TW307769B - - Google Patents

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Publication number
TW307769B
TW307769B TW082105942A TW82105942A TW307769B TW 307769 B TW307769 B TW 307769B TW 082105942 A TW082105942 A TW 082105942A TW 82105942 A TW82105942 A TW 82105942A TW 307769 B TW307769 B TW 307769B
Authority
TW
Taiwan
Prior art keywords
hydrochloride
patent application
water
crystalline hydrate
hydrate
Prior art date
Application number
TW082105942A
Other languages
English (en)
Chinese (zh)
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co filed Critical Shionogi & Co
Application granted granted Critical
Publication of TW307769B publication Critical patent/TW307769B/zh

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
TW082105942A 1992-07-31 1993-07-26 TW307769B (cg-RX-API-DMAC7.html)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP20496592 1992-07-31

Publications (1)

Publication Number Publication Date
TW307769B true TW307769B (cg-RX-API-DMAC7.html) 1997-06-11

Family

ID=16499234

Family Applications (1)

Application Number Title Priority Date Filing Date
TW082105942A TW307769B (cg-RX-API-DMAC7.html) 1992-07-31 1993-07-26

Country Status (23)

Country Link
US (1) US5407929A (cg-RX-API-DMAC7.html)
EP (1) EP0581552B1 (cg-RX-API-DMAC7.html)
KR (1) KR100245938B1 (cg-RX-API-DMAC7.html)
CN (1) CN1037683C (cg-RX-API-DMAC7.html)
AT (1) ATE165360T1 (cg-RX-API-DMAC7.html)
AU (1) AU657866B2 (cg-RX-API-DMAC7.html)
BR (1) BR9303235A (cg-RX-API-DMAC7.html)
CA (1) CA2101502A1 (cg-RX-API-DMAC7.html)
DE (1) DE69318077T2 (cg-RX-API-DMAC7.html)
ES (1) ES2115725T3 (cg-RX-API-DMAC7.html)
FI (1) FI933391A7 (cg-RX-API-DMAC7.html)
GR (1) GR3026699T3 (cg-RX-API-DMAC7.html)
HU (1) HU219637B (cg-RX-API-DMAC7.html)
IL (1) IL106516A (cg-RX-API-DMAC7.html)
MX (1) MX9304611A (cg-RX-API-DMAC7.html)
NO (1) NO303734B1 (cg-RX-API-DMAC7.html)
NZ (1) NZ248285A (cg-RX-API-DMAC7.html)
PH (1) PH30109A (cg-RX-API-DMAC7.html)
PL (2) PL172830B1 (cg-RX-API-DMAC7.html)
RU (1) RU2118959C1 (cg-RX-API-DMAC7.html)
TW (1) TW307769B (cg-RX-API-DMAC7.html)
UA (1) UA37181C2 (cg-RX-API-DMAC7.html)
ZA (1) ZA935529B (cg-RX-API-DMAC7.html)

Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA03007349A (es) * 2001-02-24 2003-12-04 Boehringer Ingelheim Pharma Derivados de xantina, su preparacion y su empleo como medicamentos.
AT413282B (de) * 2002-02-01 2006-01-15 Sandoz Ag Kristalline salze der 7-(((5-amino-1,2,4-thiadiazol-3-yl) (fluoromethoxy-imino)acetyl)amino)-3- ((imino-1-piperazinylmethyl)
KR20030076759A (ko) * 2002-03-21 2003-09-29 주식회사 엘지생명과학 신규 세팔로스포린 화합물 및 그의 제조 방법
US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US6727277B1 (en) 2002-11-12 2004-04-27 Kansas State University Research Foundation Compounds affecting cholesterol absorption
CN101219992B (zh) 2003-02-12 2011-08-31 日产化学工业株式会社 匹伐他汀钙的晶形
BRPI0408716B1 (pt) 2003-03-27 2017-08-29 Basilea Pharmaceutica Ag. Cefalosporin in crystalline form, process for its preparation and its uses, and preparation of cephalosporin
US7501426B2 (en) * 2004-02-18 2009-03-10 Boehringer Ingelheim International Gmbh 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
DE102004054054A1 (de) * 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
DE102005035891A1 (de) * 2005-07-30 2007-02-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
EP1852108A1 (en) 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG DPP IV inhibitor formulations
PE20080251A1 (es) * 2006-05-04 2008-04-25 Boehringer Ingelheim Int Usos de inhibidores de dpp iv
NZ600394A (en) 2006-05-04 2014-04-30 Boehringer Ingelheim Int Polymorphs of a dpp-iv enzyme inhibitor
ES2733348T3 (es) * 2007-08-17 2019-11-28 Boehringer Ingelheim Int Derivados de purina para uso en el tratamiento de enfermedades relacionadas con FAP
AR071175A1 (es) 2008-04-03 2010-06-02 Boehringer Ingelheim Int Composicion farmaceutica que comprende un inhibidor de la dipeptidil-peptidasa-4 (dpp4) y un farmaco acompanante
PE20100156A1 (es) * 2008-06-03 2010-02-23 Boehringer Ingelheim Int Tratamiento de nafld
KR20190016601A (ko) 2008-08-06 2019-02-18 베링거 인겔하임 인터내셔날 게엠베하 메트포르민 요법이 부적합한 환자에서의 당뇨병 치료
UY32030A (es) 2008-08-06 2010-03-26 Boehringer Ingelheim Int "tratamiento para diabetes en pacientes inapropiados para terapia con metformina"
CA2735562C (en) * 2008-08-15 2017-10-17 Boehringer Ingelheim International Gmbh Dpp-4 inhibitors for wound healing
MX2011002558A (es) 2008-09-10 2011-04-26 Boehringer Ingelheim Int Terapia de combinacion para el tratamiento de diabetes y estados relacionados.
US20200155558A1 (en) 2018-11-20 2020-05-21 Boehringer Ingelheim International Gmbh Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug
CA2745037C (en) 2008-12-23 2020-06-23 Boehringer Ingelheim International Gmbh Salt forms of 1-[(4-methyl-quinazolin-2-yl)methyl]-3-methyl-7-(2-butyn-1-yl)-8(3-(r)-amino-piperidin-1-yl)-xanthine
AR074990A1 (es) 2009-01-07 2011-03-02 Boehringer Ingelheim Int Tratamiento de diabetes en pacientes con un control glucemico inadecuado a pesar de la terapia con metformina
CN102753161A (zh) 2009-11-27 2012-10-24 贝林格尔.英格海姆国际有限公司 基因型糖尿病患者利用dpp-iv抑制剂例如利拉利汀的治疗
CN107961377B (zh) 2010-05-05 2022-11-22 勃林格殷格翰国际有限公司 组合疗法
MX2012014247A (es) 2010-06-24 2013-01-18 Boehringer Ingelheim Int Terapia para la diabetes.
AR083878A1 (es) 2010-11-15 2013-03-27 Boehringer Ingelheim Int Terapia antidiabetica vasoprotectora y cardioprotectora, linagliptina, metodo de tratamiento
PL2731947T3 (pl) 2011-07-15 2019-07-31 Boehringer Ingelheim International Gmbh Podstawiona dimeryczna pochodna chinazoliny, sposób jej wytwarzania i jej zastosowanie w kompozycjach farmaceutycznych do leczenia cukrzycy typu I i II
US9555001B2 (en) 2012-03-07 2017-01-31 Boehringer Ingelheim International Gmbh Pharmaceutical composition and uses thereof
US20130303462A1 (en) 2012-05-14 2013-11-14 Boehringer Ingelheim International Gmbh Use of a dpp-4 inhibitor in podocytes related disorders and/or nephrotic syndrome
US20130303554A1 (en) 2012-05-14 2013-11-14 Boehringer Ingelheim International Gmbh Use of a dpp-4 inhibitor in sirs and/or sepsis
WO2013174767A1 (en) 2012-05-24 2013-11-28 Boehringer Ingelheim International Gmbh A xanthine derivative as dpp -4 inhibitor for use in modifying food intake and regulating food preference
WO2015128453A1 (en) 2014-02-28 2015-09-03 Boehringer Ingelheim International Gmbh Medical use of a dpp-4 inhibitor
CA3022202A1 (en) 2016-06-10 2017-12-14 Boehringer Ingelheim International Gmbh Combinations of linagliptin and metformin

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES475573A1 (es) * 1977-07-12 1980-01-16 Fujisawa Pharmaceutical Co Un procedimiento para preparar nuevos compuestos de cefem
IE65926B1 (en) * 1990-07-19 1995-11-29 Shionogi & Co Thioalkylthio cephalosporin derivatives

Also Published As

Publication number Publication date
MX9304611A (es) 1994-02-28
CN1037683C (zh) 1998-03-11
FI933391L (fi) 1994-02-01
KR100245938B1 (ko) 2000-04-01
CA2101502A1 (en) 1994-02-01
DE69318077T2 (de) 1998-10-29
HUT68602A (en) 1995-06-28
EP0581552A2 (en) 1994-02-02
CN1089948A (zh) 1994-07-27
PL172830B1 (pl) 1997-12-31
EP0581552B1 (en) 1998-04-22
IL106516A0 (en) 1993-11-15
ZA935529B (en) 1994-02-24
PL299870A1 (en) 1994-02-07
DE69318077D1 (de) 1998-05-28
FI933391A7 (fi) 1994-02-01
ES2115725T3 (es) 1998-07-01
AU657866B2 (en) 1995-03-23
PH30109A (en) 1996-12-27
UA37181C2 (uk) 2001-05-15
NZ248285A (en) 1994-07-26
NO932745D0 (no) 1993-07-30
AU4422793A (en) 1994-02-03
FI933391A0 (fi) 1993-07-29
IL106516A (en) 1998-06-15
US5407929A (en) 1995-04-18
RU2118959C1 (ru) 1998-09-20
ATE165360T1 (de) 1998-05-15
HU9302194D0 (en) 1993-10-28
NO303734B1 (no) 1998-08-24
NO932745L (no) 1994-02-01
KR940005636A (ko) 1994-03-22
EP0581552A3 (en) 1994-06-01
HU219637B (hu) 2001-06-28
PL172835B1 (pl) 1997-12-31
GR3026699T3 (en) 1998-07-31
BR9303235A (pt) 1994-03-01

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