP1506174B1/en not_active Expired - Lifetime
- 2003-05-16 EP EP15186541.7A patent/EP2987788A1/en not_active Withdrawn
- 2003-11-17 TW TWOPIOIDANA patent/TWI275591B/zh not_active IP Right Cessation
-
2010
- 2010-08-24 AU AU2010212517A patent/AU2010212517A1/en not_active Abandoned
-
2013
- 2013-11-01 JP JP2013228118A patent/JP6165592B2/ja not_active Expired - Fee Related
-
2015
- 2015-04-24 JP JP2015089558A patent/JP6193298B2/ja not_active Expired - Lifetime
-
2016
- 2016-07-18 HK HK16108452.6A patent/HK1220452A1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP2987788A1 (en) | 2016-02-24 |
| MXPA04011327A (es) | 2005-08-15 |
| EP1506174A2 (en) | 2005-02-16 |
| WO2003097608A3 (en) | 2004-03-18 |
| EP1506174B1 (en) | 2015-09-30 |
| JP6165592B2 (ja) | 2017-07-19 |
| JP2015155449A (ja) | 2015-08-27 |
| CN1653050A (zh) | 2005-08-10 |
| HK1220452A1 (en) | 2017-06-09 |
| JP2005530798A (ja) | 2005-10-13 |
| AU2003234621A1 (en) | 2003-12-02 |
| CA2486157C (en) | 2013-04-16 |
| JP2014043452A (ja) | 2014-03-13 |
| CN103405431B (zh) | 2016-04-13 |
| CN1653050B (zh) | 2013-04-24 |
| CA2486157A1 (en) | 2003-11-27 |
| TW200427690A (en) | 2004-12-16 |
| AU2010212517A1 (en) | 2010-09-16 |
| WO2003097608A2 (en) | 2003-11-27 |
| JP5438250B2 (ja) | 2014-03-12 |
| CN103405431A (zh) | 2013-11-27 |
| HK1192711A1 (zh) | 2014-08-29 |
| JP6193298B2 (ja) | 2017-09-06 |
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| MM4A | Annulment or lapse of patent due to non-payment of fees |